| Compound ID |
Compound Name |
Compound Formula |
|
CP0451057
|
N-[3-chloro-4-(2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)phenyl]-3-methylpyrazole-1-carboxamide
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|
C22H21ClN4O2
|
2
|
| 1 |
EC50 = 4 nM
|
|
|
| 2 |
IC50 = 13 nM
|
|
|
|
CP0368353
|
2-[(R)-1-(2-Chloro-4-pyrrolidin-1-yl-benzoyl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-5-yl]-N-isopropyl-acetamide
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|
C26H32ClN3O2
|
2
|
| 1 |
EC50 = 189 nM
|
|
|
| 2 |
Ki = 91.9 nM
|
|
|
|
CP0228540
|
N-[4-(7-chloro-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)-3-methylphenyl]-2-(2-methylphenoxy)acetamide
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|
C27H27ClN2O3
|
1
|
| 1 |
IC50 = 0.95 nM
|
|
|
|
CP0383782
|
(4-Amino-2-methyl-phenyl)-(7-chloro-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C18H19ClN2O
|
1
|
| 1 |
IC50 = 4.1 nM
|
|
|
|
CP0397426
|
(2-Chloro-4-ethylamino-phenyl)-(7-chloro-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C19H20Cl2N2O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0457328
|
(4-Allylamino-2-chloro-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C20H21ClN2O
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0404376
|
(2-Chloro-4-pyrrol-1-yl-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H19ClN2O
|
1
|
| 1 |
IC50 = 7.5 nM
|
|
|
|
CP0448407
|
(2-Chloro-4-pyrazol-1-yl-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C20H18ClN3O
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0289061
|
(2-Chloro-4-pyrrolidin-1-yl-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H23ClN2O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0397695
|
[2-chloro-4-(3-methylpyrazol-1-yl)phenyl]-(2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone
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|
C21H20ClN3O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0460518
|
(2-Chloro-4-dimethylamino-phenyl)-(7-chloro-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C19H20Cl2N2O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0460519
|
(2-Chloro-4-pyrrolidin-1-yl-phenyl)-(7-chloro-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H22Cl2N2O
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0403010
|
(2-Chloro-4-dimethylamino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C19H21ClN2O
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0449036
|
(2-Chloro-4-propylamino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C20H23ClN2O
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0422971
|
(2-Chloro-4-diethylamino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H25ClN2O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0377662
|
(4-Butylamino-2-chloro-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H25ClN2O
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0448442
|
(2-Chloro-4-pentylamino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C22H27ClN2O
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0395251
|
(2-Chloro-4-ethylamino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C19H21ClN2O
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0397570
|
(2-Chloro-4-methylamino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C18H19ClN2O
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0463156
|
[2-chloro-4-(3-methylpyrrolidin-1-yl)phenyl]-(2,3,4,5-tetrahydro-1-benzazepin-1-yl)methanone
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|
C22H25ClN2O
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0404485
|
(2-Chloro-4-piperidin-1-yl-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C22H25ClN2O
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0410534
|
(4-Amino-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C17H18N2O
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0448139
|
(7-Chloro-2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-(4-pyrrolidin-1-yl-phenyl)-methanone
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|
C21H23ClN2O
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0459256
|
(4-Pyrrol-1-yl-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H20N2O
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0397543
|
(4-Pyrrolidin-1-yl-phenyl)-(2,3,4,5-tetrahydro-benzo[b]azepin-1-yl)-methanone
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|
C21H24N2O
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0392030
|
N-[4-(7-chloro-5-hydroxy-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)-3-methylphenyl]-2-methylbenzamide
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|
C26H25ClN2O3
|
1
|
| 1 |
Ki = 0.43 nM
|
|
|
|
CP0178094
|
N-[4-[5-(dimethylamino)-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl]phenyl]-2-methylbenzamide
Show/Hide
|
C27H29N3O2
|
1
|
| 1 |
Ki = 9.42 nM
|
|
|
