Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT06350 , Taste receptor type 2 member 46
Gene Name TAS2R46
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P59540
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT06350
 
Compound ID Compound Name Compound Formula
CP0928920
3-Betahydroxy dihydro costunolide acetate
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C17H24O4
 1
1
EC50 = 1100 nM
   TI
   LI
   LO
   TS
CP0938746
3-beta-hydroxy dihydro costunolide acetate
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C17H24O4
 1
1
EC50 = 1100 nM
   TI
   LI
   LO
   TS
CP0866307
3-beta-hydroxy dihydro costunolide
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C15H22O3
 8
1
EC50 = 2740 nM
   TI
   LI
   LO
   TS
2
EC50 = 5390 nM
   TI
   LI
   LO
   TS
3
EC50 = 21720 nM
   TI
   LI
   LO
   TS
4
IC50 = 4810 nM
   TI
   LI
   LO
   TS
5
IC50 = 4930 nM
   TI
   LI
   LO
   TS
6
IC50 = 6780 nM
   TI
   LI
   LO
   TS
7
IC50 = 14100 nM
   TI
   LI
   LO
   TS
8
IC50 = 15300 nM
   TI
   LI
   LO
   TS
CP0964772
dihydro costunolide
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C15H22O2
 1
1
EC50 = 8300 nM
   TI
   LI
   LO
   TS
CP0901635
Dihydro costunolide
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C15H22O2
 1
1
EC50 = 8300 nM
   TI
   LI
   LO
   TS
CP0051720
(3aS,6E,10E,11aR)-6,10-dimethyl-3-methylidene-3a,4,5,8,9,11a-hexahydrocyclodeca[b]furan-2-one
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C15H20O2
 1
1
EC50 = 8600 nM
   TI
   LI
   LO
   TS
CP0970191
Costunolide
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C15H20O2
 1
1
EC50 = 8600 nM
   TI
   LI
   LO
   TS
CP0850084
3-Betahydroxy dihydro costunolide
   Show/Hide
C15H22O3
 5
1
IC50 = 4810 nM
   TI
   LI
   LO
   TS
2
IC50 = 4930 nM
   TI
   LI
   LO
   TS
3
IC50 = 6780 nM
   TI
   LI
   LO
   TS
4
IC50 = 14100 nM
   TI
   LI
   LO
   TS
5
IC50 = 15300 nM
   TI
   LI
   LO
   TS
CP0850085
3-betahydroxy pelenolide
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C15H24O3
 5
1
IC50 = 22900 nM
   TI
   LI
   LO
   TS
2
IC50 = 44500 nM
   TI
   LI
   LO
   TS
3
IC50 = 51400 nM
   TI
   LI
   LO
   TS
4
IC50 = 57800 nM
   TI
   LI
   LO
   TS
5
IC50 = 84900 nM
   TI
   LI
   LO
   TS
CP0862834
3-beta hydroxy pelenolide
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C15H24O3
 5
1
IC50 = 22900 nM
   TI
   LI
   LO
   TS
2
IC50 = 44500 nM
   TI
   LI
   LO
   TS
3
IC50 = 51400 nM
   TI
   LI
   LO
   TS
4
IC50 = 57800 nM
   TI
   LI
   LO
   TS
5
IC50 = 84900 nM
   TI
   LI
   LO
   TS
CP0963570
3-keto dihydro costunolide
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C15H20O3
 1
1
IC50 = 97800 nM
   TI
   LI
   LO
   TS
CP0963444
3-Keto dihydro costunolide
   Show/Hide
C15H20O3
 1
1
IC50 = 97800 nM
   TI
   LI
   LO
   TS