N-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]naphthalene-2-carboxamide

N-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]-6-fluoronaphthalene-2-carboxamide

4-fluoro-N-[(1R,2S)-2-(1H-indol-3-ylmethylamino)cyclohexyl]benzamide

4-fluoro-N-[(1R,2R)-2-(1H-indol-3-ylmethylamino)cyclohexyl]benzamide

N-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]-3,4-difluorobenzamide

N-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]-4-fluorobenzamide

N-[(1R,2S)-2-(3,3-dimethylbutylamino)cyclohexyl]-4-fluorobenzamide

4-fluoro-N-[(1R,2S)-2-[(4-methoxyphenyl)methylamino]cyclohexyl]benzamide

(1R,2S)-N-(4-fluorophenyl)-2-(1H-indol-3-ylmethylamino)cyclohexane-1-carboxamide

4-fluoro-N-[(1R,2S)-2-[(4-fluorophenyl)methylamino]cyclohexyl]benzamide

N-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]naphthalene-1-carboxamide

N-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]quinoline-2-carboxamide

N-[(1R,2S)-2-[[4-(diethylamino)phenyl]methylamino]cyclohexyl]-4-fluorobenzamide

4-fluoro-N-[(1R,2S)-2-[(3-hydroxyphenyl)methylamino]cyclohexyl]benzamide

4-fluoro-N-[(1R,2S)-2-(3-phenylpropylamino)cyclohexyl]benzamide

1-[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl]-3-(4-fluorophenyl)urea

4-fluoro-N-[(1R,2S)-2-[(4-methylphenyl)methylamino]cyclohexyl]benzamide

3,4-difluoro-N-[(1R,2R)-2-(1H-indol-3-ylmethylamino)cyclopentyl]benzamide

4-fluoro-N-[(1S,2R)-2-(1H-indol-3-ylmethylamino)cyclohexyl]benzamide

(1R,2R)-N-(4-fluorophenyl)-2-(1H-indol-3-ylmethylamino)cyclohexane-1-carboxamide

4-fluoro-N-[(1R,2S)-2-[1H-indol-3-ylmethyl(methyl)amino]cyclohexyl]benzamide

4-fluoro-N-[2-(1H-indol-3-ylmethylamino)ethyl]benzamide

4-[[[(1S,2R)-2-[(4-fluorobenzoyl)amino]cyclohexyl]amino]methyl]benzoic acid

[(1R,2S)-2-[(3,4-dichlorophenyl)methylamino]cyclohexyl] N-(4-fluorophenyl)carbamate

15-28-Somatostatin-28

1,1-Dipentyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

3-[(1R,3R)-3-[5-(4-fluorophenyl)-1H-imidazol-2-yl]-1-(1-methylpyrazol-4-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methyl-1,2,4-oxadiazole

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US8754099, 21

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(3R)-1,1-dibutyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indole

(3S)-1,1-dibutyl-3-(5-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indole

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1-Cyclohexyl-1-methyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

2-[13-(4-Amino-butyl)-7,22-dibenzyl-10-(1-hydroxy-ethyl)-16,19-bis-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaaza-cyclopentacos-5-yl]-acetamide

1-Cyclohexyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline oxalate salt

2-[25-Amino-13-(4-amino-butyl)-7,22-dibenzyl-10-(1-hydroxy-ethyl)-16,19-bis-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaaza-cyclohexacos-5-yl]-acetamide

1,1-Dibutyl-6-chloro-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

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(4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-16-benzyl-N-[(2S,3R)-1,3-dihydroxybutan-2-yl]-7-[(1R)-1-hydroxyethyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carboxamide

1-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-4-[5-(4-fluorophenyl)-1H-imidazol-2-yl]piperidine

6-Methyl-1,1-dipentyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

4-{8-[(2,6-diethoxy-4'-fluorobiphenyl-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]dec-2-yl}benzoic acid trifluoromethyl acetate

2-Amino-N-[13-(4-amino-butyl)-7,22-dibenzyl-5-carbamoylmethyl-10-(1-hydroxy-ethyl)-16,19-bis-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaaza-cyclohexacos-25-yl]-3-phenyl-propionamide

2-[9-(4-Amino-butyl)-3,18-dibenzyl-6-(1-hydroxy-ethyl)-12,15-bis-(1H-indol-3-ylmethyl)-2,5,8,11,14,17,20,25-octaoxo-1,4,7,10,13,16,19,24octaaza-cyclooctacos-1-yl]-acetamide

2-[13-(4-Amino-butyl)-7,22-dibenzyl-10-(1-hydroxy-ethyl)-16,19-bis-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaaza-cyclohexacos-5-yl]-acetamide

2-[(7R,10S,13R,16R,19R,22S)-26-[2-amino-3-(naphthalen-1-yl)propanoyl]-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-16,19-bis(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23,26-octaazacyclooctacosan-5-yl]acetamide

2-amino-N-[(7R,10S,13R,16R,19R,22S)-13-(4-aminobutyl)-7,22-dibenzyl-5-(carbamoylmethyl)-10-[(1R)-1-hydroxyethyl]-16,19-bis(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaazacyclohexacosan-25-yl]-3-phenylpropanamide

2-[(7R,10S,13R,16R,19R,22S)-26-(2-amino-3-phenylpropanoyl)-13-(4-aminobutyl)-7,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-16,19-bis(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23,26-octaazacyclooctacosan-5-yl]acetamide

(4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2

(4-amino)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2

(4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2

(4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Thr-NH2

(4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2

(4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Asp-NH2

(4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2

(3S)-4-amino-3-[[(4S,7R,10S,13R,16S,19R)-10-(4-aminobutyl)-19-[[(2S)-2-amino-3-phenylpropanoyl]amino]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-7-propan-2-yl-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]amino]-4-oxobutanoic acid

(4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-Cys]-Asp-NH2

(4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH2

(4R,7S,10R,13S,16R,19S,22R,25S,28R,31S)-13,28-bis(4-aminobutyl)-25-(2-amino-2-oxoethyl)-31-[[2-[[(2S)-2-aminopropanoyl]amino]acetyl]amino]-19,22-dibenzyl-10-[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-16-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30-nonaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29-nonazacyclodotriacontane-4-carboxylic acid

[(1S,2R,3S,5R,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[3-[[(2R)-3-amino-2-[[(4R,7S,10S,13R,16S,19R)-10-(4-aminobutyl)-19-[[(2R)-2-amino-3-phenylpropanoyl]amino]-7-[(1R)-1-hydroxyethyl]-16-[(4-hydroxyphenyl)methyl]-13-(1H-indol-3-ylmethyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentazacycloicosane-4-carbonyl]amino]-3-oxopropyl]disulfanyl]propanoyl-methylamino]propanoate

Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys] (SRIF14)

1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline with oxalate salt

1,1-Diethyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

1-Pentyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

3-(4-phenyl-1H-2-imidazolyl)-(3S)-spiro[2,3,4,9-tetrahydro-1H-b-carboline-1,2'-(2',3'-dihydro-1'H-indene)]

6-Benzyloxy-1,1-dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

1,1-Dihexyl-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

Dimethyl-{4-[3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carbolin-1-yl]-phenyl}-amine

1-(4-Methoxy-phenyl)-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

1-[3-(4-phenyl-1H-2-imidazolyl)-(3S)-spiro[2,3,4,9-tetrahydro-1H-b-carboline-1,4'-(hexahydropyridine)]-1-yl]-1-ethanone

3-(4-phenyl-1H-2-imidazolyl)-(3S)-spiro[2,3,4,9-tetrahydro-1H-b-carboline-1,2'-tricyclo[3.3.1.13,7]decane];2 hydrochloride salt

1-(2-Nitro-phenyl)-3-(4-phenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

3-(4-Phenyl-1H-imidazol-2-yl)-1-pyridin-4-yl-2,3,4,9-tetrahydro-1H-beta-carboline

1,1-Dibutyl-3-(4-phenyl-1H-imidazol-2-yl)-1,2,3,4-tetrahydro-benzo[4,5]thieno[2,3-c]pyridine

1-Cyclohexyl-3-(4-phenyl-1H-imidazol-2-yl)-9H-beta-carboline

N-[(2R)-1-(5-aminopentylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl]spiro[indene-1,4'-piperidine]-1'-carboxamide

1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarbamoyl]-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide

1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide

1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarbamoyl]-2-(1H-3-indolyl)-(1S)-ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide

1,1-Dibutyl-3-(4-phenyl-thiazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline with hydrochloride salt

1,1-Dibutyl-3-(4,5-diphenyl-1H-imidazol-2-yl)-2,3,4,9-tetrahydro-1H-beta-carboline

1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)ethyl]spiro[1H-indene-1,4'-(hexahydropyridine)]-1'-carboxamide