Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01279 , Adenosine receptor A3
Gene Name ADORA3
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P0DMS8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01279
 
Compound ID Compound Name Compound Formula
CP0421485
2,4-Bis-n-propyl-4,9-dihydro-5-n-propyloxy-2,4,7,9-tetraaza-fluorene-1,3-dione
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C18H24N4O3
 1
1
Ki = 3.82 nM
   TI
   LI
   LO
   TS
CP0372084
2,4-dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione
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C11H12N4O2
 1
1
Ki = 13.9 nM
   TI
   LI
   LO
   TS
CP0398283
2,4-Dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione
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C11H10N4O2
 1
1
Ki = 13.9 nM
   TI
   LI
   LO
   TS
CP0421479
2,4-bis-n-propyl-4,9-dihydro-2,4,7,-9-tetraaza-fluorene-1,3-dione
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C15H18N4O2
 1
1
Ki = 16.8 nM
   TI
   LI
   LO
   TS
CP0039348
(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
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C12H16N6O4
 2
1
Ki = 20 nM
   TI
   LI
   LO
   TS
2
Ki = 17700 nM
   TI
   LI
   LO
   TS
CP0422919
2,4-Bis-n-propyl-4,9-dihydro-7-n-propyloxy-2,4,5,-9-tetraaza-fluorene-1,3-dione
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C18H24N4O3
 1
1
Ki = 209 nM
   TI
   LI
   LO
   TS
CP0496657
2,4-Bis-n-propyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione
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C15H18N4O2
 1
1
Ki = 290 nM
   TI
   LI
   LO
   TS
CP0372085
2,5,9-trimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione
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C12H14N4O2
 1
1
Ki = 332 nM
   TI
   LI
   LO
   TS
CP0371882
2,4-dimethyl-4,9-dihydro-2,4,5,9-tetraaza-fluorene-1,3-dione
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C11H12N4O2
 1
1
Ki = 526 nM
   TI
   LI
   LO
   TS
CP0398284
2,4-Dimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione
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C11H10N4O2
 1
1
Ki = 526 nM
   TI
   LI
   LO
   TS
CP0371881
5,7-dibromo-9H-pyrido[3,4-b]indol-6-ol
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C11H6Br2N2O
 1
1
Ki = 2050 nM
   TI
   LI
   LO
   TS
CP0424860
2,4,9-trimethyl-4,9-dihydro-2,4,7,9-tetraaza-fluorene-1,3-dione
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C12H14N4O2
 1
1
Ki = 3190 nM
   TI
   LI
   LO
   TS
CP0534845
8-Hydroxy-7,9-dimethyl-delta-carboline
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C13H12N2O
 1
1
Ki = 4430 nM
   TI
   LI
   LO
   TS
CP0437932
8-Hydroxy-5,7,9-trimethyl-delta-carboline
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C14H14N2O
 1
1
Ki = 13300 nM
   TI
   LI
   LO
   TS
CP0437930
6-Hydroxy-5,7-dimethyl-beta-carboline
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C13H12N2O
 1
1
Ki = 17700 nM
   TI
   LI
   LO
   TS
CP0894539
6-Hydroxy-2,5,7-trimethyl-9H-beta-carbolin-2-ium
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C14H15IN2O
 1
1
Ki = 29700 nM
   TI
   LI
   LO
   TS
CP0437931
6-Hydroxy-5,7,9-trimethyl-beta-carboline
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C14H14N2O
 1
1
Ki = 43400 nM
   TI
   LI
   LO
   TS
CP0043620
1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
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C8H10N4O2
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS
CP0910732
6-Hydroxy-2,5,7,9-tetramethyl-9H-beta-carbolin-2-ium
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C15H17IN2O
 1
1
Ki > 100000 nM
   TI
   LI
   LO
   TS