| Compound ID |
Compound Name |
Compound Formula |
|
CP0454741
|
[5-chloro-2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C19H13BClF3N2O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0410366
|
N-[4-chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-6-[4-(trifluoromethyl)phenoxy]pyridine-3-carboxamide
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|
C25H23BClF3N2O4
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
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CP0224642
|
[5-chloro-2-[2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
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|
C19H19BClF3N2O4
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0575902
|
[5-fluoro-2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C19H13BF4N2O4
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0447611
|
N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-6-[4-(trifluoromethyl)phenoxy]pyridine-3-carboxamide
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|
C25H24BF3N2O4
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0457327
|
[4-fluoro-2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C19H13BF4N2O4
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0237932
|
[5-methoxy-2-[2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
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|
C20H22BF3N2O5
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0517804
|
[5-methyl-2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C20H16BF3N2O4
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0483595
|
N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-6-[3-(trifluoromethoxy)phenoxy]pyridine-3-carboxamide
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|
C25H24BF3N2O5
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0517805
|
[4-chloro-2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C19H13BClF3N2O4
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0548568
|
N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-6-[4-(trifluoromethoxy)phenoxy]pyridine-3-carboxamide
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|
C25H24BF3N2O5
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0478976
|
6-[N-methyl-4-(trifluoromethoxy)anilino]-N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyridine-3-carboxamide
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|
C26H27BF3N3O4
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0517803
|
[2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C19H14BF3N2O4
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0458002
|
[4-methoxy-2-[[6-[4-(trifluoromethyl)phenoxy]pyridine-3-carbonyl]amino]phenyl]boronic acid
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|
C20H16BF3N2O5
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0315031
|
[5-fluoro-2-[2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
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|
C19H19BF4N2O4
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0420330
|
[2-[[4-[5-(trifluoromethyl)pyridin-2-yl]oxybenzoyl]amino]phenyl]boronic acid
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|
C19H14BF3N2O4
|
1
|
| 1 |
IC50 = 91 nM
|
|
|
|
CP0224640
|
[2-[2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
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|
C19H20BF3N2O4
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0148538
|
[2-[2-oxo-2-[4-[4-(trifluoromethyl)phenoxy]piperidin-1-yl]ethyl]phenyl]boronic acid
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|
C20H21BF3NO4
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0558965
|
N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-5-[4-(trifluoromethyl)phenoxy]pyridine-2-carboxamide
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|
C25H24BF3N2O4
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0564722
|
N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-4-[5-(trifluoromethyl)pyridin-2-yl]oxybenzamide
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|
C25H24BF3N2O4
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0224641
|
[2-[1-hydroxy-2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
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|
C19H20BF3N2O5
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0099287
|
[2-[2-oxo-2-[4-[[5-(trifluoromethyl)pyridin-2-yl]oxymethyl]piperidin-1-yl]ethyl]phenyl]boronic acid
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|
C20H22BF3N2O4
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0567125
|
2-methyl-N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-4-[5-(trifluoromethyl)pyridin-2-yl]oxybenzamide
Show/Hide
|
C26H26BF3N2O4
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0431637
|
[2-[[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]methyl]phenyl]boronic acid
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|
C18H20BF3N2O3
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
|
CP0153097
|
[2-[2-oxo-2-[4-[6-(trifluoromethyl)pyridin-3-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
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|
C19H20BF3N2O4
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0461871
|
[2-[3-oxo-3-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]propyl]phenyl]boronic acid
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|
C20H22BF3N2O4
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0494033
|
[2-[[5-[5-(trifluoromethyl)pyridin-2-yl]oxypyridine-2-carbonyl]amino]phenyl]boronic acid
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|
C18H13BF3N3O4
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0479895
|
N-[2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-5-[5-(trifluoromethyl)pyridin-2-yl]oxypyridine-2-carboxamide
Show/Hide
|
C24H23BF3N3O4
|
1
|
| 1 |
IC50 = 920 nM
|
|
|
|
CP0356750
|
[2-[1-methoxy-2-oxo-2-[4-[5-(trifluoromethyl)pyridin-2-yl]oxypiperidin-1-yl]ethyl]phenyl]boronic acid
Show/Hide
|
C20H22BF3N2O5
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0148539
|
[2-[2-[4-[5-(dimethylcarbamoyl)pyridin-2-yl]oxypiperidin-1-yl]-2-oxoethyl]phenyl]boronic acid
Show/Hide
|
C21H26BN3O5
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
