| Compound ID |
Compound Name |
Compound Formula |
|
CP0105272
|
4-methoxy-N-[[4-phenyl-3-(trifluoromethyl)phenyl]carbamoyl]pyridine-3-carboxamide
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|
C21H16F3N3O3
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0233685
|
1-[[6-[(2-methoxy-4-propylphenyl)methoxy]-1-methyl-3,4-dihydronaphthalen-2-yl]methyl]azetidine-3-carboxylic acid
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|
C27H33NO4
|
2
|
| 1 |
EC50 > 30000 nM
|
|
|
| 2 |
Ki > 5450 nM
|
|
|
|
CP0355224
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-[4-(methylcarbamoyl)phenoxy]phenyl]-4-hydroxypiperidine-1-carboxamide
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|
C32H38FN3O5
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0375037
|
N-[3-(4-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C31H36FN3O5
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0379497
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-sulfamoylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamide
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|
C30H36FN3O6S
|
1
|
| 1 |
IC50 = 4.1 nM
|
|
|
|
CP0388589
|
N-[3-[4-(dimethylcarbamoyl)phenoxy]-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C33H40FN3O5
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0387270
|
N-[3-(3-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C31H36FN3O5
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0387271
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-4-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide
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|
C29H34FN3O4
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0411436
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-methylsulfonylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamide
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|
C31H37FN2O6S
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0398734
|
N-[3-(2-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C31H36FN3O5
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0411434
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-2-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide
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|
C29H34FN3O4
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0395995
|
US8975409, Example 9(3)
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|
C31H26F2N2O6
|
1
|
| 1 |
IC50 = 430 nM
|
|
|
|
CP0388588
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-methylphenyl]-4-hydroxypiperidine-1-carboxamide
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|
C25H33FN2O3
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0409055
|
2-[4-[3-(4-fluorophenoxy)-5-[[3-hydroxy-3-(2-methylpropyl)pyrrolidine-1-carbonyl]amino]phenoxy]phenyl]-2-methylpropanoic acid
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|
C31H35FN2O6
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0387268
|
N-[3-chloro-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C24H30ClFN2O3
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0477277
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-3-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide
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|
C29H34FN3O4
|
1
|
| 1 |
IC50 = 940 nM
|
|
|
|
CP0398647
|
N-[3,5-bis(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C30H34F2N2O4
|
1
|
| 1 |
IC50 = 980 nM
|
|
|
|
CP0494561
|
US8975409, Comparative compound B
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|
C24H31FN2O3
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0398502
|
N-[3-ethoxy-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
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|
C26H35FN2O4
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
