Brief Information of the Cell Line and Protein
Cell Line ID: CL000025 , HEK-293T
Synonyms
Hek293T
HEK-293T
HEK 293T
HEK-293-T
HEK 293 T
293-T
293 T
293T
Human Embryonic Kidney 293T
293tsA1609neo
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0063
Protein ID: PT00933 , Macrophage-stimulating protein receptor
Gene Name MST1R
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID Q04912
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000025  Protein ID: PT00933
 
Compound ID Compound Name Compound Formula
CP0850979
N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-4-yl)thieno[3,2-b]pyridin-7-yloxy)phenyl)-1-phenyl-2-(trifluoromethyl)-1H-pyrrole-3-carboxamide
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C29H19F4N5O2S
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0046759
N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide
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C28H18F4N6O2S
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0413130
N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)imidazole-4-carboxamide
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C28H18F4N6O2S
 1
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
CP0195506
N-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluorophenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide
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C28H20F4N4O4
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0395262
N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-5-(trifluoromethyl)triazole-4-carboxamide
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C27H17F4N7O2S
 1
1
IC50 = 17 nM
   TI
   LI
   LO
   TS
CP0420379
N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-(4-fluorophenyl)-5-(trifluoromethyl)pyrazole-4-carboxamide
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C28H17F5N6O2S
 1
1
IC50 = 44 nM
   TI
   LI
   LO
   TS
CP0413129
N-[3-fluoro-4-[2-(1-methylimidazol-4-yl)thieno[3,2-b]pyridin-7-yl]oxyphenyl]-1-phenyl-3-(trifluoromethyl)pyrazole-4-carboxamide
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C28H18F4N6O2S
 1
1
IC50 = 95 nM
   TI
   LI
   LO
   TS
CP0686403
N-(3-fluoro-4-(2-(1-methyl-1H-imidazol-4-yl)thieno[3,2-b]pyridin-7-yloxy)phenyl)-N-methyl-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
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C29H20F4N6O2S
 1
1
IC50 = 580 nM
   TI
   LI
   LO
   TS