| Compound ID |
Compound Name |
Compound Formula |
|
CP0539833
|
5-[4-[(3S)-3-(4-fluorophenyl)morpholin-4-yl]-2-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]quinazolin-6-yl]-1,3-dimethylpyridin-2-one
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|
C32H33FN6O3
|
2
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 < 100 nM
|
|
|
|
CP0528739
|
5-[2-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]-4-[(3S)-3-phenylmorpholin-4-yl]quinazolin-6-yl]-1,3-dimethylpyridin-2-one
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|
C32H34N6O3
|
2
|
| 1 |
IC50 = 11 nM
|
|
|
| 2 |
IC50 < 100 nM
|
|
|
|
CP0548212
|
1-[4-[6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-[(3S)-3-(4-fluorophenyl)morpholin-4-yl]quinazolin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C30H31FN6O3
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0229168
|
1-[4-[6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-[(3S)-3-phenylmorpholin-4-yl]quinazolin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C30H32N6O3
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0004236
|
(+)-JQ1
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|
C23H25ClN4O2S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0552885
|
5-[2-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]-4-[(3S)-3-phenylmorpholin-4-yl]quinazolin-6-yl]-1-methylpyridin-2-one
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|
C31H32N6O3
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0356954
|
2-[4-[6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-(3-phenylmorpholin-4-yl)quinazolin-2-yl]pyrazol-1-yl]ethanol
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|
C28H28N6O3
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0552952
|
1-[4-[4-[(3S)-3-cyclopropylmorpholin-4-yl]-6-(3,5-dimethyl-1,2-oxazol-4-yl)quinazolin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C27H32N6O3
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0547444
|
1-[4-[6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-[(2S)-4-methylsulfonyl-2-phenylpiperazin-1-yl]quinazolin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C31H35N7O4S
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0570905
|
5-[4-[(3S)-3-cyclopropylmorpholin-4-yl]-2-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]quinazolin-6-yl]-1,3-dimethylpyridin-2-one
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|
C29H34N6O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0902755
|
(S)-4-(2-(1-(2-hydroxy-2-methylpropyl)-1H-pyrazol-4-yl)-4-(3-phenylmorpholino)quinazolin-6-yl)-6-methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one
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|
C33H33N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0902756
|
(S)-4-(4-(3-cyclopropylmorpholino)-2-(1-(2-hydroxy-2-methylpropyl)-1H-pyrazol-4-yl)quinazolin-6-yl)-6-methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one
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|
C30H33N7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0967237
|
(S)-4-(4-(3-(4-fluorophenyl)morpholino)-2-(1-(2-hydroxy-2-methylpropyl)-1H-pyrazol-4-yl)quinazolin-6-yl)-6-methyl-1H-pyrrolo[2,3-c]pyridin-7(6H)-one
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|
C33H32FN7O3
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0512516
|
1-[(3S)-4-[6-(3,5-dimethyl-1,2-oxazol-4-yl)-2-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]quinazolin-4-yl]-3-phenylpiperazin-1-yl]ethanone
Show/Hide
|
C32H35N7O3
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0548213
|
1-[4-[4-[(3S)-3-(4-chlorophenyl)morpholin-4-yl]-6-(3,5-dimethyl-1,2-oxazol-4-yl)quinazolin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C30H31ClN6O3
|
1
|
| 1 |
IC50 = 155 nM
|
|
|
|
CP0565975
|
5-[2-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]-4-[(3R)-3-thiophen-2-ylmorpholin-4-yl]quinazolin-6-yl]-1-methylpyridin-2-one
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|
C29H30N6O3S
|
1
|
| 1 |
IC50 = 165 nM
|
|
|
|
CP0153135
|
5-chloro-2-methoxy-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C20H15ClN2O4S
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0531344
|
1-[4-[6-(3,5-dimethyl-1,2-oxazol-4-yl)-4-[(3R)-3-thiophen-2-ylmorpholin-4-yl]quinazolin-2-yl]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C28H30N6O3S
|
1
|
| 1 |
IC50 = 364 nM
|
|
|
|
CP0559746
|
2-methoxy-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C20H16N2O4S
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0475539
|
3-chloro-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C19H13ClN2O3S
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
|
CP0476451
|
4-chloro-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C19H13ClN2O3S
|
1
|
| 1 |
IC50 = 850 nM
|
|
|
|
CP0484082
|
4-chloro-2-methoxy-N-(2-oxochromen-6-yl)benzenesulfonamide
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|
C16H12ClNO5S
|
1
|
| 1 |
IC50 = 930 nM
|
|
|
|
CP0531584
|
4-tert-butyl-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C23H22N2O3S
|
1
|
| 1 |
IC50 = 1130 nM
|
|
|
|
CP0544168
|
2-chloro-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C19H13ClN2O3S
|
1
|
| 1 |
IC50 = 1250 nM
|
|
|
|
CP0575244
|
4-methoxy-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C20H16N2O4S
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
|
CP0475611
|
N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C19H14N2O3S
|
1
|
| 1 |
IC50 = 1640 nM
|
|
|
|
CP0475538
|
3-cyano-N-(6-oxo-5H-phenanthridin-2-yl)benzenesulfonamide
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|
C20H13N3O3S
|
1
|
| 1 |
IC50 = 1790 nM
|
|
|
|
CP0575216
|
N-(6-oxo-5H-phenanthridin-2-yl)-1-phenylmethanesulfonamide
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|
C20H16N2O3S
|
1
|
| 1 |
IC50 = 5170 nM
|
|
|
|
CP0576188
|
N-(6-oxo-5H-phenanthridin-2-yl)butane-1-sulfonamide
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|
C17H18N2O3S
|
1
|
| 1 |
IC50 = 5540 nM
|
|
|
|
CP0455551
|
N-(6-oxo-5H-phenanthridin-2-yl)cyclohexanesulfonamide
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|
C19H20N2O3S
|
1
|
| 1 |
IC50 = 5920 nM
|
|
|
|
CP0475555
|
phenyl N-(6-oxo-5H-phenanthridin-2-yl)carbamate
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|
C20H14N2O3
|
1
|
| 1 |
IC50 = 6020 nM
|
|
|
|
CP0475537
|
N-(6-oxo-5H-phenanthridin-2-yl)cyclopentanesulfonamide
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|
C18H18N2O3S
|
1
|
| 1 |
IC50 = 6170 nM
|
|
|
|
CP0475556
|
N-(6-oxo-5H-phenanthridin-2-yl)propane-1-sulfonamide
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|
C16H16N2O3S
|
1
|
| 1 |
IC50 = 6710 nM
|
|
|
|
CP0519434
|
N-(6-oxo-5H-phenanthridin-2-yl)thiophene-2-sulfonamide
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|
C17H12N2O3S2
|
1
|
| 1 |
IC50 = 6740 nM
|
|
|
|
CP0538043
|
N-(6-oxo-5H-phenanthridin-2-yl)naphthalene-2-sulfonamide
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|
C23H16N2O3S
|
1
|
| 1 |
IC50 = 7230 nM
|
|
|
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CP0476450
|
1-(6-oxo-5H-phenanthridin-2-yl)-3-phenylurea
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|
C20H15N3O2
|
1
|
| 1 |
IC50 = 9930 nM
|
|
|
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CP0575245
|
N-(6-oxo-5H-phenanthridin-2-yl)-2,3-dihydro-1-benzofuran-5-sulfonamide
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|
C21H16N2O4S
|
1
|
| 1 |
IC50 = 13120 nM
|
|
|
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CP0103977
|
N-(6-oxo-5H-phenanthridin-2-yl)benzamide
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|
C20H14N2O2
|
1
|
| 1 |
IC50 = 18610 nM
|
|
|
