Brief Information of the Cell Line and Protein
Cell Line ID: CL000017 , HeLa
Synonyms
HELA
Hela
He La
He-La
HeLa-CCL2
Henrietta Lacks cells
Helacyton gartleri
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0030
Protein ID: PT01588 , Corticotropin-releasing factor receptor 1
Gene Name CRHR1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P34998
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000017  Protein ID: PT01588
 
Compound ID Compound Name Compound Formula
CP0896982
DPhe-His-Leu-Leu-Arg-Glu-Val-Leu-Glu-Nle-Ala-Arg-Ala-Glu-Gln-Leu-Ala-Gln-Glu-Ala-His-Lys-Asn-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C164H275N49O41
 1
1
Ki = 2 nM
   TI
   LI
   LO
   TS
CP0398942
Ac-(Glu-Aib-Glu-Lys)-Leu-Arg-Lys-Leu-Cha-Asp-Ile-Ile-NH2
   Show/Hide
C70H112N18O21
 1
1
Ki = 3 nM
   TI
   LI
   LO
   TS
CP0475667
Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Cha-Asp-Ile-Ile-NH2
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C68H117N19O19
 1
1
Ki = 3.1 nM
   TI
   LI
   LO
   TS
CP0460806
Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Phe-Asp-Ile-Ile-NH2
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C68H117N19O19
 1
1
Ki = 5.5 nM
   TI
   LI
   LO
   TS
CP0953776
Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Nle-Asp-Ile-Ile-NH2
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C65H113N19O19
 1
1
Ki = 36.7 nM
   TI
   LI
   LO
   TS
CP0892323
Ac-(Glu-Ala-Lys-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C67H120N20O17
 1
1
Ki = 44.8 nM
   TI
   LI
   LO
   TS
CP0895356
Ac-(Glu-Ala-His-Lys)-Leu-Lys-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C67H115N19O17
 1
1
Ki = 45.1 nM
   TI
   LI
   LO
   TS
CP0878021
Ac-(Glu-Ala-Leu-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C67H119N19O17
 1
1
Ki = 48.9 nM
   TI
   LI
   LO
   TS
CP0874485
Ac-(Glu-Ala-His-Lys)-Asn-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C67H115N21O17
 1
1
Ki = 50 nM
   TI
   LI
   LO
   TS
CP0530992
Ac-(Glu-Ala-His-Lys)-Leu-Ala-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C67H113N17O17
 1
1
Ki = 70.9 nM
   TI
   LI
   LO
   TS
CP0391996
Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Phe-Asp-Ile-Ile-NH2
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C69H112N18O19
 1
1
Ki = 81 nM
   TI
   LI
   LO
   TS
CP0957141
Ac-(Glu-Ala-Glu-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C66H115N19O19
 1
1
Ki = 130 nM
   TI
   LI
   LO
   TS
CP0846132
Ac-(Glu-Ala-His-Lys)-Gln-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C68H117N21O17
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0850078
Ac-(Glu-Asp-His-Lys)-Asn-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
   Show/Hide
C68H115N21O19
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0853591
Ac-(Glu-Ala-His-Lys)-Dab-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C68H119N21O16
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0859206
Ac-(Glu-Ala-His-Lys)-Asp-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
   Show/Hide
C67H114N20O18
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0874400
Ac-(Glu-Dap-His-Lys)-Asn-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C67H116N22O17
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0919157
Ac-(Glu-Ala-Phe-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C70H117N19O17
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0919179
Ac-(Glu-Ala-Asp-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C65H113N19O19
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0942688
Ac-(Glu-Ala-His-Lys)-Leu-Gly-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C63H106N18O17
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0967496
Ac-(Glu-Ala-His-Lys)-Leu-Arg-Lys-Leu-Nle-Glu-Ile-Ile-NH2
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C69H120N20O16
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS