| Compound ID |
Compound Name |
Compound Formula |
|
CP0058361
|
CHEMBL3774855
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|
C28H39N5O2
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
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CP0414833
|
3-[4-cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C24H34N4O
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
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CP0459830
|
(1S,2S,4S)-2-[4-cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)-4-hydroxycyclopentane-1-carboxamide
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|
C27H38N4O2
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
|
CP0458491
|
3-[4-cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C24H34N4O
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
|
CP0551795
|
3-[4-cyclopropyl-5-[5-(2-methylpropyl)-1,2-oxazol-3-yl]-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C23H29N5O2
|
1
|
| 1 |
EC50 = 54 nM
|
|
|
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CP0414832
|
3-[4-cyclopropyl-5-[4-(2-methylpropyl)phenyl]-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C26H32N4O
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
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CP0559971
|
(3R,4S)-4-[4-cyclopropyl-5-[3-(2-methylpropyl)cyclobutyl]-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)-1-methylpiperidine-3-carboxamide
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|
C28H41N5O
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0555703
|
3-[5-(2-cyclohexylethyl)-4-ethyl-1,2,4-triazol-3-yl]-N-naphthalen-1-ylpropanamide
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|
C25H32N4O
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0414830
|
3-[5-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,2,4-triazol-3-yl]-N-naphthalen-1-ylpropanamide
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|
C26H26N4O
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
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CP0551794
|
3-[5-(2-cyclohexylethyl)-4-cyclopropyl-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C24H34N4O
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0397886
|
3-[5-(2-cyclohexylethyl)-4-(2,2-difluorocyclopropyl)-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C24H32F2N4O
|
1
|
| 1 |
EC50 = 500 nM
|
|
|
|
CP0181318
|
3-[5-(2-cyclohexylethyl)-4-ethyl-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C23H34N4O
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0542045
|
3-[4-cyclopropyl-5-(4-methylpentyl)-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C22H32N4O
|
1
|
| 1 |
EC50 = 610 nM
|
|
|
|
CP0414834
|
3-[4-ethyl-5-(2-phenylethyl)-1,2,4-triazol-3-yl]-N-naphthalen-1-ylpropanamide
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|
C25H26N4O
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
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CP0381787
|
N-(3-chloro-2-methylphenyl)-3-[5-(2-cyclohexylethyl)-4-ethyl-1,2,4-triazol-3-yl]propanamide
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|
C22H31ClN4O
|
1
|
| 1 |
EC50 = 640 nM
|
|
|
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CP0455009
|
3-[5-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,2,4-triazol-3-yl]-2-methyl-N-naphthalen-1-ylpropanamide
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|
C27H28N4O
|
1
|
| 1 |
EC50 = 670 nM
|
|
|
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CP0360184
|
2-[[5-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-naphthalen-1-ylacetamide
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|
C25H24N4OS
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0555704
|
3-[5-(3,3-dimethylbutyl)-4-ethyl-1,2,4-triazol-3-yl]-N-naphthalen-1-ylpropanamide
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|
C23H30N4O
|
1
|
| 1 |
EC50 = 830 nM
|
|
|
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CP0555702
|
3-[5-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,2,4-triazol-3-yl]-N-naphthalen-1-ylbutanamide
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|
C27H28N4O
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
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CP0414831
|
3-[4-cyclopropyl-5-(4,4-dimethylpentyl)-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C23H34N4O
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
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CP0375785
|
3-[4-ethyl-5-(3-methylbutyl)-1,2,4-triazol-3-yl]-N-naphthalen-1-ylpropanamide
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|
C22H28N4O
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
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CP0375786
|
3-[4-cyclopropyl-5-(3-methylpentyl)-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C22H32N4O
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
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CP0375787
|
3-[4-cyclobutyl-5-(2-cyclohexylethyl)-1,2,4-triazol-3-yl]-N-(2,4-dimethylphenyl)propanamide
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|
C25H36N4O
|
1
|
| 1 |
EC50 = 1800 nM
|
|
|
|
CP0397884
|
3-[5-(cyclohexylmethyl)-4-ethyl-1,2,4-triazol-3-yl]-N-naphthalen-1-ylpropanamide
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|
C24H30N4O
|
1
|
| 1 |
EC50 = 2600 nM
|
|
|
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CP0381794
|
3-[5-(2-cyclohexylethyl)-4-ethyl-1,2,4-triazol-3-yl]-N-(3,5-dimethylphenyl)propanamide
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|
C23H34N4O
|
1
|
| 1 |
EC50 = 3100 nM
|
|
|
|
CP0561097
|
3-(5-cyclohexyl-4-ethyl-1,2,4-triazol-3-yl)-N-naphthalen-1-ylpropanamide
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|
C23H28N4O
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
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CP0414829
|
2-[[5-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,2,4-triazol-3-yl]oxy]-N-naphthalen-1-ylacetamide
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|
C25H24N4O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0474191
|
3-[5-(2,3-dihydro-1H-inden-2-yl)-4-ethyl-1,2,4-triazol-3-yl]-3-hydroxy-N-naphthalen-1-ylpropanamide
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|
C26H26N4O2
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
