| Compound ID |
Compound Name |
Compound Formula |
|
CP0542771
|
4-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamide
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|
C21H19FN2O2
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0546999
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-6-pyridin-4-ylpyridine-3-carboxamide
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|
C20H19N3O2
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0576408
|
6-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]pyridine-3-carboxamide
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|
C20H18FN3O2
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0574451
|
(2R)-N-[(1R)-1-(3-fluoro-5-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
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|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0574450
|
4-(3-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]piperazine-1-carboxamide
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|
C19H23FN4O2
|
1
|
| 1 |
IC50 = 1830 nM
|
|
|
|
CP0544232
|
(2R)-4-(3-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methylpiperazine-1-carboxamide
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|
C20H25FN4O2
|
1
|
| 1 |
IC50 = 2250 nM
|
|
|
|
CP0546163
|
(2R)-N-[(1R)-1-(4-fluoro-3-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
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|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 2340 nM
|
|
|
|
CP0571159
|
6-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]pyridazine-3-carboxamide
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|
C19H17FN4O2
|
1
|
| 1 |
IC50 = 3600 nM
|
|
|
|
CP0547000
|
CHEMBL5184099
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|
C21H26N2O2
|
1
|
| 1 |
IC50 = 5030 nM
|
|
|
|
CP0579459
|
(2R)-4-(3-fluoropyridin-4-yl)-2-methyl-N-[(1R)-1-pyrazolo[1,5-a]pyridin-4-ylethyl]piperazine-1-carboxamide
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|
C20H23FN6O
|
1
|
| 1 |
IC50 = 6650 nM
|
|
|
|
CP0576775
|
(2R)-4-(3-fluoropyridin-4-yl)-N-[(1R)-1-imidazo[1,2-a]pyridin-5-ylethyl]-2-methylpiperazine-1-carboxamide
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|
C20H23FN6O
|
1
|
| 1 |
IC50 = 8140 nM
|
|
|
|
CP0571313
|
(2R)-N-[(1R)-1-(2-chloro-5-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
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|
C20H24ClFN4O2
|
1
|
| 1 |
IC50 = 11600 nM
|
|
|
|
CP0569283
|
(2R)-N-[(1R)-1-(2-fluoro-5-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
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|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 13100 nM
|
|
|
|
CP0579036
|
(2R)-4-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methylpiperazine-1-carboxamide
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|
C20H25FN4O2
|
1
|
| 1 |
IC50 = 18900 nM
|
|
|
|
CP0551241
|
(2R,4R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
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|
C21H27N3O2
|
1
|
| 1 |
IC50 = 19400 nM
|
|
|
|
CP0572222
|
(2R,4S)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
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|
C21H27N3O2
|
1
|
| 1 |
IC50 = 23000 nM
|
|
|
|
CP0576410
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-ylcyclohexane-1-carboxamide
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|
C21H26N2O2
|
1
|
| 1 |
IC50 = 24300 nM
|
|
|
|
CP0542773
|
4-(3-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]piperidine-1-carboxamide
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|
C20H24FN3O2
|
1
|
| 1 |
IC50 = 31800 nM
|
|
|
|
CP0551242
|
(1S,2R,4S)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylcyclohexane-1-carboxamide
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|
C22H28N2O2
|
1
|
| 1 |
IC50 = 33800 nM
|
|
|
|
CP0547001
|
(2R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyrimidin-4-ylpiperazine-1-carboxamide
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|
C19H25N5O2
|
1
|
| 1 |
IC50 = 36500 nM
|
|
|
|
CP0576682
|
(2S,4S)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
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|
C21H27N3O2
|
1
|
| 1 |
IC50 = 48800 nM
|
|
|
|
CP0572223
|
(2R)-N-[(1R)-1-(2-fluoro-3-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
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|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 50900 nM
|
|
|
|
CP0542772
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-ylpiperidine-1-carboxamide
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|
C20H25N3O2
|
1
|
| 1 |
IC50 = 52800 nM
|
|
|
|
CP0574619
|
(2S,4R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
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|
C21H27N3O2
|
1
|
| 1 |
IC50 = 53700 nM
|
|
|
|
CP0382649
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C50H56BF2N7O7
|
1
|
| 1 |
Kd = 85 nM
|
|
|
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CP0382724
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C49H54BF2N7O7
|
1
|
| 1 |
Kd = 109 nM
|
|
|
