Compound ID |
Compound Name |
Compound Formula |
CP0008147
|
methyl 4-methoxy-3-[[2-piperidin-1-yl-5-(trifluoromethyl)phenyl]sulfamoyl]benzoate
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|
C21H23F3N2O5S
|
1
|
1 |
AC50 = 42000 nM
|
|
|
CP0662662
|
(S)-2-((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-ylcarbamoyl)-4-methylpentyl((R)-1-amino-3-phenylpropyl)phosphinic acid
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|
C27H37N4O4P
|
2
|
1 |
IC50 = 11 nM
|
|
|
2 |
IC50 = 80 nM
|
|
|
CP0473585
|
[(2S)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]pent-4-ynyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C24H30N3O4P
|
1
|
1 |
IC50 = 37 nM
|
|
|
CP0458633
|
[(2S)-2-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C25H36N3O5P
|
1
|
1 |
IC50 = 55 nM
|
|
|
CP0517735
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(4-hydroxyphenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C31H35N4O6P
|
1
|
1 |
IC50 = 56 nM
|
|
|
CP0519441
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(2-hydroxyphenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C31H35N4O6P
|
1
|
1 |
IC50 = 83 nM
|
|
|
CP0447357
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C32H37N4O6P
|
1
|
1 |
IC50 = 84 nM
|
|
|
CP0493458
|
[(2S)-2-[[(2S)-1-amino-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C19H32N3O4P
|
1
|
1 |
IC50 = 96 nM
|
|
|
CP0481975
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[(3,5-diphenylphenyl)methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C40H42N3O4P
|
1
|
1 |
IC50 = 105 nM
|
|
|
CP0560309
|
[(2S)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C25H36N3O4P
|
1
|
1 |
IC50 = 109 nM
|
|
|
CP0473582
|
[(2S)-2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C22H38N3O4P
|
1
|
1 |
IC50 = 118 nM
|
|
|
CP0493459
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C31H34ClN4O5P
|
1
|
1 |
IC50 = 123 nM
|
|
|
CP0473583
|
[(2S)-2-[[(2S)-1-amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C22H34N5O4P
|
1
|
1 |
IC50 = 128 nM
|
|
|
CP0447354
|
[(2S)-2-[[(2S)-1-amino-3-hydroxy-1-oxopropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C19H32N3O5P
|
1
|
1 |
IC50 = 129 nM
|
|
|
CP0493460
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C32H37N4O6P
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0538815
|
[(1R)-1-amino-3-phenylpropyl]-[(2S)-2-[(2S)-2-carbamoylpyrrolidine-1-carbonyl]-4-methylpentyl]phosphinic acid
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|
C21H34N3O4P
|
1
|
1 |
IC50 = 144 nM
|
|
|
CP0541454
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-oxo-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]propyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C31H35N4O5P
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0534737
|
[(2S)-2-[[(2R)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4-methylpentyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C25H36N3O4P
|
1
|
1 |
IC50 = 211 nM
|
|
|
CP0473580
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C32H37N4O6P
|
1
|
1 |
IC50 = 217 nM
|
|
|
CP0534738
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(3-chlorophenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C31H34ClN4O5P
|
1
|
1 |
IC50 = 225 nM
|
|
|
CP0418669
|
(2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acid
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|
C24H29N5O4
|
1
|
1 |
IC50 = 237 nM
|
|
|
CP0473584
|
(4S)-5-amino-4-[[(2S)-2-[[[(1R)-1-amino-3-phenylpropyl]-hydroxyphosphoryl]methyl]-4-methylpentanoyl]amino]-5-oxopentanoic acid
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|
C21H34N3O6P
|
1
|
1 |
IC50 = 243 nM
|
|
|
CP0487808
|
[(2S)-2-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C32H42N3O4P
|
1
|
1 |
IC50 = 246 nM
|
|
|
CP0550440
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-(3,4,5-trifluorophenoxy)butanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
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|
C28H33F3N4O6
|
1
|
1 |
IC50 = 250 nM
|
|
|
CP0447355
|
[(1R)-1-amino-3-phenylpropyl]-[(2S)-2-[[(2S)-1,6-diamino-1-oxohexan-2-yl]carbamoyl]-4-methylpentyl]phosphinic acid
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|
C22H39N4O4P
|
1
|
1 |
IC50 = 271 nM
|
|
|
CP0458634
|
[(2S)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[[3-(4-chlorophenyl)-1,2-oxazol-5-yl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C31H34ClN4O5P
|
1
|
1 |
IC50 = 345 nM
|
|
|
CP0517736
|
[(2S)-2-(1-adamantylmethyl)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C32H44N3O4P
|
1
|
1 |
IC50 = 412 nM
|
|
|
CP0568124
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-5-(3-chlorophenoxy)-2-hydroxypentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C29H37ClN4O6
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0380563
|
methyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C23H31N7O5
|
1
|
1 |
IC50 = 518 nM
|
|
|
CP0568086
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-5-(3-chlorophenoxy)-2-hydroxypentanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoate
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|
C27H36ClN3O7
|
1
|
1 |
IC50 = 580 nM
|
|
|
CP0568802
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(4-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C29H38N4O7
|
1
|
1 |
IC50 = 580 nM
|
|
|
CP0856385
|
(S)-2-(4-Amino-3-((S)-2-amino-5-guanidinopentanamido)-benzamido)-3-(1H-indol-3-yl)propanoic Acid
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|
C24H30N8O4
|
1
|
1 |
IC50 = 589 nM
|
|
|
CP0856383
|
(S)-Benzyl 2-(3-Amino-4-((S)-2-aminohexanamido)-benzamido)-3-(1H-indol-3-yl)propanoate
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|
C31H35N5O4
|
1
|
1 |
IC50 = 709 nM
|
|
|
CP0224548
|
[(2S)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C35H40N3O4P
|
1
|
1 |
IC50 = 740 nM
|
|
|
CP0445953
|
methyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
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|
C23H30N4O5
|
1
|
1 |
IC50 = 755 nM
|
|
|
CP0545509
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-(4-hydroxyphenoxy)butanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C28H36N4O7
|
1
|
1 |
IC50 = 760 nM
|
|
|
CP0447356
|
[(2R)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-oxo-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]propyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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|
C31H35N4O5P
|
1
|
1 |
IC50 = 878 nM
|
|
|
CP0543693
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(3-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C27H37N3O8
|
1
|
1 |
IC50 = 1000 nM
|
|
|
CP0460384
|
(2S)-2-[[3-amino-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
|
C24H30N8O4
|
1
|
1 |
IC50 = 1100 nM
|
|
|
CP0480665
|
methyl 3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoate
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|
C14H21N3O3
|
1
|
1 |
IC50 = 1100 nM
|
|
|
CP0400683
|
methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C23H31N7O5
|
1
|
1 |
IC50 = 1400 nM
|
|
|
CP0210942
|
benzyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoate
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|
C31H35N5O4
|
1
|
1 |
IC50 = 1600 nM
|
|
|
CP0573643
|
(2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(3-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
|
C28H36N4O7
|
1
|
1 |
IC50 = 1600 nM
|
|
|
CP0578887
|
methyl (2S)-2-[[(2R,3S)-2-amino-3-hydroxy-4-[[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-methoxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C32H43N5O8
|
1
|
1 |
IC50 = 1600 nM
|
|
|
CP0573644
|
benzyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-phenylpentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C35H42N4O5
|
1
|
1 |
IC50 = 1700 nM
|
|
|
CP0570209
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(2-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C27H37N3O8
|
1
|
1 |
IC50 = 1800 nM
|
|
|
CP0907780
|
(S)-2-(3,4-Diaminobenzamido)-3-(1H-indol-3-yl)propanoic Acid
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|
C18H18N4O3
|
1
|
1 |
IC50 = 1900 nM
|
|
|
CP0569772
|
(2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(2-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
|
C28H36N4O7
|
1
|
1 |
IC50 = 1900 nM
|
|
|
CP0481974
|
[(2R)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]-4,4-diphenylbutyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C35H40N3O4P
|
1
|
1 |
IC50 = 1922 nM
|
|
|
CP0573642
|
(2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(4-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
|
C28H36N4O7
|
1
|
1 |
IC50 = 2000 nM
|
|
|
CP0460387
|
(2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-methylpentanoyl]amino]benzoyl]amino]hexanoic acid
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|
C19H31N5O4
|
1
|
1 |
IC50 = 2100 nM
|
|
|
CP0560310
|
[(2R)-2-(1-adamantylmethyl)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C32H44N3O4P
|
1
|
1 |
IC50 = 2271 nM
|
|
|
CP0547329
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(4-hydroxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C27H37N3O8
|
1
|
1 |
IC50 = 2300 nM
|
|
|
CP0395514
|
methyl 3-amino-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoate
Show/Hide
|
C14H22N6O3
|
1
|
1 |
IC50 = 2500 nM
|
|
|
CP0400681
|
methyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-5-(diaminomethylideneamino)pentanoate
Show/Hide
|
C20H33N7O4
|
1
|
1 |
IC50 = 2500 nM
|
|
|
CP0493462
|
[(2S)-3-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-[(3,5-diphenylphenyl)methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C37H44N3O4P
|
1
|
1 |
IC50 = 2565 nM
|
|
|
CP0414323
|
(2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-3-phenylpropanoyl]amino]benzoyl]amino]hexanoic acid
Show/Hide
|
C22H29N5O4
|
1
|
1 |
IC50 = 2600 nM
|
|
|
CP0460386
|
4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoic acid
Show/Hide
|
C16H17N3O4
|
1
|
1 |
IC50 = 3200 nM
|
|
|
CP0395517
|
methyl 4-amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoate
Show/Hide
|
C14H22N6O3
|
1
|
1 |
IC50 = 3700 nM
|
|
|
CP0413517
|
(2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
|
C24H29N5O4
|
1
|
1 |
IC50 = 3800 nM
|
|
|
CP0570210
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(2-hydroxyethylamino)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C25H39N5O6
|
1
|
1 |
IC50 = 3800 nM
|
|
|
CP0476829
|
(2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]hexanoic acid
Show/Hide
|
C22H29N5O5
|
1
|
1 |
IC50 = 4500 nM
|
|
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CP0473586
|
[(2R)-3-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-2-[(3,5-diphenylphenyl)methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
Show/Hide
|
C40H42N3O4P
|
1
|
1 |
IC50 = 4622 nM
|
|
|
CP0414329
|
methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoyl]amino]hexanoate
Show/Hide
|
C24H33N5O5
|
1
|
1 |
IC50 = 4800 nM
|
|
|
CP0865677
|
(S)-2-(3-Amino-4-((S)-2-amino-3-(4-hydroxyphenyl)-propanamido)benzamido)-3-(1H-indol-3-yl)propanoic Acid
Show/Hide
|
C27H27N5O5
|
1
|
1 |
IC50 = 4800 nM
|
|
|
CP0568084
|
methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2,7-dihydroxyheptanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C23H37N3O7
|
1
|
1 |
IC50 = 4900 nM
|
|
|
CP0386653
|
(2S)-2-[[4-amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]-3-methylbutanoic acid
Show/Hide
|
C18H29N7O4
|
1
|
1 |
IC50 = 5000 nM
|
|
|
CP0386661
|
methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
|
C27H30N4O5
|
1
|
1 |
IC50 = 5500 nM
|
|
|
CP0552067
|
benzyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(4-phenylmethoxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
|
C42H48N4O7
|
1
|
1 |
IC50 = 5500 nM
|
|
|
CP0386655
|
benzyl (2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoate
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C25H34N4O4
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1
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1 |
IC50 = 6200 nM
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CP0413511
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methyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
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C23H30N4O5
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1
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1 |
IC50 = 6400 nM
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CP0568255
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(4-phenylmethoxyphenoxy)pentanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoate
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C34H43N3O8
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1
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1 |
IC50 = 7500 nM
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CP0543750
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methyl (2S)-2-[[(3R,4S)-3-amino-4-hydroxy-5-[[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-methoxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentyl]amino]-3-(4-hydroxyphenyl)propanoate
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C33H45N5O8
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1
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1 |
IC50 = 7900 nM
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CP0573645
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3-[[(3R,4S)-3-amino-4-hydroxy-5-[[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-methoxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-oxopentyl]amino]propanoic acid
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C26H39N5O7
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1
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1 |
IC50 = 8200 nM
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CP0414325
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methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]hexanoate
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C20H33N5O4
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1
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1 |
IC50 = 8300 nM
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CP0458316
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(2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]hexanoic acid
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C23H31N5O4
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1
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1 |
IC50 = 8900 nM
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CP0866550
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(S)-2-(3-Amino-4-((S)-2-amino-4-(4-hydroxyphenyl)-butanamido)benzamido)-3-(1H-indol-3-yl)propanoic Acid
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C28H29N5O5
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1
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1 |
IC50 = 9400 nM
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CP0574513
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-5-(1,3-dihydroxypropan-2-ylamino)-2-hydroxypentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
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C26H41N5O7
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1
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1 |
IC50 = 9600 nM
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CP0449988
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methyl 4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoate
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C14H21N3O3
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1
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1 |
IC50 = 9800 nM
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CP0856382
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(S)-Benzyl 2-(3-Amino-4-((S)-2-amino-4-phenylbutanamido)benzamido)-3-(1H-indol-3-yl)propanoate
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C35H35N5O4
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1
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1 |
IC50 = 11000 nM
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CP0579203
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benzyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2,4-dihydroxybutanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
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C28H36N4O6
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1
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1 |
IC50 = 11000 nM
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CP0379588
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benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-methylbutanoate
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C29H34N4O4
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1
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1 |
IC50 = 11500 nM
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CP0445952
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methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-5-(diaminomethylideneamino)pentanoate
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C24H33N7O4
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1
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1 |
IC50 = 11800 nM
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CP0460385
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methyl (2S)-6-amino-2-[[3-amino-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]hexanoate
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C20H34N8O4
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1
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1 |
IC50 = 11800 nM
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CP0480663
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methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-(4-phenylmethoxyphenyl)butanoyl]amino]benzoyl]amino]hexanoate
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C31H39N5O5
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1
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1 |
IC50 = 13000 nM
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CP0552108
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(5R,6S)-5-amino-6-hydroxy-7-[[(2S)-1-[[(2S)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-7-oxoheptanoic acid
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C23H35N3O8
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1
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1 |
IC50 = 13000 nM
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CP0568804
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(4R,5S)-4-amino-5-hydroxy-6-[[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-oxo-1-phenylmethoxypropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-6-oxohexanoic acid
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C30H38N4O7
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1
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1 |
IC50 = 13000 nM
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CP0571162
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-[2-hydroxyethyl(methyl)amino]pentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
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C26H41N5O6
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1
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1 |
IC50 = 13000 nM
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CP0473581
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[(2S)-3-[[(2S)-1-amino-4-methyl-1-oxopentan-2-yl]amino]-2-[[3,5-bis(3-chlorophenyl)phenyl]methyl]-3-oxopropyl]-[(1R)-1-amino-3-phenylpropyl]phosphinic acid
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C37H42Cl2N3O4P
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1
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1 |
IC50 = 13814 nM
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CP0413512
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methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
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C26H28N4O6
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1
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1 |
IC50 = 15100 nM
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CP0395515
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methyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-3-(4-phenylmethoxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
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C33H34N4O6
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1
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1 |
IC50 = 16000 nM
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CP0413513
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methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoyl]amino]hexanoate
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C20H34N8O4
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1
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1 |
IC50 = 17000 nM
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CP0567748
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(2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-phenylpentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
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C28H36N4O5
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1
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1 |
IC50 = 17000 nM
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CP0569771
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-4-(2-hydroxyethylamino)butanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
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C24H37N5O6
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1
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1 |
IC50 = 18000 nM
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CP0568256
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(4R,5S)-4-amino-6-[[(2S)-1-[[(1S)-1-carboxy-2-(1H-indol-3-yl)ethyl]amino]-4-methyl-1-oxopentan-2-yl]amino]-5-hydroxy-6-oxohexanoic acid
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C23H32N4O7
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1
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1 |
IC50 = 19000 nM
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CP0856386
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(S)-Benzyl 2-(3-Amino-4-((S)-2-amino-3-(4-(benzyloxy)-phenyl)propanamido)benzamido)-3-(1H-indol-3-yl)-propanoate
Show/Hide
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C41H39N5O5
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1
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1 |
IC50 = 20500 nM
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CP0856387
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(S)-Benzyl 2-(3-Amino-4-((S)-2-amino-4-methylpentanamido)benzamido)-3-(1H-indol-3-yl)propanoate
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C31H35N5O4
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1
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1 |
IC50 = 21000 nM
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CP0411593
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benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C35H35N5O4
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1
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1 |
IC50 = 23900 nM
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CP0465905
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methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]hexanoate
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C24H33N5O4
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1
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1 |
IC50 = 24900 nM
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CP0577096
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-4-(1,3-dihydroxypropan-2-ylamino)-2-hydroxybutanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
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C25H39N5O7
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1
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1 |
IC50 = 27000 nM
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CP0569774
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-(2-hydroxyethylamino)-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C25H37N5O7
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1
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1 |
IC50 = 30000 nM
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CP0578347
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benzyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-2,5-dihydroxypentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C29H38N4O6
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1
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1 |
IC50 = 30000 nM
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CP0489242
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methyl (2S)-6-amino-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]hexanoate
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C20H33N5O4
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1
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1 |
IC50 = 30600 nM
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CP0547217
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(5R,6S)-5-amino-6-hydroxy-7-[[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-oxo-1-phenylmethoxypropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-7-oxoheptanoic acid
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C31H40N4O7
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1
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1 |
IC50 = 31000 nM
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CP0449986
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methyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
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C26H28N4O6
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1
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1 |
IC50 = 33000 nM
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CP0569773
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(2S)-2-[[(3R,4S)-3-amino-5-[[(2S)-1-[[(1S)-1-carboxy-2-(1H-indol-3-yl)ethyl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-hydroxy-5-oxopentyl]amino]-3-(4-hydroxyphenyl)propanoic acid
Show/Hide
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C31H41N5O8
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1
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1 |
IC50 = 37000 nM
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CP0400680
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(2S)-2-[[3-amino-4-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoic acid
Show/Hide
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C18H28N4O4
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1
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1 |
IC50 = 38000 nM
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CP0413515
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methyl (2S,3R)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-hydroxybutanoate
Show/Hide
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C21H26N4O6
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1
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1 |
IC50 = 39000 nM
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CP0883490
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(S)-Benzyl 2-(4-Amino-3-((S)-2-amino-3-(4-hydroxyphenyl)-propanamido)benzamido)-3-(1H-indol-3-yl)propanoate
Show/Hide
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C34H33N5O5
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1
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1 |
IC50 = 40000 nM
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CP0453812
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benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-methylbutanoate
Show/Hide
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C28H32N4O5
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1
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1 |
IC50 = 50000 nM
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CP0414324
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methyl (2S)-6-amino-2-[[4-amino-3-[[(2S)-2-amino-4-methylpentanoyl]amino]benzoyl]amino]hexanoate
Show/Hide
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C20H33N5O4
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1
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1 |
IC50 = 52000 nM
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CP0386654
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methyl 3-amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoate
Show/Hide
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C17H19N3O4
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1
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1 |
IC50 = 58000 nM
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CP0395513
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methyl 3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoate
Show/Hide
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C18H21N3O3
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1
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1 |
IC50 = 58000 nM
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CP0866549
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(S)-Benzyl 2-(3-Amino-4-((S)-2-amino-4-(4-(benzyloxy)-phenyl)butanamido)benzamido)-3-(1H-indol-3-yl)propanoate
Show/Hide
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C42H41N5O5
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1
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1 |
IC50 = 70000 nM
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CP0396765
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4-methoxy-3-[(2-piperidin-1-ylphenyl)sulfamoyl]benzoic acid
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C19H22N2O5S
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1
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1 |
IC50 = 81200 nM
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CP0446943
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4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoic acid
Show/Hide
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C17H19N3O3
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1
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1 |
IC50 > 100000 nM
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CP0446944
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methyl 4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoate
Show/Hide
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C18H21N3O3
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1
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1 |
IC50 > 100000 nM
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CP0473679
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methyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-(4-hydroxyphenyl)propanoate
Show/Hide
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C27H30N4O5
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1
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1 |
IC50 > 100000 nM
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CP0386657
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methyl 3-amino-4-[[(2S)-2-amino-4-methylpentanoyl]amino]benzoate
Show/Hide
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C14H21N3O3
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1
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1 |
IC50 > 100000 nM
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CP0386660
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(2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-methylbutanoic acid
Show/Hide
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C22H28N4O4
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1
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1 |
IC50 > 100000 nM
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CP0413508
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(2S)-2-[[4-amino-3-[[(2S)-2-amino-4-(4-hydroxyphenyl)butanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
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C28H29N5O5
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1
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1 |
IC50 > 100000 nM
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CP0413510
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(2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoic acid
Show/Hide
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C18H28N4O4
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1
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1 |
IC50 > 100000 nM
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CP0413514
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(2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-methylbutanoic acid
Show/Hide
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C21H26N4O5
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1
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1 |
IC50 > 100000 nM
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CP0414326
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methyl (2S)-6-amino-2-[[3-amino-4-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]hexanoate
Show/Hide
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C23H31N5O5
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1
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1 |
IC50 > 100000 nM
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CP0418659
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methyl 4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoate
Show/Hide
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C17H19N3O4
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1
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1 |
IC50 > 100000 nM
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CP0445950
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benzyl (2S)-2-[[4-amino-3-[[(2S)-2-aminohexanoyl]amino]benzoyl]amino]-3-methylbutanoate
Show/Hide
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C25H34N4O4
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1
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1 |
IC50 > 100000 nM
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CP0476814
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4-amino-3-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]benzoic acid
Show/Hide
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C13H20N6O3
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1
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1 |
IC50 > 100000 nM
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CP0480660
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(2S)-2-[[4-amino-3-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoic acid
Show/Hide
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C27H27N5O5
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1
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1 |
IC50 > 100000 nM
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CP0480661
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benzyl (2S)-2-[[4-amino-3-[[(2S)-2-amino-4-(4-phenylmethoxyphenyl)butanoyl]amino]benzoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C42H41N5O5
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1
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1 |
IC50 > 100000 nM
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CP0487730
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benzyl (2S)-2-[[3-amino-4-[[(2S)-2-amino-4-phenylbutanoyl]amino]benzoyl]amino]-3-methylbutanoate
Show/Hide
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C29H34N4O4
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1
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1 |
IC50 > 100000 nM
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CP0508029
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benzyl (2S)-2-[(3,4-diaminobenzoyl)amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C25H24N4O3
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1
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1 |
IC50 > 100000 nM
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CP0037780
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(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
Show/Hide
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C16H24N2O4
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1
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1 |
IC50 > 100000 nM
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CP0568254
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(2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-phenylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
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C17H26N2O4
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1
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1 |
IC50 > 100000 nM
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CP0572845
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methyl (2S)-2-[[(2S)-2-[[(2S,3R)-3-amino-5-(1,3-dihydroxypropan-2-ylamino)-2-hydroxy-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoate
Show/Hide
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C26H39N5O8
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1
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1 |
IC50 > 100000 nM
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CP0578519
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methyl (2S)-2-[[(2S,3R)-3-amino-2-hydroxy-5-phenylpentanoyl]amino]-4-methylpentanoate
Show/Hide
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C18H28N2O4
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1
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1 |
IC50 > 100000 nM
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