| Compound ID |
Compound Name |
Compound Formula |
|
CP0307541
|
N-[4-(4-methylpiperazine-1-carbonyl)-2-phenylphenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C25H23N5O3S
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
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CP0573834
|
N-[2-(1-fluoroethoxy)-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C21H22FN5O4S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
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CP0386393
|
N-[4-(4-methylpiperazine-1-carbonyl)-2-propan-2-ylphenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C22H25N5O3S
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
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CP0574865
|
N-[2-(dimethylamino)-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C21H24N6O3S
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
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CP0469576
|
N-[2-(1,1,1,3,3,3-hexafluoropropan-2-yloxy)-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C22H19F6N5O4S
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
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CP0560906
|
N-[2-chloro-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C19H18ClN5O3S
|
1
|
| 1 |
IC50 = 5.8 nM
|
|
|
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CP0555432
|
N-[2-cyclohexyl-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C25H29N5O3S
|
1
|
| 1 |
IC50 = 6.7 nM
|
|
|
|
CP0454723
|
N-[2-bromo-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C19H18BrN5O3S
|
1
|
| 1 |
IC50 = 7.3 nM
|
|
|
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CP0454724
|
N-[2-[ethyl(methyl)amino]-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C22H26N6O3S
|
1
|
| 1 |
IC50 = 9.3 nM
|
|
|
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CP0234174
|
N-[3-(4-methylpiperazine-1-carbonyl)-2-propan-2-yloxyphenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C22H25N5O4S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0555434
|
N-[2-methoxy-4-[3-(4-methylpiperazin-1-yl)propylcarbamoyl]phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C23H28N6O4S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0459410
|
N-[2-methoxy-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C20H21N5O4S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0557064
|
N-[2-methyl-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C20H21N5O3S
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
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CP0420720
|
N-[2-fluoro-4-(4-methylpiperazine-1-carbonyl)phenyl]-4-oxo-3H-thieno[3,2-d]pyrimidine-7-carboxamide
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|
C19H18FN5O3S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0469568
|
N-[2-methoxy-4-[3-(4-methylpiperazin-1-yl)propylcarbamoyl]phenyl]thieno[3,2-d]pyrimidine-7-carboxamide
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|
C23H28N6O3S
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0532331
|
N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]thieno[3,2-d]pyrimidine-7-carboxamide
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|
C19H21N5O2S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
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CP0420723
|
N-[2-methoxy-4-(4-methylpiperazine-1-carbonyl)phenyl]thieno[3,2-d]pyrimidine-7-carboxamide
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|
C20H21N5O3S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
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CP0432894
|
1-[5-(4-methylpiperazin-1-yl)naphthalen-2-yl]-3-[4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]urea
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|
C29H28N6O2
|
1
|
| 1 |
Kd = 12 nM
|
|
|
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CP0382724
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C49H54BF2N7O7
|
1
|
| 1 |
Kd = 44 nM
|
|
|
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CP0088463
|
US9255110, 17
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|
C17H12N4O2S
|
2
|
| 1 |
Kd = 59 nM
|
|
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| 2 |
Kd = 150 nM
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CP0382649
|
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
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|
C50H56BF2N7O7
|
1
|
| 1 |
Kd = 60 nM
|
|
|
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CP0018477
|
4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-N-methylpyridine-2-carboxamide
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|
C21H16ClF3N4O3
|
2
|
| 1 |
Kd = 600 nM
|
|
|
| 2 |
Kd = 1300 nM
|
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CP0029805
|
({[({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}oxy)phosphonic acid
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|
C10H16N5O13P3
|
1
|
| 1 |
Kd = 2800 nM
|
|
|
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CP0043494
|
ADP
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|
C10H15N5O10P2
|
2
|
| 1 |
Kd = 4100 nM
|
|
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| 2 |
Kd = 63000 nM
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|
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CP0001102
|
(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol
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|
C10H13N5O4
|
2
|
| 1 |
Kd = 4400 nM
|
|
|
| 2 |
Kd = 34000 nM
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