| Compound ID |
Compound Name |
Compound Formula |
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CP0000189
|
4-{[(2S,4S)-1-[2-(3-chloro-4-{[(2-methylphenyl)carbamoyl]amino}phenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
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|
C28H27ClFN3O5
|
2
|
| 1 |
IC50 = 0.51 nM
|
|
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| 2 |
IC50 = 7.2 nM
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|
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CP0112732
|
4-{[(2S,4S)-1-[2-(3-bromo-4-{[(2-methylphenyl)carbamoyl]amino}phenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
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|
C28H27BrFN3O5
|
2
|
| 1 |
IC50 = 0.78 nM
|
|
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| 2 |
IC50 = 8.4 nM
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CP0346334
|
4-{[(2S,4S)-1-[2-(4-{[(2-chlorophenyl)carbamoyl]amino}-3-methoxyphenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
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|
C28H27ClFN3O6
|
2
|
| 1 |
IC50 = 0.87 nM
|
|
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| 2 |
IC50 = 6.2 nM
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CP0511029
|
4-{[(2S,4S)-4-fluoro-1-[2-(3-methoxy-4-{[(2-methylphenyl)carbamoyl]amino}phenyl)acetyl]pyrrolidin-2-yl]methoxy}benzoic acid
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|
C29H30FN3O6
|
2
|
| 1 |
IC50 = 1.2 nM
|
|
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| 2 |
IC50 = 3.7 nM
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CP0112731
|
4-{[(2S,4S)-1-[2-(3-bromo-4-{[(2-chlorophenyl)carbamoyl]amino}phenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C27H24BrClFN3O5
|
2
|
| 1 |
IC50 = 1.3 nM
|
|
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| 2 |
IC50 = 51 nM
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CP0346336
|
4-{[(2S,4S)-1-[2-(3-chloro-4-{[(2-chlorophenyl)carbamoyl]amino}phenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C27H24Cl2FN3O5
|
2
|
| 1 |
IC50 = 1.3 nM
|
|
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| 2 |
IC50 = 81 nM
|
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CP0276640
|
4-{[(2S,4S)-1-[2-(3-bromo-4-{[(2-bromophenyl)carbamoyl]amino}phenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C27H24Br2FN3O5
|
2
|
| 1 |
IC50 = 1.4 nM
|
|
|
| 2 |
IC50 = 95 nM
|
|
|
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CP0346333
|
4-{[(2S,4S)-1-[2-(4-{[(2-bromophenyl)carbamoyl]amino}-3-methoxyphenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C28H27BrFN3O6
|
2
|
| 1 |
IC50 = 1.6 nM
|
|
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| 2 |
IC50 = 16 nM
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|
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CP0062222
|
4-{[(2S,4S)-1-[2-(4-{[(2-bromophenyl)carbamoyl]amino}-3-chlorophenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C27H24BrClFN3O5
|
2
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
IC50 = 137 nM
|
|
|
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CP0112733
|
4-{[(2S,4S)-4-fluoro-1-[2-(3-methyl-4-{[(2-methylphenyl)carbamoyl]amino}phenyl)acetyl]pyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C29H30FN3O5
|
2
|
| 1 |
IC50 = 2.3 nM
|
|
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| 2 |
IC50 = 49 nM
|
|
|
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CP0000190
|
4-[[(2S,4S)-4-fluoro-1-[2-[2-(2-methylanilino)-1,3-benzoxazol-6-yl]acetyl]pyrrolidin-2-yl]methoxy]cyclohexane-1-carboxylic acid
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|
C28H32FN3O5
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
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CP0306021
|
4-{[(2S,4S)-4-fluoro-1-[2-(3-methoxy-4-{[(2-methoxyphenyl)carbamoyl]amino}phenyl)acetyl]pyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C29H30FN3O7
|
2
|
| 1 |
IC50 = 9.2 nM
|
|
|
| 2 |
IC50 = 268 nM
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CP0442128
|
4-{[(2S,4S)-1-[2-(4-{[(2-bromophenyl)carbamoyl]amino}-3-methylphenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C28H27BrFN3O5
|
2
|
| 1 |
IC50 = 9.8 nM
|
|
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| 2 |
IC50 = 622 nM
|
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|
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CP0171979
|
4-{[(2S,4S)-1-[2-(4-{[(2-chlorophenyl)carbamoyl]amino}-3-methylphenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C28H27ClFN3O5
|
2
|
| 1 |
IC50 = 13 nM
|
|
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| 2 |
IC50 = 416 nM
|
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CP0369218
|
4-{[(2S,4S)-1-[2-(3-ethyl-4-{[(2-methylphenyl)carbamoyl]amino}phenyl)acetyl]-4-fluoropyrrolidin-2-yl]methoxy}benzoic acid
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|
C30H32FN3O5
|
2
|
| 1 |
IC50 = 15 nM
|
|
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| 2 |
IC50 = 282 nM
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CP0502974
|
4-{[(2S,4S)-4-fluoro-1-[2-(4-{[(2-methylphenyl)carbamoyl]amino}-3-(trifluoromethyl)phenyl)acetyl]pyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C29H27F4N3O5
|
2
|
| 1 |
IC50 = 15 nM
|
|
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| 2 |
IC50 = 486 nM
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CP0530335
|
4-[[2-(2-Methylphenylamino)-6-benzoxazolylacetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid
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|
C28H32FN3O5
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
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CP0490685
|
1-[(4S)-Fluoro-1-[2-(2-methylphenylamino)-6-benzoxazolylacetyl]-(2S)-pyrrolidinylcarbonyl]-4-piperidinylacetic acid
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|
C28H31FN4O5
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
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CP0535344
|
4-[(4S)-fluoro-1-[2-(2-methylphenylamino)-6-benzoxazolylacetyl]-(2S)-pyrrolidinylmethoxy]benzoic acid
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|
C28H26FN3O5
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0505328
|
4-[(4S)-Fluoro-1-[2-(2-methylphenylamino)-6-benzoxazolylacetyl]-(2S)-pyrrolidinylcarbonyl]-1-piperazinylacetic acid
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|
C27H30FN5O5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0309463
|
4-{[(2S,4S)-4-fluoro-1-{2-[3-methoxy-4-({[2-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]acetyl}pyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C29H27F4N3O6
|
2
|
| 1 |
IC50 = 106 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
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CP0522744
|
6-[(4S)-Fluoro-1-[2-(2-methylphenyl)amino-6-benzoxazolylacetyl]-(2S)-pyrrolidinylmethoxy]hexanoic acid
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|
C27H32FN3O5
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0535345
|
5-[(4S)-Fluoro-1-[2-(2-methylphenyl)amino-6-benzoxazolylacetyl]-(2S)-pyrrolidinylmethoxy]pentanoic acid
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|
C26H30FN3O5
|
1
|
| 1 |
IC50 = 198 nM
|
|
|
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CP0551829
|
4-{[(2S,4S)-4-fluoro-1-[2-(4-{[(2-methylphenyl)carbamoyl]amino}-3-(propan-2-yl)phenyl)acetyl]pyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C31H34FN3O5
|
2
|
| 1 |
IC50 = 216 nM
|
|
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| 2 |
IC50 > 1000 nM
|
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|
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CP0437942
|
4-[[(2S,4S)-4-fluoro-1-[2-[2-(2-methylanilino)-1,3-benzoxazol-6-yl]acetyl]pyrrolidin-2-yl]methoxy]cyclohexane-1-carboxylic acid
Show/Hide
|
C28H32FN3O5
|
1
|
| 1 |
IC50 = 443 nM
|
|
|
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CP0334956
|
4-{[(2S,4S)-4-fluoro-1-{2-[3-methoxy-4-({[2-(propan-2-yl)phenyl]carbamoyl}amino)phenyl]acetyl}pyrrolidin-2-yl]methoxy}benzoic acid
Show/Hide
|
C31H34FN3O6
|
2
|
| 1 |
IC50 = 769 nM
|
|
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| 2 |
IC50 > 1000 nM
|
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CP0489402
|
4-[(4S)-fluoro-1-[2-(2-methylphenylamino)-6-benzoxazolylacetyl]-(2S)-pyrrolidinylmethoxy]butanoic acid
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|
C25H28FN3O5
|
1
|
| 1 |
IC50 = 831 nM
|
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|
