Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT00975 , Dipeptidyl peptidase 8
Gene Name DPP8
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID Q6V1X1
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT00975
 
Compound ID Compound Name Compound Formula
CP0067537
(R)-1-((S)-2-amino-3-methylbutanoyl)pyrrolidin-2-ylboronic acid
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C9H19BN2O3
 1
1
Ki = 1.5 nM
   TI
   LI
   LO
   TS
CP0139059
(R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic acid
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C7H15BN2O3
 1
1
Ki = 2 nM
   TI
   LI
   LO
   TS
CP0231981
(R)-1-(2-aminoacetyl)pyrrolidin-2-ylboronic acid
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C6H13BN2O3
 1
1
Ki = 3.1 nM
   TI
   LI
   LO
   TS
CP0229143
(S)-4-amino-5-((R)-2-boronopyrrolidin-1-yl)-5-oxopentanoic acid
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C9H17BN2O5
 1
1
Ki = 11 nM
   TI
   LI
   LO
   TS
CP0099440
(R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic acid
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C7H17BN2O3
 1
1
Ki = 96 nM
   TI
   LI
   LO
   TS
CP0519860
(R)-1-((S)-2,5-diamino-5-oxopentanamido)ethylboronic acid
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C7H16BN3O4
 1
1
Ki = 140 nM
   TI
   LI
   LO
   TS
CP0423068
(S)-4-amino-5-((R)-1-boronoethylamino)-5-oxopentanoic acid
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C7H15BN2O5
 1
1
Ki = 880 nM
   TI
   LI
   LO
   TS
CP0511291
(R)-1-((S)-2-acetamido-3-methylbutanoyl)pyrrolidin-2-ylboronic acid
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C11H21BN2O4
 1
1
Ki = 8400 nM
   TI
   LI
   LO
   TS