Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT01071 , Tyrosine-protein kinase ABL1
Gene Name ABL1
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P00519
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT01071
 
Compound ID Compound Name Compound Formula
CP0018808
4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide
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C23H28Cl2N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0130748
4-(cyclohexylamino)-2-[(2,5-dibromo-4-methylphenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide
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C25H32Br2N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0313025
4-(cyclopentylamino)-2-[(2,5-dibromo-4-methylphenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide
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C24H30Br2N6O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0534020
2-[(4-chlorophenyl)methyl-ethylamino]-4-(cyclopentylamino)-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
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C26H35ClN6O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0559075
4-(cyclopentylamino)-2-[(2,4-dichlorophenyl)methylamino]-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
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C24H30Cl2N6O2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0355448
5-amino-N-[[4-[[(2S)-4-cyclohexyl-1-(ethylamino)-1-oxobutan-2-yl]carbamoyl]phenyl]methyl]-1-phenylpyrazole-4-carboxamide
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C30H38N6O3
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0030881
SR-302
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C32H42N6O5S
 1
1
IC50 > 25000 nM
   TI
   LI
   LO
   TS