Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01154 , Mineralocorticoid receptor
Gene Name NR3C2
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID P08235
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01154
 
Compound ID Compound Name Compound Formula
CP0476139
[3-methyl-4-[2-(8-methyl-3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]phenyl] acetate
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C20H21NO4
 1
1
IC50 = 1.3 nM
   TI
   LI
   LO
   TS
CP0457610
[3-methyl-4-[2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]phenyl] acetate
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C19H19NO4
 1
1
IC50 < 2 nM
   TI
   LI
   LO
   TS
CP0414462
[4-[2-(2-methylphenyl)ethyl]pyridin-2-yl]urea
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C15H17N3O
 1
1
IC50 = 19 nM
   TI
   LI
   LO
   TS
CP0403354
US8722709, 48
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C15H16FN3O
 1
1
IC50 = 31 nM
   TI
   LI
   LO
   TS
CP0548733
US8722709, 32
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C16H19N3O
 1
1
IC50 = 43 nM
   TI
   LI
   LO
   TS
CP0558679
US8722709, 31
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C20H19N3O
 1
1
IC50 = 44 nM
   TI
   LI
   LO
   TS
CP0548734
5-methyl-6-(3-methylphenyl)-4H-1,4-benzoxazin-3-one
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C16H15NO2
 1
1
IC50 = 47 nM
   TI
   LI
   LO
   TS
CP0723935
(S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carboxamide
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C21H22N4O3
 1
1
IC50 = 58 nM
   TI
   LI
   LO
   TS
CP0468737
[6-[2-(2-methoxyphenyl)ethyl]pyridin-2-yl]urea
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C15H17N3O2
 1
1
IC50 = 97 nM
   TI
   LI
   LO
   TS
CP0403355
US8722709, 16
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C15H12ClN5O
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0393731
US8722709, 28
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C15H17N3O
 1
1
IC50 = 2800 nM
   TI
   LI
   LO
   TS