| Compound ID |
Compound Name |
Compound Formula |
|
CP0198178
|
3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-benzoimidazol-1-yl]-propan-1-ol
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|
C21H21N5O
|
1
|
| 1 |
IC50 = 352 nM
|
|
|
|
CP0461161
|
1-methyl-6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1Hbenzoimidazole
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|
C19H17N5
|
1
|
| 1 |
IC50 = 395 nM
|
|
|
|
CP0015520
|
4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline
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|
C17H12N4
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0198179
|
1-methyl-6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo-[1,2-b]pyrazol-3-yl]-1H-benzoimidazole
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|
C20H19N5
|
1
|
| 1 |
IC50 = 668 nM
|
|
|
|
CP0140650
|
3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazol-1-yl)propan-1-ol
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|
C22H23N5O
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0208736
|
6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1Hbenzoimidazole
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|
C19H17N5
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0134782
|
5-(2-(pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazole
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|
C18H15N5
|
1
|
| 1 |
IC50 = 8730 nM
|
|
|
|
CP0208733
|
6-(2-(pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-(3-(pyrrolidin-1-yl)propyl)-1H-benzo[d]imidazole
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|
C25H28N6
|
1
|
| 1 |
IC50 = 10840 nM
|
|
|
|
CP0339841
|
5-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-[3-(tetrahydro-pyran-2-yloxy)-propyl]-1H-benzoimidazole
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|
C27H31N5O2
|
1
|
| 1 |
IC50 = 14540 nM
|
|
|
|
CP0132093
|
1-methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzoimidazole
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|
C19H17N5
|
1
|
| 1 |
IC50 = 19630 nM
|
|
|
|
CP0299325
|
4-(3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-benzo[d]imidazol-1-yl)propyl)morpholine
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|
C26H30N6O
|
1
|
| 1 |
IC50 = 19750 nM
|
|
|
|
CP0153367
|
N,N-dimethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine
Show/Hide
|
C24H28N6
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0199523
|
5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1-[3-(tetrahydro-pyran-2-yloxy)-propyl]-1H-benzoimidazole
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|
C26H29N5O2
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0208734
|
N,N-diethyl-3-[6-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]benzimidazol-1-yl]propan-1-amine
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|
C26H32N6
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0208737
|
1-methyl-5-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1H-indole
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|
C21H20N4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0324264
|
N,N-dimethyl-3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)benzimidazol-1-yl]propan-1-amine
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|
C23H26N6
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0339842
|
6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-pyrrolidin-1-yl-propyl)-1H-benzoimidazole
Show/Hide
|
C26H30N6
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0343570
|
6-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]-1-(3-piperidin-1-yl-propyl)-1H-benzoimidazole
Show/Hide
|
C27H32N6
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
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CP0439470
|
1-methyl-5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole
Show/Hide
|
C20H18N4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0508199
|
5-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)-1H-indole
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|
C19H16N4
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0382724
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C49H54BF2N7O7
|
1
|
| 1 |
Kd = 854 nM
|
|
|
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CP0382649
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
Show/Hide
|
C50H56BF2N7O7
|
1
|
| 1 |
Kd > 2000 nM
|
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