| Compound ID |
Compound Name |
Compound Formula |
|
CP0126650
|
5-methyl-8-(1H-pyrrol-2-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C15H12N4O
|
1
|
| 1 |
IC50 = 0.1 nM
|
|
|
|
CP0310520
|
5-methyl-8-(1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C14H11N5O
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0501885
|
5-methyl-8-(4-(piperazin-1-ylmethyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C22H23N5O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0502436
|
5-methyl-8-(3-(piperazin-1-ylmethyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C22H23N5O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0506032
|
5-methyl-8-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C23H25N5O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0514463
|
5-methyl-8-(4-(morpholinomethyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C22H22N4O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0088592
|
8-(4-(hydroxymethyl)phenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C18H15N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0489440
|
8-(4-(2-(diethylamino)ethoxy)phenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C23H26N4O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0502437
|
8-(furan-2-yl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C15H11N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0435748
|
10-Hydroxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrolo[3,4-c]carbazole-5,7-(6H,12H)-dione
Show/Hide
|
C19H10N4O3
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0531236
|
5-METHYL-8-PYRIDIN-4-YL[1,2,4]TRIAZOLO[4,3-A]QUINOLIN-1(2H)-ONE
Show/Hide
|
C16H12N4O
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0083030
|
11H-2,5,11-triaza-benzo[a]trindene-1,3,4,6-tetraone
Show/Hide
|
C16H7N3O4
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0151078
|
5-methyl-8-(thiophen-2-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C15H11N3OS
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0523806
|
N-ethyl-4-(5-methyl-1-oxo-2H-[1,2,4]triazolo[4,3-a]quinolin-8-yl)benzamide
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0345050
|
4,7,11-trihydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2H,8H)-dione
Show/Hide
|
C18H10N2O5
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0412551
|
10-Benzyloxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]-pyrrolo[3,4-c]carbazole-5,7-(6H,12H)-dione
Show/Hide
|
C26H16N4O3
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0479267
|
5-methyl-8-(1H-pyrrol-3-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C15H12N4O
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0641259
|
11-hydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(2H,8H)-tetraone
Show/Hide
|
C18H8N2O5
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0528439
|
9-Hydroxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrolo[3,4-c]carbazole-5,7-(6H,12H)-dione
Show/Hide
|
C19H10N4O3
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0489441
|
5-methyl-8-(4-(2-morpholinoethoxy)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C23H24N4O3
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0385494
|
4-(5-methyl-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinolin-8-yl)benzamide
Show/Hide
|
C18H14N4O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0489444
|
5-methyl-8-(4-((methylamino)methyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C19H18N4O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0501886
|
8-(3-(hydroxymethyl)phenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C18H15N3O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0144754
|
6,7-dihydro-1H-cyclopenta[a]pyrrolo[3,4-c]carbazole-1,3,4-(2H,5H)-trione
Show/Hide
|
C17H10N2O3
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0522102
|
8-(4-hydroxy-3-methylphenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C18H15N3O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0479261
|
5-methyl-8-(4-(morpholine-4-carbonyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C22H20N4O3
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0479265
|
5-methyl-8-(4-methylthiophen-2-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C16H13N3OS
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0021175
|
1,11-dihydro-1,3,5,11-tetraaza-benzo[a]trindene-4,6-dione
Show/Hide
|
C15H8N4O2
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0489442
|
5-methyl-8-(4-(methylsulfinyl)phenyl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C18H15N3O2S
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0511448
|
4-(5-methyl-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinolin-8-yl)benzonitrile
Show/Hide
|
C18H12N4O
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0523805
|
8-(4-hydroxyphenyl)-5-methyl-2H-[1,2,4]triazolo[4,3-a]quinolin-1-one
Show/Hide
|
C17H13N3O2
|
1
|
| 1 |
IC50 < 100 nM
|
|
|
|
CP0826879
|
11-methylbenzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(2H,8H)-tetraone
Show/Hide
|
C19H10N2O4
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0506033
|
5-methyl-8-(pyridin-3-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C16H12N4O
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0514464
|
8-(1H-imidazol-4-yl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C14H11N5O
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0015449
|
4,7-dihydroxy-11-methylbenzo[a]pyrrolo[3,4-c]carbazole-1,3-(2H,8H)-dione
Show/Hide
|
C19H12N2O4
|
1
|
| 1 |
IC50 = 161 nM
|
|
|
|
CP0541588
|
8-(3-hydroxyphenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C17H13N3O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0533330
|
2-(4-(5-methyl-1-oxo-1,2-dihydro-[1,2,4]triazolo[4,3-a]quinolin-8-yl)phenyl)acetonitrile
Show/Hide
|
C19H14N4O
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0541513
|
N-[4-(5-methyl-1-oxo-2H-[1,2,4]triazolo[4,3-a]quinolin-8-yl)phenyl]acetamide
Show/Hide
|
C19H16N4O2
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0684598
|
benzo[a]pyrrolo[3,4-c]carbazole-1,3,4,7(2H,8H)-tetraone
Show/Hide
|
C18H8N2O4
|
1
|
| 1 |
IC50 = 269 nM
|
|
|
|
CP0144722
|
4,7-dihydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2H,8H)-dione
Show/Hide
|
C18H10N2O4
|
1
|
| 1 |
IC50 = 311 nM
|
|
|
|
CP0016545
|
11H-2,5,11,11b-Tetraaza-benzo[a]trindene-4,6-dione
Show/Hide
|
C15H8N4O2
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0501884
|
8-(4-methoxyphenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C18H15N3O2
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0372484
|
8-(2-(hydroxymethyl)phenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C18H15N3O2
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0529728
|
4-hydroxy-11-methyl-7-hydroxysulfonyloxybenzo[a]pyrrolo-[3,4-c]carbazole-1,3(2H,8H)-dione
Show/Hide
|
C19H12N2O7S
|
1
|
| 1 |
IC50 = 893 nM
|
|
|
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CP0185307
|
4-hydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2H,8H)-dione
Show/Hide
|
C18H10N2O3
|
1
|
| 1 |
IC50 = 904 nM
|
|
|
|
CP0457476
|
9-Benzyloxy-1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6H,12H)-dione
Show/Hide
|
C26H16N4O3
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
|
CP0522103
|
5-methyl-8-(pyrazin-2-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C15H11N5O
|
1
|
| 1 |
IC50 = 1590 nM
|
|
|
|
CP0531235
|
N-methyl-4-(5-methyl-1-oxo-2H-[1,2,4]triazolo[4,3-a]quinolin-8-yl)benzamide
Show/Hide
|
C19H16N4O2
|
1
|
| 1 |
IC50 = 1590 nM
|
|
|
|
CP0489446
|
8-(furan-3-yl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C15H11N3O2
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0449053
|
4-hydroxy-7-hydroxysulfonyloxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2H,8H)-dione
Show/Hide
|
C18H10N2O7S
|
1
|
| 1 |
IC50 = 1790 nM
|
|
|
|
CP0508111
|
5-methyl-8-(thiazol-2-yl)-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C14H10N4OS
|
1
|
| 1 |
IC50 = 2960 nM
|
|
|
|
CP0489445
|
8-(4-(methoxymethyl)phenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C19H17N3O2
|
1
|
| 1 |
IC50 = 3490 nM
|
|
|
|
CP0378540
|
7-tert-butylcarbonyloxy-4-hydroxybenzo[a]pyrrolo[3,4-c]carbazole-1,3(2H,8H)-dione
Show/Hide
|
C23H18N2O5
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
|
CP0436458
|
1H-pyrido[3'4':4,5]pyrrolo[2,3-a]pyrrolo[3,4-c]-carbazole-5,7-(6H,12H)-dione
Show/Hide
|
C19H10N4O2
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0436503
|
10-Hydroxy-6-methyl-1H-pyrido[3'4':4,5]pyrrolo-[2,3-a]pyrrolo[3,4-c]carbazole-5,7-(6H,12H)-dione
Show/Hide
|
C20H12N4O3
|
1
|
| 1 |
IC50 = 5000 nM
|
|
|
|
CP0489443
|
8-(2-aminophenyl)-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1(2H)-one
Show/Hide
|
C17H14N4O
|
1
|
| 1 |
IC50 = 24400 nM
|
|
|
