| Compound ID |
Compound Name |
Compound Formula |
|
CP0476143
|
18-[[(1S)-5-[3-[2-[2-[3-[2-[2-[[2-[(2R)-3-[(2-amino-2-oxoethyl)amino]-2-[[2-[[(3R,6S,9S,12S,15S)-6-(2-amino-2-oxoethyl)-9-(3-amino-3-oxopropyl)-12-[(2S)-butan-2-yl]-15-[(4-hydroxyphenyl)methyl]-5,8,11,14,17-pentaoxo-1-thia-4,7,10,13,16-pentazacycloicosane-3-carbonyl]amino]acetyl]amino]-3-oxopropyl]sulfanylacetyl]amino]ethoxy]ethoxy]propanoylamino]ethoxy]ethoxy]propanoylamino]-1-carboxypentyl]amino]-18-oxooctadecanoic acid
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|
C78H129N15O24S2
|
1
|
| 1 |
EC50 = 1800 nM
|
|
|
|
CP0474311
|
N-[4-[(5S)-5-hydroxy-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
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|
C25H24N2O3
|
1
|
| 1 |
Ki = 4.87 nM
|
|
|
|
CP0548474
|
N-[4-(5-hydroxy-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)phenyl]-2-methylbenzamide
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|
C25H24N2O3
|
1
|
| 1 |
Ki = 7.56 nM
|
|
|
|
CP0474312
|
N-[4-[(5R)-5-hydroxy-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
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|
C25H24N2O3
|
1
|
| 1 |
Ki = 8.3 nM
|
|
|
|
CP0573811
|
N-[4-[(5S)-5-hydroxy-6-methyl-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
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|
C26H26N2O3
|
1
|
| 1 |
Ki = 46 nM
|
|
|
|
CP0521728
|
N-[4-[(5S)-5-hydroxy-9-methyl-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
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|
C26H26N2O3
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0543049
|
N-[4-[(5R)-5-hydroxy-9-methyl-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
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|
C26H26N2O3
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0521729
|
N-[4-(5-hydroxy-6-methyl-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)phenyl]-2-methylbenzamide
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|
C26H26N2O3
|
1
|
| 1 |
Ki = 160 nM
|
|
|
|
CP0548473
|
N-[4-(5-hydroxy-9-methyl-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)phenyl]-2-methylbenzamide
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|
C26H26N2O3
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0195952
|
(2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl)-3-(2-methoxyphenyl)-2-oxoindolin-3-yl)-4-hydroxy-N,N-dimethylpyrrolidine-2-carboxamide
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|
C30H32ClN3O8S
|
1
|
| 1 |
Ki = 325 nM
|
|
|
|
CP0543048
|
N-[4-[(5R)-5-hydroxy-6-methyl-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
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|
C26H26N2O3
|
1
|
| 1 |
Ki = 1790 nM
|
|
|
|
CP0845382
|
N-(cyclohexylmethyl)-1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)piperidin-4-amine hydrochloride
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|
C31H46ClN3O6S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0874438
|
N-(cyclohexylmethyl)-1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetrahydroquinolin-2-yl)ethylsulfonyl)piperidin-4-amine hydrobromide
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|
C31H46BrN3O6S2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
