| Compound ID |
Compound Name |
Compound Formula |
|
CP0089615
|
3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(1-methylethyl)isoxazol-4-yl]methoxy}phenyl)ethenyl]benzoic acid
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|
C28H22Cl3NO4
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0579341
|
propan-2-yl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
Show/Hide
|
C35H39N3O3
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0081982
|
(E)-3-{3-[Cyclohexanecarbonyl-(4'-dimethylamino-biphenyl-4-ylmethyl)-amino]-phenyl}-acrylic acid methyl ester
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|
C32H36N2O3
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0546480
|
propan-2-yl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-5-fluorophenyl]prop-2-enoate
Show/Hide
|
C35H38FN3O3
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0546481
|
propan-2-yl (E)-3-[5-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-2-fluorophenyl]prop-2-enoate
Show/Hide
|
C35H38FN3O3
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0552083
|
methyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
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|
C33H35N3O3
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0564628
|
cyclopropyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
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|
C35H37N3O3
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0564629
|
propan-2-yl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-2-fluorophenyl]prop-2-enoate
Show/Hide
|
C35H38FN3O3
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0573662
|
methyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)-2-fluorophenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
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|
C33H34FN3O3
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0577647
|
methyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-5-fluorophenyl]prop-2-enoate
Show/Hide
|
C33H34FN3O3
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0569363
|
ethyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-5-fluorophenyl]prop-2-enoate
Show/Hide
|
C34H36FN3O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0569899
|
ethyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-2-fluorophenyl]prop-2-enoate
Show/Hide
|
C34H36FN3O3
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0546484
|
methyl (E)-3-[3-[[4-[2-chloro-4-(dimethylamino)phenyl]-3-cyanophenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
Show/Hide
|
C33H34ClN3O3
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0552084
|
ethyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
Show/Hide
|
C34H37N3O3
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0550464
|
methyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-2-fluorophenyl]prop-2-enoate
Show/Hide
|
C33H34FN3O3
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0573663
|
ethyl (E)-3-[5-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-2-fluorophenyl]prop-2-enoate
Show/Hide
|
C34H36FN3O3
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0545495
|
methyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)-2-methylphenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
Show/Hide
|
C34H37N3O3
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0546482
|
methyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-4-fluorophenyl]prop-2-enoate
Show/Hide
|
C33H34FN3O3
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0578418
|
methyl (E)-3-[5-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-2-fluorophenyl]prop-2-enoate
Show/Hide
|
C33H34FN3O3
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0547249
|
ethyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]-4-fluorophenyl]prop-2-enoate
Show/Hide
|
C34H36FN3O3
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0570121
|
methyl (E)-3-[3-[[3-cyano-4-[2-cyano-4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
Show/Hide
|
C34H34N4O3
|
1
|
| 1 |
EC50 = 1600 nM
|
|
|
|
CP0579975
|
fluoromethyl (E)-3-[3-[[3-cyano-4-[4-(dimethylamino)phenyl]phenyl]methyl-(cyclohexanecarbonyl)amino]phenyl]prop-2-enoate
Show/Hide
|
C33H34FN3O3
|
1
|
| 1 |
EC50 = 2600 nM
|
|
|
|
CP0546478
|
methyl (E)-3-[3-[cyclohexanecarbonyl-[[7-(dimethylamino)-9,10-dihydrophenanthren-2-yl]methyl]amino]phenyl]prop-2-enoate
Show/Hide
|
C34H38N2O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0546479
|
methyl (E)-3-[3-[cyclohexanecarbonyl-[[7-(dimethylamino)phenanthren-2-yl]methyl]amino]phenyl]prop-2-enoate
Show/Hide
|
C34H36N2O3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0546483
|
methyl (E)-3-[3-[cyclohexanecarbonyl-[[4-[4-(dimethylamino)phenyl]-3-(methoxymethyl)phenyl]methyl]amino]phenyl]prop-2-enoate
Show/Hide
|
C34H40N2O4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
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