| Compound ID |
Compound Name |
Compound Formula |
|
CP0039348
|
(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
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|
C12H16N6O4
|
2
|
| 1 |
EC50 = 11.22 nM
|
|
|
| 2 |
EC50 = 17.6 nM
|
|
|
|
CP0001102
|
(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol
Show/Hide
|
C10H13N5O4
|
1
|
| 1 |
EC50 = 25.12 nM
|
|
|
|
CP0280427
|
4-[2-[6-amino-9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]purin-2-yl]sulfanylethyl]benzenesulfonic acid
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|
C18H21N5O7S2
|
1
|
| 1 |
EC50 = 117 nM
|
|
|
|
CP0488244
|
(2R,3R,4S,5R)-2-[6-[[(1R,2R)-2-(3-chlorophenoxy)cyclopentyl]amino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol
Show/Hide
|
C21H24ClN5O5
|
1
|
| 1 |
EC50 = 549.54 nM
|
|
|
|
CP0488425
|
(2R,3R,4S,5R)-2-[6-[[(1R,2R)-2-(2-chlorophenoxy)cyclopentyl]amino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol
Show/Hide
|
C21H24ClN5O5
|
1
|
| 1 |
EC50 = 1096.48 nM
|
|
|
|
CP0488422
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-(3-chlorophenoxy)cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C23H27ClN6O5
|
1
|
| 1 |
EC50 = 1380.38 nM
|
|
|
|
CP0495148
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-[(2-chlorophenyl)methoxy]cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C24H29ClN6O5
|
1
|
| 1 |
EC50 = 2089.3 nM
|
|
|
|
CP0488416
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-(2-chlorophenoxy)cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C23H27ClN6O5
|
1
|
| 1 |
EC50 = 2137.96 nM
|
|
|
|
CP0495143
|
(2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-[6-[[(1R,2R)-2-phenoxycyclopentyl]amino]purin-9-yl]oxolane-2-carboxamide
Show/Hide
|
C23H28N6O5
|
1
|
| 1 |
EC50 = 3311.31 nM
|
|
|
|
CP0488420
|
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-[6-[[(1R,2R)-2-(3-methoxyphenoxy)cyclopentyl]amino]purin-9-yl]oxolane-3,4-diol
Show/Hide
|
C22H27N5O6
|
1
|
| 1 |
EC50 = 5754.4 nM
|
|
|
|
CP0494931
|
(2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-[6-[[(1R,2R)-2-(3-methoxyphenoxy)cyclopentyl]amino]purin-9-yl]oxolane-2-carboxamide
Show/Hide
|
C24H30N6O6
|
1
|
| 1 |
EC50 = 6309.57 nM
|
|
|
|
CP0546622
|
(2R,3R,4S,5R)-2-[6-[[(1R,2R)-2-[(2-chlorophenyl)methoxy]cyclopentyl]amino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol
Show/Hide
|
C22H26ClN5O5
|
1
|
| 1 |
EC50 = 6760.83 nM
|
|
|
|
CP0488424
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-[(3-chlorophenyl)methoxy]cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C24H29ClN6O5
|
1
|
| 1 |
EC50 = 9120.11 nM
|
|
|
|
CP0381926
|
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-[6-[[(1R,2R)-2-phenylmethoxycyclopentyl]amino]purin-9-yl]oxolane-3,4-diol
Show/Hide
|
C22H27N5O5
|
1
|
| 1 |
EC50 = 11220.18 nM
|
|
|
|
CP0488249
|
(2R,3R,4S,5R)-2-[6-[[(1R,2R)-2-(4-chlorophenoxy)cyclopentyl]amino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol
Show/Hide
|
C21H24ClN5O5
|
1
|
| 1 |
EC50 = 13803.84 nM
|
|
|
|
CP0495164
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-(4-chlorophenoxy)cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C23H27ClN6O5
|
1
|
| 1 |
EC50 = 13803.84 nM
|
|
|
|
CP0534813
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-(4-tert-butylphenoxy)cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C27H36N6O5
|
1
|
| 1 |
EC50 = 14454.4 nM
|
|
|
|
CP0488250
|
(2S,3S,4R,5R)-5-[6-[[(1R,2R)-2-(3-bromophenoxy)cyclopentyl]amino]purin-9-yl]-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
Show/Hide
|
C23H27BrN6O5
|
1
|
| 1 |
EC50 = 26302.68 nM
|
|
|
|
CP0041613
|
Anapriline
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|
C16H21NO2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0066236
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-8-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0366351
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-5-yl)oxy]propan-2-ol
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|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0558089
|
5-[5-amino-2-[(3-chloro-5-fluoropyridin-2-yl)methyl]-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1H-pyridin-2-one
Show/Hide
|
C22H15ClFN7O
|
1
|
| 1 |
IC50 = 0.29 nM
|
|
|
|
CP0544730
|
5-[5-amino-7-(4-fluorophenyl)-2-[(5-fluoropyridin-2-yl)methyl]-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1H-pyridin-2-one
Show/Hide
|
C22H15F2N7O
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0544336
|
5-[5-amino-2-[(R)-(3-fluoropyridin-2-yl)-hydroxymethyl]-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1-methylpyridin-2-one
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|
C23H18FN7O2
|
1
|
| 1 |
IC50 = 0.52 nM
|
|
|
|
CP0573987
|
5-[5-amino-2-[(3-fluoropyridin-2-yl)methyl]-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1-methylpyridin-2-one
Show/Hide
|
C23H18FN7O
|
1
|
| 1 |
IC50 = 0.57 nM
|
|
|
|
CP0544728
|
5-[5-amino-7-(4-fluorophenyl)-2-(3,3,3-trifluoropropyl)-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1H-pyridin-2-one
Show/Hide
|
C19H14F4N6O
|
1
|
| 1 |
IC50 = 0.74 nM
|
|
|
|
CP0544729
|
5-[5-amino-7-(4-fluorophenyl)-2-(piperidin-1-ylmethyl)-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-3-methyl-1H-pyridin-2-one
Show/Hide
|
C23H24FN7O
|
1
|
| 1 |
IC50 = 5.72 nM
|
|
|
|
CP0558090
|
5-[5-amino-2-[(5-methoxypyridin-2-yl)methyl]-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1-methylpyridin-2-one
Show/Hide
|
C24H21N7O2
|
1
|
| 1 |
IC50 = 7.72 nM
|
|
|
|
CP0554492
|
5-[5-amino-7-(4-fluorophenyl)-2-[(R)-(3-fluoropyridin-2-yl)-hydroxymethyl]-[1,2,4]triazolo[1,5-c]pyrimidin-8-yl]-1-methylpyridin-2-one
Show/Hide
|
C23H17F2N7O2
|
1
|
| 1 |
IC50 = 8.7 nM
|
|
|
|
CP0544727
|
2-[(3-fluoropyridin-2-yl)methyl]-7-phenyl-8-pyridazin-4-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-amine
Show/Hide
|
C21H15FN8
|
1
|
| 1 |
IC50 = 9.07 nM
|
|
|
|
CP0496978
|
(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(thiophen-2-yl)methanone
Show/Hide
|
C17H12N4OS2
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0496981
|
[6-chloro-2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]-thiophen-2-ylmethanone
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|
C17H11ClN4OS2
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0558091
|
2-(oxolan-2-ylmethyl)-7-phenyl-8-pyridazin-4-yl-[1,2,4]triazolo[1,5-c]pyrimidin-5-amine
Show/Hide
|
C20H19N7O
|
1
|
| 1 |
IC50 = 83.87 nM
|
|
|
|
CP0384259
|
(5-methylthiophen-2-yl)(2-(1-(pyridin-3-yl)ethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C19H16N4OS2
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0384264
|
(5-methylthiophen-2-yl)(2-(pyrimidin-4-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C17H13N5OS2
|
1
|
| 1 |
IC50 = 116 nM
|
|
|
|
CP0501313
|
(5-methylthiophen-2-yl)(2-(1-(pyridin-2-yl)ethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C19H16N4OS2
|
1
|
| 1 |
IC50 = 118 nM
|
|
|
|
CP0476167
|
(2-(ethylamino)thieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
Show/Hide
|
C14H13N3OS2
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
|
CP0504370
|
N-[4-(5-methylthiophene-2-carbonyl)thieno[3,2-d]pyrimidin-2-yl]pyridine-3-carboxamide
Show/Hide
|
C18H12N4O2S2
|
1
|
| 1 |
IC50 = 161 nM
|
|
|
|
CP0476169
|
(5-methylthiophen-2-yl)(2-(2-(pyridin-3-yl)ethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C19H16N4OS2
|
1
|
| 1 |
IC50 = 177 nM
|
|
|
|
CP0447389
|
(5-methylthiophen-2-yl)(2-(pyridin-2-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C18H14N4OS2
|
1
|
| 1 |
IC50 = 186 nM
|
|
|
|
CP0390930
|
(2-aminothieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
Show/Hide
|
C12H9N3OS2
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0390927
|
(5-methylthiophen-2-yl)(2-(2-(pyridin-2-yl)ethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C19H16N4OS2
|
1
|
| 1 |
IC50 = 351 nM
|
|
|
|
CP0384261
|
(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(thiophen-3-yl)methanone
Show/Hide
|
C17H12N4OS2
|
1
|
| 1 |
IC50 = 405 nM
|
|
|
|
CP0384265
|
(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(p-tolyl)methanone
Show/Hide
|
C20H16N4OS
|
1
|
| 1 |
IC50 = 442 nM
|
|
|
|
CP0390929
|
(S)-[2-(1-Pyridin-3-yl-ethylamino)-thieno[3,2-d]pyrimidin-4-yl]-pyrrolidin-1-yl-methanone
Show/Hide
|
C18H19N5OS
|
1
|
| 1 |
IC50 = 468 nM
|
|
|
|
CP0496979
|
(4-methoxyphenyl)(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C20H16N4O2S
|
1
|
| 1 |
IC50 = 637 nM
|
|
|
|
CP0390928
|
2-[(Pyridin-3-ylmethyl)-amino]-thieno[3,2-d]pyrimidine-4-carboxylic acid cyclo-propylamide
Show/Hide
|
C16H15N5OS
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0447393
|
(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(thiazol-2-yl)methanone
Show/Hide
|
C16H11N5OS2
|
1
|
| 1 |
IC50 = 732 nM
|
|
|
|
CP0384266
|
[6-(methylamino)-2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]-thiophen-2-ylmethanone
Show/Hide
|
C18H15N5OS2
|
1
|
| 1 |
IC50 = 965 nM
|
|
|
|
CP0384258
|
(5-methylthiophen-2-yl)(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C18H14N4OS2
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0390932
|
(5-methylthiophen-2-yl)(2-(1-phenylethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C20H17N3OS2
|
1
|
| 1 |
IC50 = 1077 nM
|
|
|
|
CP0496980
|
pyridin-3-yl-[2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]methanone
Show/Hide
|
C18H13N5OS
|
1
|
| 1 |
IC50 = 1168 nM
|
|
|
|
CP0447391
|
(5-methylfuran-2-yl)(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C18H14N4O2S
|
1
|
| 1 |
IC50 = 1252 nM
|
|
|
|
CP0447387
|
[6-(dimethylamino)-2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]-thiophen-2-ylmethanone
Show/Hide
|
C19H17N5OS2
|
1
|
| 1 |
IC50 = 1417 nM
|
|
|
|
CP0384260
|
(5-chlorothiophen-2-yl)(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C17H11ClN4OS2
|
1
|
| 1 |
IC50 = 1541 nM
|
|
|
|
CP0384262
|
phenyl-[2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]methanone
Show/Hide
|
C19H14N4OS
|
1
|
| 1 |
IC50 = 1619 nM
|
|
|
|
CP0501314
|
(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(thiazol-5-yl)methanone
Show/Hide
|
C16H11N5OS2
|
1
|
| 1 |
IC50 = 1715 nM
|
|
|
|
CP0496983
|
(2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(pyridin-4-yl)methanone
Show/Hide
|
C18H13N5OS
|
1
|
| 1 |
IC50 = 1942 nM
|
|
|
|
CP0470014
|
(2-(methyl(pyridin-3-ylmethyl)amino)thieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
Show/Hide
|
C19H16N4OS2
|
1
|
| 1 |
IC50 = 2271 nM
|
|
|
|
CP0496982
|
(+/-)-[2-(1-Pyridin-3-yl-ethylamino)-thieno[3,2-d]pyrimidin-4-yl]-pyrrolidin-1-yl-methanone
Show/Hide
|
C18H19N5OS
|
1
|
| 1 |
IC50 = 2347 nM
|
|
|
|
CP0447384
|
[6-(ethylamino)-2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]-thiophen-2-ylmethanone
Show/Hide
|
C19H17N5OS2
|
1
|
| 1 |
IC50 = 2485 nM
|
|
|
|
CP0459103
|
2-[(Pyridin-3-ylmethyl)-amino]-thieno[3,2-d]pyrimidine-4-carboxylic acid ethyl-amide
Show/Hide
|
C15H15N5OS
|
1
|
| 1 |
IC50 = 2516 nM
|
|
|
|
CP0440060
|
2-[(Pyridin-3-ylmethyl)-amino]-thieno[3,2-d]pyrimidine-4-carboxylic acid iso-propylamide
Show/Hide
|
C16H17N5OS
|
1
|
| 1 |
IC50 = 2610 nM
|
|
|
|
CP0390935
|
2-[(Pyridin-3-ylmethyl)-amino]-thieno[3,2-d]pyrimidine-4-carboxylic acid cyclo-hexylamide
Show/Hide
|
C19H21N5OS
|
1
|
| 1 |
IC50 = 3093 nM
|
|
|
|
CP0496977
|
(2-ethylthieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
Show/Hide
|
C14H12N2OS2
|
1
|
| 1 |
IC50 = 3852 nM
|
|
|
|
CP0440061
|
[2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]-pyrrolidin-1-ylmethanone
Show/Hide
|
C17H17N5OS
|
1
|
| 1 |
IC50 = 6136 nM
|
|
|
|
CP0501316
|
(5-methylthiophen-2-yl)(thieno[3,2-d]pyrimidin-4-yl)methanone
Show/Hide
|
C12H8N2OS2
|
1
|
| 1 |
IC50 = 6685 nM
|
|
|
|
CP0501315
|
(R)-[2-(1-Pyridin-3-yl-ethylamino)-thieno[3,2-d]pyrimidin-4-yl]-pyrrolidin-1-yl-methanone
Show/Hide
|
C18H19N5OS
|
1
|
| 1 |
IC50 = 6760 nM
|
|
|
|
CP0476145
|
2-[(Pyridin-3-ylmethyl)-amino]-thieno[3,2-d]pyrimidine-4-carboxylic acid methyl-amide
Show/Hide
|
C14H13N5OS
|
1
|
| 1 |
IC50 = 7107 nM
|
|
|
|
CP0384256
|
(2-(benzylamino)thieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
Show/Hide
|
C19H15N3OS2
|
1
|
| 1 |
IC50 = 7146 nM
|
|
|
|
CP0501312
|
(2-methylthieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
Show/Hide
|
C13H10N2OS2
|
1
|
| 1 |
IC50 = 7847 nM
|
|
|
|
CP0384263
|
[6-amino-2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin-4-yl]-thiophen-2-ylmethanone
Show/Hide
|
C17H13N5OS2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0390931
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(2-(cyclohexylmethylamino)thieno[3,2-d]pyrimidin-4-yl)(5-methylthiophen-2-yl)methanone
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C19H21N3OS2
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1
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| 1 |
IC50 > 10000 nM
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CP0439129
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3-[4-amino-6-[(2-chlorophenyl)methyl]thieno[2,3-d]pyrimidin-2-yl]benzonitrile
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C20H13ClN4S
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1
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| 1 |
Ki = 1.4 nM
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CP0497573
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6-benzyl-2-pyrazin-2-ylthieno[2,3-d]pyrimidin-4-amine
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C17H13N5S
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1
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| 1 |
Ki = 2.4 nM
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CP0560179
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N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)-3,6-dihydro-2H-pyridine-1-carboxamide
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C18H22N4O3S
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1
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| 1 |
Ki = 2.4 nM
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CP0576118
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4-(fluoromethyl)-4-hydroxy-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
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C19H25FN4O4S
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1
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| 1 |
Ki = 2.8 nM
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CP0467091
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6-[(2-chlorophenyl)methyl]-2-(5-methylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
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C18H14ClN3OS
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1
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| 1 |
Ki = 2.9 nM
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CP0137617
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]pyrazole-4-carboxamide
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C24H22F3N5O3S
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1
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| 1 |
Ki = 3 nM
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CP0388260
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-1-[(3-fluorophenyl)methyl]pyrazole-4-carboxamide
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C23H22FN5O3S
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1
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| 1 |
Ki = 3 nM
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CP0406020
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4-fluoro-N-(7-(N-isobutylacetamido)-4-methoxybenzo[d]thiazol-2-yl)benzamide
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C21H22FN3O3S
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1
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| 1 |
Ki = 3 nM
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CP0571395
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4-fluoro-4-(hydroxymethyl)-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
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C19H25FN4O4S
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1
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| 1 |
Ki = 3.6 nM
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CP0576200
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4-(fluoromethyl)-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
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C19H25FN4O3S
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1
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| 1 |
Ki = 3.6 nM
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CP0467093
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6-[(2-fluorophenyl)methyl]-2-(5-methylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
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C18H14FN3OS
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1
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| 1 |
Ki = 3.7 nM
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CP0572012
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4-hydroxy-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
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C18H24N4O4S
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1
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| 1 |
Ki = 3.8 nM
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CP0234129
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A2A
Show/Hide
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C19H26N4O4S
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1
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| 1 |
Ki = 3.9 nM
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CP0409948
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6-benzyl-2-(1,3-oxazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
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C16H12N4OS
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1
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| 1 |
Ki = 4.7 nM
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CP0559950
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4-fluoro-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C18H23FN4O3S
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1
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| 1 |
Ki = 4.9 nM
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CP0406021
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methyl 2-[acetyl-[2-[(4-fluorobenzoyl)amino]-4-methoxy-1,3-benzothiazol-7-yl]amino]acetate
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C20H18FN3O5S
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1
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| 1 |
Ki = 5 nM
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CP0095767
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6-[[(2S,6R)-2,6-dimethylpiperidin-1-yl]methyl]-2-(furan-2-yl)thieno[2,3-d]pyrimidin-4-amine
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C18H22N4OS
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1
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| 1 |
Ki = 5.3 nM
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CP0573418
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N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C18H24N4O3S
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1
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| 1 |
Ki = 6 nM
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CP0409950
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3-[4-amino-6-[(2-methoxyphenyl)methyl]thieno[2,3-d]pyrimidin-2-yl]benzonitrile
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C21H16N4OS
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1
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| 1 |
Ki = 6.2 nM
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CP0515569
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4-(2-fluoro-1-hydroxyethyl)-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C20H27FN4O4S
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1
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| 1 |
Ki = 6.4 nM
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CP0571394
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3-fluoro-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C18H23FN4O3S
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1
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| 1 |
Ki = 6.4 nM
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CP0853657
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6-(3,6-dihydro-2H-pyridin-1-ylmethyl)-2-furan-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H16N4OS
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1
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| 1 |
Ki = 6.5 nM
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CP0119411
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6-[(3,3-difluoropiperidin-1-yl)methyl]-2-(furan-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C16H16F2N4OS
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1
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| 1 |
Ki = 6.6 nM
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CP0396328
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6-[(2-chlorophenyl)methyl]-2-(4-methyl-1,3-thiazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H13ClN4S2
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1
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| 1 |
Ki = 6.9 nM
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CP0946683
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6-((2,5-dihydro-1H-pyrrol-1-yl)methyl)-2-(furan-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C15H14N4OS
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1
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| 1 |
Ki = 7.2 nM
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CP0378950
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3-[4-amino-6-[(2-fluorophenyl)methyl]thieno[2,3-d]pyrimidin-2-yl]benzonitrile
Show/Hide
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C20H13FN4S
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1
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| 1 |
Ki = 7.3 nM
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CP0864802
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6-(3,3-difluoro-pyrrolidin-1-ylmethyl)-2-furan-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H14F2N4OS
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1
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| 1 |
Ki = 8.7 nM
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CP0523778
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6-benzyl-2-(1,3-oxazol-5-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C16H12N4OS
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1
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| 1 |
Ki = 9 nM
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CP0864794
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2-(5-chloro-furan-2-yl)-6-(3,3-difluoro-piperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H15ClF2N4OS
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1
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| 1 |
Ki = 9.1 nM
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CP0864803
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2-(furan-2-yl)-6-(thiomorpholinomethyl)thieno-[2,3-d]pyrimidin-4-amine
Show/Hide
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C15H16N4OS2
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1
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| 1 |
Ki = 9.2 nM
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CP0513784
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4-(2-fluoroethyl)-4-hydroxy-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C20H27FN4O4S
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1
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| 1 |
Ki = 9.4 nM
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CP0498601
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6-[(2-fluorophenyl)methyl]-2-(4-methyl-1,3-thiazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H13FN4S2
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1
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| 1 |
Ki = 9.7 nM
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CP0877428
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2-(5-chloro-furan-2-yl)-6-(2,5-dihydro-pyrrol-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H13ClN4OS
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1
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| 1 |
Ki = 10 nM
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CP0901908
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6-(3-fluoro-pyrrolidin-1-ylmethyl)-2-furan-2-ylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H15FN4OS
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1
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| 1 |
Ki = 10.3 nM
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CP0378960
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6-[(2-methoxyphenyl)methyl]-2-(5-methylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H17N3O2S
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1
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| 1 |
Ki = 11 nM
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CP0849517
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2-(5-chloro-furan-2-yl)-6-(3,6-dihydro-2Hpyridin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H15ClN4OS
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1
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| 1 |
Ki = 11 nM
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CP0409949
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6-benzyl-2-(5-methylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H15N3OS
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1
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| 1 |
Ki = 11.1 nM
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CP0439130
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3-(4-amino-6-benzylthieno[2,3-d]pyrimidin-2-yl)benzonitrile
Show/Hide
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C20H14N4S
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1
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| 1 |
Ki = 11.4 nM
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CP0880224
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2-(5-bromofuran-2-yl)-6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H21BrN4OS
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1
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| 1 |
Ki = 12.1 nM
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CP0467092
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2-[5-(difluoromethyl)furan-2-yl]-6-[(2-methoxyphenyl)methyl]thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H15F2N3O2S
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1
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| 1 |
Ki = 13.1 nM
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CP0375733
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6-[(2-methoxyphenyl)methyl]-2-(4-methyl-1,3-thiazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H16N4OS2
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1
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| 1 |
Ki = 13.2 nM
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CP0850770
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3-[4-amino-6-(3,6-dihydro-2H-pyridin-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
Show/Hide
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C19H17N5S
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1
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| 1 |
Ki = 13.2 nM
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CP0377192
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N-[7-[acetyl(ethyl)amino]-4-chloro-1,3-benzothiazol-2-yl]-4-fluorobenzamide
Show/Hide
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C18H15ClFN3O2S
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1
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| 1 |
Ki = 15 nM
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CP0850771
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2-(5-chloro-furan-2-yl)-6-(3,3-difluoro-pyrrolidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H13ClF2N4OS
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1
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| 1 |
Ki = 15.9 nM
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CP0378957
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6-benzyl-2-(4-methyl-1,3-thiazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H14N4S2
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1
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| 1 |
Ki = 16.1 nM
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CP0959023
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6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)-2-(5-isopropylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C21H28N4OS
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1
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| 1 |
Ki = 17 nM
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CP0381544
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6-benzyl-2-pyrimidin-2-ylthieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H13N5S
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1
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| 1 |
Ki = 17.1 nM
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CP0377196
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-1H-pyrrole-3-carboxamide
Show/Hide
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C17H18N4O3S
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1
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| 1 |
Ki = 18 nM
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CP0901909
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6-(4-fluoro-piperidin-1-ylmethyl)-2-furan-2-ylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H17FN4OS
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1
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| 1 |
Ki = 19.7 nM
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CP0371895
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-fluorobenzamide
Show/Hide
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C19H18FN3O3S
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1
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| 1 |
Ki = 22 nM
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CP0881302
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2-(5-chloro-furan-2-yl)-6-pyrrolidin-1-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H15ClN4OS
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1
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| 1 |
Ki = 22.2 nM
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CP0853658
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2-(5-bromo-furan-2-yl)-6-pyrrolidin-1-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H15BrN4OS
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1
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| 1 |
Ki = 22.5 nM
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CP0555507
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4-(2-fluoroethoxy)-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C20H27FN4O4S
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1
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| 1 |
Ki = 23.9 nM
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CP0497575
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6-benzyl-2-[5-(difluoromethyl)furan-2-yl]thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H13F2N3OS
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1
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| 1 |
Ki = 25.2 nM
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CP0849518
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6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)-2-(5-ethylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C20H26N4OS
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1
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| 1 |
Ki = 25.2 nM
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CP0472456
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1-N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-N-(2-methoxyethyl)-4-N-methylbenzene-1,4-dicarboxamide
Show/Hide
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C24H28N4O5S
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1
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| 1 |
Ki = 26 nM
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CP0536867
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6-(4-amino-6-benzylthieno[2,3-d]pyrimidin-2-yl)pyridine-2-carbonitrile
Show/Hide
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C19H13N5S
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1
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| 1 |
Ki = 26 nM
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CP0958450
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2-(5-methyl-furan-2-yl)-6-pyrrolidin-1-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H18N4OS
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1
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| 1 |
Ki = 26.1 nM
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CP0475417
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-[(2-oxopyrrolidin-1-yl)methyl]benzamide
Show/Hide
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C24H26N4O4S
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1
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| 1 |
Ki = 27 nM
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CP0849566
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6-(azepan-1-ylmethyl)-2-(furan-2-yl)thieno[2,3-d]-pyrimidin-4-amine
Show/Hide
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C17H20N4OS
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1
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| 1 |
Ki = 27.6 nM
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CP0877429
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2-furan-2-yl-6-pyrrolidin-1-ylmethyl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H16N4OS
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1
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| 1 |
Ki = 28.1 nM
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CP0898624
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2-(5-(difluoromethyl)furan-2-yl)-6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H22F2N4OS
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1
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| 1 |
Ki = 28.6 nM
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CP0880225
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2-(5-methyl-furan-2-yl)-6-piperidin-1-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H20N4OS
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1
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| 1 |
Ki = 28.8 nM
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CP0438989
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4-fluoro-N-(7-(N-(3-hydroxypropyl)acetamido)-4-methoxybenzo[d]thiazol-2-yl)benzamide
Show/Hide
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C20H20FN3O4S
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1
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| 1 |
Ki = 29 nM
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CP0124542
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2-(furan-2-yl)-6-(morpholin-4-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C15H16N4O2S
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1
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| 1 |
Ki = 29 nM
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CP0381547
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6-benzyl-2-phenylthieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H15N3S
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1
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| 1 |
Ki = 29.8 nM
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CP0849562
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2-(5-bromo-furan-2-yl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H15BrN4O2S
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1
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| 1 |
Ki = 30 nM
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CP0880226
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2-(5-difluoromethyl-furan-2-yl)-6-morpholin-4-ylmethyl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H16F2N4O2S
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1
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| 1 |
Ki = 30.8 nM
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CP0409954
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2-(4-methyl-1,3-thiazol-2-yl)-6-(1-phenylethenyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H14N4S2
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1
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| 1 |
Ki = 31 nM
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CP0881294
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2-(5-methyl-furan-2-yl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H18N4O2S
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1
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| 1 |
Ki = 32.8 nM
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CP0512130
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4-methoxy-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C19H26N4O4S
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1
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| 1 |
Ki = 33 nM
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CP0850772
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6-azepan-1-ylmethyl-2-(5-chloro-furan-2-yl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H19ClN4OS
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1
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| 1 |
Ki = 33.4 nM
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CP0439004
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4-fluoro-N-(4-methoxy-7-(N-(2,2,2-trifluoroethyl)acetamido)benzo[d]thiazol-2-yl)benzamide
Show/Hide
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C19H15F4N3O3S
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1
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| 1 |
Ki = 35 nM
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CP0486347
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4-(2-fluoroethoxymethyl)-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C21H29FN4O4S
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1
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| 1 |
Ki = 35.1 nM
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CP0849519
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6-cyclopropylaminomethyl-2-furan-2-yl-thieno-[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C14H14N4OS
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1
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| 1 |
Ki = 36 nM
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CP0849564
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3-(4-amino-6-morpholin-4-ylmethyl-thieno[2,3-d]-pyrimidin-2-yl)-benzonitrile
Show/Hide
|
C18H17N5OS
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1
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| 1 |
Ki = 36.1 nM
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CP0913904
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2-(5-chloro-furan-2-yl)-6-(4-fluoro-piperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H16ClFN4OS
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1
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| 1 |
Ki = 36.7 nM
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CP0486348
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4-(1-fluoro-2-hydroxypropan-2-yl)-N-(4-methoxy-7-morpholin-4-yl-1,3-benzothiazol-2-yl)piperidine-1-carboxamide
Show/Hide
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C21H29FN4O4S
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1
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| 1 |
Ki = 37.9 nM
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CP0377195
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4-fluoro-N-(4-methoxy-7-(N-(2-methoxyethyl)acetamido)benzo[d]thiazol-2-yl)benzamide
Show/Hide
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C20H20FN3O4S
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1
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| 1 |
Ki = 38 nM
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CP0377190
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4-fluoro-N-(4-methoxy-7-(N-methylacetamido)benzo[d]thiazol-2-yl)benzamide
Show/Hide
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C18H16FN3O3S
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1
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| 1 |
Ki = 39 nM
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CP0880227
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3-[4-amino-6-(3,3-difluoro-piperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
Show/Hide
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C19H17F2N5S
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1
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| 1 |
Ki = 39 nM
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CP0378959
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2-(5-methylfuran-2-yl)-6-(1-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H17N3OS
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1
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| 1 |
Ki = 40.1 nM
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CP0377193
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-1-methylpyrazole-4-carboxamide
Show/Hide
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C17H19N5O3S
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1
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| 1 |
Ki = 41 nM
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CP0467090
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6-benzyl-2-(3-fluorophenyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H14FN3S
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1
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| 1 |
Ki = 42 nM
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CP0864797
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2-(5-difluoromethyl-furan-2-yl)-6-(4-fluoropiperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H17F3N4OS
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1
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| 1 |
Ki = 42.2 nM
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CP0946688
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2-(5-difluoromethyl-furan-2-yl)-6-(3,3-difluoropiperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H16F4N4OS
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1
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| 1 |
Ki = 43.2 nM
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CP0898592
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2-(5-chloro-furan-2-yl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H15ClN4O2S
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1
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| 1 |
Ki = 45.4 nM
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CP0439007
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-(methanesulfonamido)benzamide
Show/Hide
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C20H22N4O5S2
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1
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| 1 |
Ki = 46 nM
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CP0381548
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6-benzyl-2-(5-ethylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H17N3OS
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1
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| 1 |
Ki = 49 nM
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CP0946689
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6-(4,4-difluoro-piperidin-1-ylmethyl)-2-furan-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C16H16F2N4OS
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1
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| 1 |
Ki = 49.6 nM
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CP0454301
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4-cyano-N-(7-(N-ethylacetamido)-4-methoxybenzo[d]thiazol-2-yl)benzamide
Show/Hide
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C20H18N4O3S
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1
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| 1 |
Ki = 50 nM
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CP0856398
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3-(4-amino-6-thiomorpholin-4-ylmethyl-thieno-[2,3-d]pyrimidin-2-yl)-benzonitrile
Show/Hide
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C18H17N5S2
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1
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| 1 |
Ki = 50.9 nM
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CP0164878
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-2-methylpyrazole-3-carboxamide
Show/Hide
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C17H19N5O3S
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1
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| 1 |
Ki = 51 nM
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CP0849555
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3-[4-amino-6-(4-fluoro-piperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
Show/Hide
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C19H18FN5S
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1
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| 1 |
Ki = 54.4 nM
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CP0946682
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6-diethylaminomethyl-2-furan-2-yl-thieno[2,3-d]-pyrimidin-4-ylamine
Show/Hide
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C15H18N4OS
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1
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| 1 |
Ki = 55.5 nM
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CP0467089
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6-benzyl-2-(2-methyl-1,3-thiazol-4-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H14N4S2
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1
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| 1 |
Ki = 57 nM
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CP0377191
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N-[7-[acetyl(difluoromethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-fluorobenzamide
Show/Hide
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C18H14F3N3O3S
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1
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| 1 |
Ki = 61 nM
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CP0439086
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3-[4-amino-6-(1-phenylethenyl)thieno[2,3-d]pyrimidin-2-yl]benzonitrile
Show/Hide
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C21H14N4S
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1
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| 1 |
Ki = 63.4 nM
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CP0849556
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3-(4-amino-6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)thieno[2,3-d]pyrimidin-2-yl)benzonitrile
Show/Hide
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C21H23N5S
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1
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| 1 |
Ki = 64.6 nM
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CP0371897
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-pyrazol-1-ylbenzamide
Show/Hide
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C22H21N5O3S
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1
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| 1 |
Ki = 66 nM
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CP0397691
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2-(5-methylfuran-2-yl)-6-phenylthieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H13N3OS
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1
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| 1 |
Ki = 67.3 nM
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CP0467088
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6-benzyl-2-pyridin-4-ylthieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H14N4S
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1
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| 1 |
Ki = 67.3 nM
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CP0417790
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-(pyrrolidine-1-carbonyl)benzamide
Show/Hide
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C24H26N4O4S
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1
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| 1 |
Ki = 68 nM
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CP0436825
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-[[methyl(methylsulfonyl)amino]methyl]benzamide
Show/Hide
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C22H26N4O5S2
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1
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| 1 |
Ki = 71 nM
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CP0472455
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-(morpholine-4-carbonyl)benzamide
Show/Hide
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C24H26N4O5S
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1
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| 1 |
Ki = 76 nM
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CP0425918
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-imidazol-1-ylbenzamide
Show/Hide
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C22H21N5O3S
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1
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| 1 |
Ki = 77 nM
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CP0856392
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2-(5-ethyl-furan-2-yl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H20N4O2S
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1
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| 1 |
Ki = 78.9 nM
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CP0849511
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4-[4-amino-6-(2,5-dihydro-pyrrol-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
Show/Hide
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C18H15N5S
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1
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| 1 |
Ki = 79.2 nM
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CP0438976
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-(tetrazol-1-yl)benzamide
Show/Hide
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C20H19N7O3S
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1
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| 1 |
Ki = 80 nM
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CP0856393
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3-[4-amino-6-(2,5-dihydro-pyrrol-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
Show/Hide
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C18H15N5S
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1
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| 1 |
Ki = 83.5 nM
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CP0438977
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4-N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-1-N-methylbenzene-1,4-dicarboxamide
Show/Hide
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C21H22N4O4S
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1
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| 1 |
Ki = 84 nM
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CP0472457
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-(4-methylpiperazine-1-carbonyl)benzamide
Show/Hide
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C25H29N5O4S
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1
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| 1 |
Ki = 89 nM
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CP0849560
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6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)-2-(4-methylthiazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H23N5S2
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1
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| 1 |
Ki = 89.1 nM
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CP0438975
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-methylsulfonylbenzamide
Show/Hide
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C20H21N3O5S2
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1
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| 1 |
Ki = 92 nM
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CP0898593
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6-(3,3-difluoro-piperidin-1-ylmethyl)-2-(3-methoxy-phenyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C19H20F2N4OS
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1
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| 1 |
Ki = 97.7 nM
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CP0377194
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4-fluoro-N-(7-(N-(2-hydroxyethyl)acetamido)-4-methoxybenzo[d]thiazol-2-yl)benzamide
Show/Hide
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C19H18FN3O4S
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1
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| 1 |
Ki = 98 nM
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CP0371900
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N-[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-(piperidine-1-carbonyl)benzamide
Show/Hide
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C25H28N4O4S
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1
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| 1 |
Ki = 100 nM
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CP0378958
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2-(4-methyl-1,3-thiazol-2-yl)-6-(1-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H16N4S2
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1
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| 1 |
Ki = 100 nM
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CP0396327
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2-(4-methyl-1,3-thiazol-2-yl)-6-(1-phenylcyclopropyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H16N4S2
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1
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| 1 |
Ki = 107 nM
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CP0409953
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2-(5-methylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C11H9N3OS
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1
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| 1 |
Ki = 109 nM
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CP0849557
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6-pyrrolidin-1-ylmethyl-2-thiophen-2-yl-thieno-[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H16N4S2
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1
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| 1 |
Ki = 110 nM
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CP0849558
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2-(3-fluoro-phenyl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H17FN4OS
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1
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| 1 |
Ki = 110 nM
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CP0898627
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2-(5-cyclopropylfuran-2-yl)-6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C21H26N4OS
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1
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| 1 |
Ki = 110 nM
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CP0409951
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6-benzyl-2-(3-methoxyphenyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C20H17N3OS
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1
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| 1 |
Ki = 118 nM
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CP0881303
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2-(3-chloro-phenyl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H17ClN4OS
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1
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| 1 |
Ki = 120 nM
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CP0901910
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6-morpholin-4-ylmethyl-2-thiophen-2-yl-thieno-[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H16N4OS2
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1
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| 1 |
Ki = 125 nM
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CP0860171
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6-(((2R,6S)-2,6-dimethylpiperidin-1-yl)methyl)-2-(isoxazol-3-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C17H21N5OS
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1
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| 1 |
Ki = 130 nM
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CP0856402
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6-dimethylaminomethyl-2-furan-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C13H14N4OS
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1
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| 1 |
Ki = 140 nM
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CP0856394
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3-(4-amino-6-(((2S,6R)-2,6-dimethylmorpholino)methyl)thieno[2,3-d]pyrimidin-2-yl)benzonitrile
Show/Hide
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C20H21N5OS
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1
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| 1 |
Ki = 150 nM
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CP0371893
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N-[7-[acetyl-(2-amino-2-oxoethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-fluorobenzamide
Show/Hide
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C19H17FN4O4S
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1
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| 1 |
Ki = 160 nM
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CP0498600
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6-benzyl-2-(5-propan-2-ylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C20H19N3OS
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1
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| 1 |
Ki = 168 nM
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CP0436824
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methyl 4-[[7-[acetyl(ethyl)amino]-4-methoxy-1,3-benzothiazol-2-yl]carbamoyl]benzoate
Show/Hide
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C21H21N3O5S
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1
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| 1 |
Ki = 170 nM
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CP0864793
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6-cyclohexylaminomethyl-2-furan-2-yl-thieno-[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H20N4OS
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1
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| 1 |
Ki = 170 nM
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CP0523782
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6-benzyl-2-(6-chloropyridin-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H13ClN4S
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1
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| 1 |
Ki = 173 nM
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CP0881295
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4-[4-amino-6-(3,6-dihydro-2H-pyridin-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
Show/Hide
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C19H17N5S
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1
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| 1 |
Ki = 180 nM
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CP0849547
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6-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-2-(5-methyl-furan-2-yl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C21H20N4OS
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1
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| 1 |
Ki = 200 nM
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CP0381546
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2-(5-methylfuran-2-yl)-6-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H17N3OS
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1
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| 1 |
Ki = 203 nM
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CP0556758
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2,6-diphenylthieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H13N3S
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1
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| 1 |
Ki = 207 nM
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CP0856403
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2-(4-methyl-thiazol-2-yl)-6-morpholin-4-ylmethyl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H17N5OS2
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1
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| 1 |
Ki = 210 nM
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CP0409947
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6-benzyl-2-pyridin-3-ylthieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C18H14N4S
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1
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| 1 |
Ki = 215 nM
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CP0515279
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3-[4-amino-6-(1-phenylcyclopropyl)thieno[2,3-d]pyrimidin-2-yl]benzonitrile
Show/Hide
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C22H16N4S
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1
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| 1 |
Ki = 222 nM
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CP0867275
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1-(4-amino-2-furan-2-yl-thieno[2,3-d]pyrimidin-6-ylmethyl)-piperidin-4-one
Show/Hide
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C16H16N4O2S
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1
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| 1 |
Ki = 230 nM
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CP0849559
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6-(2,5-dihydro-pyrrol-1-ylmethyl)-2-oxazol-4-ylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C14H13N5OS
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1
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| 1 |
Ki = 238 nM
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CP0849568
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6-((2,5-dihydro-1H-pyrrol-1-yl)methyl)-2-(oxazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C14H13N5OS
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1
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| 1 |
Ki = 240 nM
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CP0856395
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6-(3,6-dihydro-2H-pyridin-1-ylmethyl)-2-oxazol-4-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C15H15N5OS
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1
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| 1 |
Ki = 240 nM
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CP0856401
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6-((5,6-dihydropyridin-1(2H)-yl)methyl)-2-(oxazol-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C15H15N5OS
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1
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| 1 |
Ki = 240 nM
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CP0281180
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N-(7-acetamido-4-methoxy-1,3-benzothiazol-2-yl)-4-fluorobenzamide
Show/Hide
|
C17H14FN3O3S
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1
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| 1 |
Ki = 250 nM
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CP0898636
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6-morpholin-4-ylmethyl-2-thiazol-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C14H15N5OS2
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1
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| 1 |
Ki = 250 nM
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CP0397690
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6-benzyl-2-(5-cyclopropylfuran-2-yl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C20H17N3OS
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1
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| 1 |
Ki = 263 nM
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CP0856396
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1-(4-amino-2-furan-2-yl-thieno[2,3-d]pyrimidin-6-ylmethyl)-piperidin-4-ol
Show/Hide
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C16H18N4O2S
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1
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| 1 |
Ki = 300 nM
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CP0910460
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6-(4-fluoro-piperidin-1-ylmethyl)-2-(3-methoxyphenyl)-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
|
C19H21FN4OS
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1
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| 1 |
Ki = 300 nM
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CP0381545
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5-(4-amino-6-benzylthieno[2,3-d]pyrimidin-2-yl)furan-2-carbonitrile
Show/Hide
|
C18H12N4OS
|
1
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| 1 |
Ki = 304 nM
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CP0438988
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4-fluoro-N-(4-methoxy-7-(N-(2-(methylamino)-2-oxoethyl)acetamido)benzo[d]thiazol-2-yl)benzamide
Show/Hide
|
C20H19FN4O4S
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1
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| 1 |
Ki = 330 nM
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CP0378956
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3-[4-amino-6-(1-phenylethyl)thieno[2,3-d]pyrimidin-2-yl]benzonitrile
Show/Hide
|
C21H16N4S
|
1
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| 1 |
Ki = 340 nM
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CP0856397
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2-benzofuran-2-yl-6-(4-fluoropiperdin-1-ylmethyl)thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C20H19FN4OS
|
1
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| 1 |
Ki = 350 nM
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CP0867274
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2-(3,5-difluoro-phenyl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
|
C17H16F2N4OS
|
1
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| 1 |
Ki = 350 nM
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CP0849561
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2-(3,4-difluoro-phenyl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C17H16F2N4OS
|
1
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| 1 |
Ki = 360 nM
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CP0946690
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6-morpholin-4-ylmethyl-2-oxazol-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
Show/Hide
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C14H15N5O2S
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1
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| 1 |
Ki = 360 nM
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CP0515571
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N-[4-(2-fluoroethoxy)-7-morpholin-4-yl-1,3-benzothiazol-2-yl]-4-hydroxy-4-methylpiperidine-1-carboxamide
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C20H27FN4O4S
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1
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| 1 |
Ki = 361 nM
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CP0853664
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2-(3-methoxy-phenyl)-6-morpholin-4-ylmethylthieno[2,3-d]pyrimidin-4-ylamine
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C18H20N4O2S
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1
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| 1 |
Ki = 370 nM
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CP0946686
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4-[4-amino-6-(4-fluoro-piperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
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C19H18FN5S
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1
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| 1 |
Ki = 390 nM
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CP0439006
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N-[7-[acetyl-[2-(dimethylamino)-2-oxoethyl]amino]-4-methoxy-1,3-benzothiazol-2-yl]-4-fluorobenzamide
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C21H21FN4O4S
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1
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| 1 |
Ki = 480 nM
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CP0467099
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2-phenylthieno[2,3-d]pyrimidin-4-amine
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C12H9N3S
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1
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| 1 |
Ki = 500 nM
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CP0381543
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6-benzyl-2-(1-methylimidazol-4-yl)thieno[2,3-d]pyrimidin-4-amine
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C17H15N5S
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1
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| 1 |
Ki = 539 nM
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CP0498598
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6-benzyl-2-pyridin-2-ylthieno[2,3-d]pyrimidin-4-amine
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C18H14N4S
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1
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| 1 |
Ki = 594 nM
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CP0958449
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2-(5-difluoromethyl-furan-2-yl)-6-(4,4-difluoropiperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-4-ylamine
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C17H16F4N4OS
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1
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| 1 |
Ki = 610 nM
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CP0499311
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6-benzyl-2-(oxolan-2-yl)thieno[2,3-d]pyrimidin-4-amine
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C17H17N3OS
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1
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| 1 |
Ki = 683 nM
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CP0849563
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2-(5-cyclopropyl-furan-2-yl)-6-morpholin-4-ylmethyl-thieno[2,3-d]pyrimidin-4-ylamine
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C18H20N4O2S
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1
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| 1 |
Ki = 960 nM
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CP0856400
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6-(morpholinomethyl)-2-phenylthieno[2,3-d]-pyrimidin-4-amine
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C17H18N4OS
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1
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| 1 |
Ki = 995 nM
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CP0946687
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2-isoxazol-3-yl-6-morpholin-4-ylmethyl-thieno-[2,3-d]pyrimidin-4-ylamine
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C14H15N5O2S
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1
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| 1 |
Ki = 1010 nM
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CP0467098
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6-benzyl-2-[3-(trifluoromethyl)phenyl]thieno[2,3-d]pyrimidin-4-amine
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C20H14F3N3S
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1
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| 1 |
Ki = 1016 nM
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CP0849565
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2-[4-amino-6-(4-fluoro-piperidin-1-ylmethyl)-thieno[2,3-d]pyrimidin-2-yl]-benzonitrile
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C19H18FN5S
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1
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| 1 |
Ki = 1030 nM
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CP0910459
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6-((2,5-dihydro-1H-pyrrol-1-yl)methyl)-2-(3-(trifluoromethyl)phenyl)thieno[2,3-d]pyrimidin-4-amine
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C18H15F3N4S
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1
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| 1 |
Ki = 1070 nM
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CP0446639
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2-(N-(2-(4-fluorobenzamido)-4-methoxybenzo[d]thiazol-7-yl)acetamido)acetic acid
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C19H16FN3O5S
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1
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| 1 |
Ki = 2200 nM
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CP0849570
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3-(4-amino-6-((4-fluoropiperidin-1-yl)methyl)thieno[2,3-d]pyrimidin-2-yl)-N,N-dimethylbenzamide
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C21H24FN5OS
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1
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| 1 |
Ki = 2250 nM
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CP0849567
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6-((4-fluoropiperidin-1-yl)methyl)-2-(3-nitrophenyl)thieno[2,3-d]pyrimidin-4-amine
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C18H18FN5O2S
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1
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| 1 |
Ki = 3760 nM
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CP0849569
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6-((4-fluoropiperidin-1-yl)methyl)-2-(3-(methylsulfonyl)phenyl)thieno[2,3-d]pyrimidin-4-amine
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C19H21FN4O2S2
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1
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| 1 |
Ki > 10000 nM
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CP0867276
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3-(4-amino-6-pyrrolidin-1-ylmethyl-thieno[2,3-d]-pyrimidin-2-yl)-benzonitrile
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C18H17N5S
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1
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| 1 |
Ki > 10000 nM
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CP0898637
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6-((4-fluoropiperidin-1-yl)methyl)-2-(3-(trifluoromethyl)phenyl)thieno[2,3-d]pyrimidin-4-amine
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C19H18F4N4S
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1
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| 1 |
Ki > 10000 nM
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CP0910461
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6-((4-fluoropiperidin-1-yl)methyl)-2-(4-(trifluoromethyl)phenyl)thieno[2,3-d]pyrimidin-4-amine
Show/Hide
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C19H18F4N4S
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1
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| 1 |
Ki > 10000 nM
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CP0910462
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6-((4-fluoropiperidin-1-yl)methyl)-2-(2-(trifluoromethyl)phenyl)thieno[2,3-d]pyrimidin-4-amine
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C19H18F4N4S
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1
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| 1 |
Ki > 10000 nM
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CP0467097
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5-(4-amino-6-benzylthieno[2,3-d]pyrimidin-2-yl)pyridine-3-carbonitrile
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C19H13N5S
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1
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| 1 |
Ki > 168 nM
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CP0409946
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2-phenyl-6-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
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C20H17N3S
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1
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| 1 |
Ki > 1000 nM
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CP0864798
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2-(5-isopropyl-furan-2-yl)-6-morpholin-4-ylmethyl-thieno[2,3-d]pyrimidin-4-ylamine
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C18H22N4O2S
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1
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| 1 |
Ki > 1360 nM
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