Brief Information of the Cell Line and Protein
Cell Line ID: CL000017 , HeLa
Synonyms
HELA
Hela
He La
He-La
HeLa-CCL2
Henrietta Lacks cells
Helacyton gartleri
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0030
Protein ID: PT01005 , D(2) dopamine receptor
Gene Name DRD2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P14416
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000017  Protein ID: PT01005
 
Compound ID Compound Name Compound Formula
CP0379542
5-(4-Methylpiperazin-1-yl)-3-(1-naphthalenesulfonyl)-1H-indazole
   Show/Hide
C22H22N4O2S
 1
1
Ki = 334 nM
   TI
   LI
   LO
   TS
CP0379544
5-(4-methylpiperazin-1-yl)-3-(phenylsulfonyl)-1H-indazole
   Show/Hide
C18H20N4O2S
 1
1
Ki = 355 nM
   TI
   LI
   LO
   TS
CP0406091
1-benzyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
   Show/Hide
C28H26N4O2S
 1
1
Ki = 605 nM
   TI
   LI
   LO
   TS
CP0479094
1-isobutyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
   Show/Hide
C25H28N4O2S
 1
1
Ki = 1903 nM
   TI
   LI
   LO
   TS
CP0379601
1-isopropyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
   Show/Hide
C24H26N4O2S
 1
1
Ki = 2036 nM
   TI
   LI
   LO
   TS
CP0379546
1-methyl-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
   Show/Hide
C22H22N4O2S
 1
1
Ki = 2243 nM
   TI
   LI
   LO
   TS
CP0379545
3-(Naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1H-indazole
   Show/Hide
C21H20N4O2S
 1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS