Compound ID |
Compound Name |
Compound Formula |
CP0017968
|
3-cyano-4-[2-[2-[(2-piperidin-4-ylethylamino)methyl]pyridin-4-yl]-4-[3-(trifluoromethyl)phenyl]phenoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
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|
C35H32F3N7O3S2
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0376628
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(3-methyl-3H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
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|
C27H30FN7O
|
1
|
1 |
Ki = 2.8 nM
|
|
|
CP0453890
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-5-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
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|
C28H29FN6O
|
1
|
1 |
Ki = 4.2 nM
|
|
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
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|
C10H12N2O
|
1
|
1 |
Ki = 4.8 nM
|
|
|
CP0448256
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-pyrazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 5.9 nM
|
|
|
CP0459887
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 6.5 nM
|
|
|
CP0492027
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-imidazol-2-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 11 nM
|
|
|
CP0126862
|
1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl)-4-methylpiperazine
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|
C24H23FN4
|
1
|
1 |
Ki = 13 nM
|
|
|
CP0490676
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-pyridin-3-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
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|
C29H30FN5O
|
1
|
1 |
Ki = 14 nM
|
|
|
CP0404715
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C26H29FN8O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0429995
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(4-methyl-4H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0382930
|
1-(2-{4-[5-(1-Ethyl-1H-[1,2,3]triazol-4-yl)-1-(4-fluoro-phenyl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H32FN7O
|
1
|
1 |
Ki = 28 nM
|
|
|
CP0392710
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C26H28FN7O
|
1
|
1 |
Ki = 31 nM
|
|
|
CP0126860
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 36 nM
|
|
|
CP0502318
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 45 nM
|
|
|
CP0228798
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C26H29FN8O
|
1
|
1 |
Ki = 48 nM
|
|
|
CP0046703
|
1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl]piperidin-1-yl}ethyl)imidazolidin-2-one
Show/Hide
|
C24H26ClFN4O
|
1
|
1 |
Ki = 56 nM
|
|
|
CP0384143
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-[1,2,3]triazol-4-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 67 nM
|
|
|
CP0151333
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C27H30FN7O
|
1
|
1 |
Ki = 68 nM
|
|
|
CP0382893
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-2-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H29FN6O
|
1
|
1 |
Ki = 76 nM
|
|
|
CP0320413
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-1-methyl-pyrrolidin-2-one
Show/Hide
|
C29H33FN6O
|
1
|
1 |
Ki = 100 nM
|
|
|
CP0277576
|
1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H31FN6O
|
1
|
1 |
Ki = 110 nM
|
|
|
CP0105167
|
3-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-2-yl-1H-indol-3-yl]-piperidin-1-yl}-propionitrile
Show/Hide
|
C26H24FN5
|
1
|
1 |
Ki = 200 nM
|
|
|
CP0406243
|
1-(2-{4-[5-(2-Ethyl-2H-[1,2,3]triazol-4-yl)-1-(4-fluoro-phenyl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-imidazolidin-2-one
Show/Hide
|
C28H32FN7O
|
1
|
1 |
Ki = 208 nM
|
|
|
CP0267173
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-oxazolidin-2-one
Show/Hide
|
C26H28FN7O2
|
1
|
1 |
Ki = 220 nM
|
|
|
CP0163622
|
3-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-propionitrile
Show/Hide
|
C25H25FN6
|
1
|
1 |
Ki = 340 nM
|
|
|
CP0134581
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-pyrimidin-2-yl-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-oxazolidin-2-one
Show/Hide
|
C28H28FN5O2
|
1
|
1 |
Ki = 360 nM
|
|
|
CP0343878
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-oxazolidin-2-one
Show/Hide
|
C27H29FN6O2
|
1
|
1 |
Ki = 480 nM
|
|
|
CP0333143
|
3-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-piperidin-1-yl}-ethyl)-1H-quinazoline-2,4-dione
Show/Hide
|
C32H30FN7O2
|
1
|
1 |
Ki = 560 nM
|
|
|
CP0379546
|
1-methyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C22H22N4O2S
|
1
|
1 |
Ki = 3624 nM
|
|
|
CP0072419
|
(SNAP-8719)[4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-octahydro-quinoxalin-1-yl]-furan-2-yl-methanone
Show/Hide
|
C22H28F3N3O2
|
1
|
1 |
Ki = 7700 nM
|
|
|
CP0379542
|
5-(4-Methylpiperazin-1-yl)-3-(1-naphthalenesulfonyl)-1H-indazole
Show/Hide
|
C22H22N4O2S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0379544
|
5-(4-methylpiperazin-1-yl)-3-(phenylsulfonyl)-1H-indazole
Show/Hide
|
C18H20N4O2S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0379545
|
3-(Naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C21H20N4O2S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0379601
|
1-isopropyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C24H26N4O2S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0406091
|
1-benzyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C28H26N4O2S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0479094
|
1-isobutyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
Show/Hide
|
C25H28N4O2S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0040814
|
[4-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl]-(furan-2-yl)methanone
Show/Hide
|
C19H21N5O4
|
1
|
1 |
Ki > 7700 nM
|
|
|