| Compound ID |
Compound Name |
Compound Formula |
|
CP0377831
|
5-amino-N-tert-butyl-2-(methylthio)-4-(3-(2-oxo-2-(prop-2-ynylamino)ethylamino)phenyl)thieno[2,3-d]pyrimidine-6-carboxamide
Show/Hide
|
C23H26N6O2S2
|
1
|
| 1 |
EC50 = 126 nM
|
|
|
|
CP0380316
|
5-amino-4-(3-(2-((1-(2-(2-(2-azidoethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)methylamino)-2-oxoethylamino)phenyl)-N-tert-butyl-2-(methylthio)thieno[2,3-d]pyrimidine-6-carboxamide
Show/Hide
|
C29H38N12O4S2
|
1
|
| 1 |
EC50 = 397 nM
|
|
|
|
CP0391883
|
1-(6-amino-2,2,4-trimethyl-4-phenyl-3H-quinolin-1-yl)ethanone
Show/Hide
|
C20H24N2O
|
1
|
| 1 |
EC50 = 4400 nM
|
|
|
|
CP0538708
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-4-propylbenzamide
Show/Hide
|
C30H34N2O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0559356
|
N-(1-acetyl-2,2,4,7-tetramethyl-4-phenyl-3H-quinolin-6-yl)-4-phenylbenzamide
Show/Hide
|
C34H34N2O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0500515
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-4-(trifluoromethyl)benzamide
Show/Hide
|
C28H27F3N2O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0518113
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-phenylbenzamide
Show/Hide
|
C33H32N2O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0435511
|
Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimethyl-4-phenyl-1,2,3,4-tetrahydro-quinolin-6-yl)-amide
Show/Hide
|
C33H32N2O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0378099
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-2-phenylbenzamide
Show/Hide
|
C33H32N2O2
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0542108
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)furan-2-carboxamide
Show/Hide
|
C25H26N2O3
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0374398
|
N-(1-acetyl-8-methoxy-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-4-phenylbenzamide
Show/Hide
|
C34H34N2O3
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0378864
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-4-chlorobenzamide
Show/Hide
|
C27H27ClN2O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0380315
|
(R)-N-(1-acetyl-2,2,4-trimethyl-4-(4-(prop-2-ynyloxy)phenyl)-1,2,3,4-tetrahydroquinolin-6-yl)biphenyl-4-carboxamide
Show/Hide
|
C36H34N2O3
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0408617
|
N-[1-acetyl-2,2,4-trimethyl-4-(4-methylphenyl)-3H-quinolin-6-yl]-4-phenylbenzamide
Show/Hide
|
C34H34N2O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0451717
|
(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl) 4-phenylbenzoate
Show/Hide
|
C33H31NO3
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0538697
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-2-[(2-methylpropan-2-yl)oxy]acetamide
Show/Hide
|
C26H34N2O3
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0408618
|
1-[2,2,4-trimethyl-4-phenyl-6-[(4-phenylphenyl)methoxy]-3H-quinolin-1-yl]ethanone
Show/Hide
|
C33H33NO2
|
1
|
| 1 |
IC50 = 166 nM
|
|
|
|
CP0455572
|
N-[1-acetyl-4-(2-methoxyphenyl)-2,2,4-trimethyl-3H-quinolin-6-yl]-4-phenylbenzamide
Show/Hide
|
C34H34N2O3
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0559355
|
N-[1-acetyl-4-(4-hydroxyphenyl)-2,2,4-trimethyl-3H-quinolin-6-yl]-4-phenylbenzamide
Show/Hide
|
C33H32N2O3
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0393745
|
(R)-N-(1-acetyl-4-(4-((1-(2-(2-(2-azidoethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)methoxy)phenyl)-2,2,4-trimethyl-1,2,3,4-tetrahydroquinolin-6-yl)biphenyl-4-carboxamide
Show/Hide
|
C42H46N8O5
|
1
|
| 1 |
IC50 = 324 nM
|
|
|
|
CP0554570
|
1-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-3-phenylurea
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
|
CP0377834
|
(R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphenyl-4-ylcarboxamido-2,2,4-trimethyl-1,2,3,4-tetrahydroquinolin-4-yl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)ethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)methylamino)-2-oxoethylamino)phenyl)-5-amino-N-tert-butyl-2-(methylthio)thieno[2,3-d]pyrimidine-6-carboxamide
Show/Hide
|
C65H72N14O7S2
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0511876
|
1-[6-[(4-tert-butylphenyl)methylamino]-2,2,4-trimethyl-4-phenyl-3H-quinolin-1-yl]ethanone
Show/Hide
|
C31H38N2O
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0393737
|
(R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-ylcarboxamido-2,2,4-trimethyl-1,2,3,4-tetrahydroquinolin-4-yl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)-3,6,9,12-tetraoxatetradecyl)-1H-1,2,3-triazol-4-yl)methylamino)-2-oxoethylamino)phenyl)-5-amino-N-tert-butyl-2-(methylthio)thieno[2,3-d]pyrimidine-6-carboxamide
Show/Hide
|
C69H80N14O9S2
|
1
|
| 1 |
IC50 = 1023 nM
|
|
|
|
CP0377830
|
(R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-biphenyl-4-ylcarboxamido-2,2,4-trimethyl-1,2,3,4-tetrahydroquinolin-4-yl)phenoxy)methyl)-1H-1,2,3-triazol-1-yl)ethoxy)ethoxy)ethoxy)ethyl)-1H-1,2,3-triazol-4-yl)methylamino)-2-oxoethylamino)phenyl)-5-amino-N-tert-butyl-2-(methylthio)thieno[2,3-d]pyrimidine-6-carboxamide
Show/Hide
|
C67H76N14O8S2
|
1
|
| 1 |
IC50 = 1662 nM
|
|
|
|
CP0554571
|
1-acetyl-N-[2-(4-methoxyphenyl)ethyl]-2,2,4-trimethyl-4-phenyl-3H-quinoline-6-carboxamide
Show/Hide
|
C30H34N2O3
|
1
|
| 1 |
IC50 = 1880 nM
|
|
|
|
CP0378100
|
N-(1-acetyl-2,2,4-trimethyl-4-phenyl-3H-quinolin-6-yl)-1-phenylmethanesulfonamide
Show/Hide
|
C27H30N2O3S
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
