| Compound ID |
Compound Name |
Compound Formula |
|
CP0706752
|
(S)-2-Phenyl-5,7-dimethylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C26H32ClN7O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0777145
|
(S)-2,5,7-Trimethylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C21H30ClN7O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0834008
|
(S)-2-Phenyl-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C25H30ClN7O2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0726931
|
(S)-2-Methyl-7-hydroxypyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C19H26ClN7O3
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0818434
|
(S)-2-tert-Butyl-5,7-dimethylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C24H36ClN7O2
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0666465
|
N-[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl}amino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride
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|
C19H26ClN7O2
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0706751
|
(S)-2,7-Dimethylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C20H28ClN7O2
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0801137
|
(S)-2-tert-Butyl-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C23H34ClN7O2
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0822112
|
(S)-2-Methyl-7-trifluoromethylpyrazolo[1,5-a]pyrimidine-6-carboxylic acid{2-[(2-cyanopyrrolidin-1-yl)-2-oxoethylamino]-2-methylpropyl}amide hydrochloride
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|
C20H25ClF3N7O2
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0048107
|
(2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}pyrrolidine-2-carbonitrile
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|
C17H25N3O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0354373
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-6-fluorobenzoic acid
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|
C21H23FN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0382978
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-5-fluorobenzoic acid
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|
C21H23FN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0412141
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-4-methoxybenzoic acid
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|
C22H26N4O5
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0412280
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-5-bromobenzoic acid
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|
C21H23BrN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0412282
|
methyl 2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-4-bromobenzoate
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|
C22H25BrN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0412283
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-4-bromobenzoic acid
Show/Hide
|
C21H23BrN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0437966
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]benzoic acid
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|
C21H24N4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0470488
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-4-cyanobenzoic acid
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|
C22H23N5O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0470490
|
2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-5-chlorobenzoic acid
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|
C21H23ClN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0551453
|
methyl 2-[[4-[(3R)-3-aminopiperidin-1-yl]-3-but-2-ynyl-2,6-dioxopyrimidin-1-yl]methyl]-6-fluorobenzoate
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|
C22H25FN4O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
