Compound ID |
Compound Name |
Compound Formula |
CP0442136
|
US8802673, 211
Show/Hide
|
C16H16ClF3N4O2
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0491107
|
US8802673, 194
Show/Hide
|
C17H19ClN4O
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0539099
|
US8802673, 171
Show/Hide
|
C17H19ClN4O
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0536190
|
US8802673, 170
Show/Hide
|
C17H19ClN4O
|
1
|
1 |
Ki = 1.2 nM
|
|
|
CP0384786
|
US8802673, 149
Show/Hide
|
C17H19ClN4O
|
1
|
1 |
Ki = 1.4 nM
|
|
|
CP0520648
|
US8802673, 203
Show/Hide
|
C16H16ClF3N4O2
|
1
|
1 |
Ki = 1.7 nM
|
|
|
CP0491106
|
US8802673, 184
Show/Hide
|
C16H16ClF3N4O2
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0491109
|
US8802673, 204
Show/Hide
|
C15H14ClF3N4O
|
1
|
1 |
Ki = 2.1 nM
|
|
|
CP0442942
|
US8802673, 209
Show/Hide
|
C16H15F5N4O2
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0484454
|
US8802673, 137
Show/Hide
|
C16H17F3N4O2
|
1
|
1 |
Ki = 2.6 nM
|
|
|
CP0521300
|
US8802673, 192
Show/Hide
|
C17H19FN4O
|
1
|
1 |
Ki = 2.6 nM
|
|
|
CP0528997
|
US8802673, 118
Show/Hide
|
C17H19FN4O
|
1
|
1 |
Ki = 3 nM
|
|
|
CP0516796
|
US8802673, 188
Show/Hide
|
C16H16F4N4O2
|
1
|
1 |
Ki = 3.3 nM
|
|
|
CP0520283
|
US8802673, 98
Show/Hide
|
C17H19FN4O
|
1
|
1 |
Ki = 3.3 nM
|
|
|
CP0539102
|
US8802673, 208
Show/Hide
|
C16H16F4N4O2
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0503591
|
US8802673, 128
Show/Hide
|
C17H21FN4O
|
1
|
1 |
Ki = 3.9 nM
|
|
|
CP0539101
|
US8802673, 196
Show/Hide
|
C15H14F4N4O
|
1
|
1 |
Ki = 4 nM
|
|
|
CP0535952
|
US8802673, 101
Show/Hide
|
C17H21FN4O
|
1
|
1 |
Ki = 4.1 nM
|
|
|
CP0491093
|
US8802673, 53
Show/Hide
|
C19H18BrN3O
|
1
|
1 |
Ki = 4.5 nM
|
|
|
CP0503700
|
US8802673, 144
Show/Hide
|
C16H16F4N4O2
|
1
|
1 |
Ki = 4.9 nM
|
|
|
CP0500141
|
US8802673, 119
Show/Hide
|
C17H19FN4O
|
1
|
1 |
Ki = 5.1 nM
|
|
|
CP0499823
|
US8802673, 97
Show/Hide
|
C16H19FN4O
|
1
|
1 |
Ki = 5.6 nM
|
|
|
CP0531765
|
US8802673, 202
Show/Hide
|
C14H14Cl2N4O
|
1
|
1 |
Ki = 6.5 nM
|
|
|
CP0491105
|
US8802673, 175
Show/Hide
|
C19H17ClF2N6O3
|
1
|
1 |
Ki = 6.6 nM
|
|
|
CP0503586
|
US8802673, 47
Show/Hide
|
C19H18ClN3O
|
1
|
1 |
Ki = 6.7 nM
|
|
|
CP0529249
|
US8802673, 145
Show/Hide
|
C16H16F4N4O2
|
1
|
1 |
Ki = 6.7 nM
|
|
|
CP0471189
|
US8802673, 129
Show/Hide
|
C17H21FN4O
|
1
|
1 |
Ki = 6.8 nM
|
|
|
CP0535954
|
US8802673, 116
Show/Hide
|
C16H19FN4O
|
1
|
1 |
Ki = 7 nM
|
|
|
CP0520660
|
US8802673, 134
Show/Hide
|
C15H14F4N4O
|
1
|
1 |
Ki = 7.9 nM
|
|
|
CP0509209
|
US8802673, 148
Show/Hide
|
C18H18N4O2
|
1
|
1 |
Ki = 8.3 nM
|
|
|
CP0519047
|
US8802673, 26
Show/Hide
|
C17H16ClN3OS
|
1
|
1 |
Ki = 8.3 nM
|
|
|
CP0555392
|
US8802673, 52
Show/Hide
|
C19H18ClN3O
|
1
|
1 |
Ki = 8.4 nM
|
|
|
CP0491098
|
US8802673, 86
Show/Hide
|
C17H20N4O
|
1
|
1 |
Ki = 9 nM
|
|
|
CP0491094
|
US8802673, 62
Show/Hide
|
C16H18BrN3O
|
1
|
1 |
Ki = 9.4 nM
|
|
|
CP0450195
|
US8802673, 121
Show/Hide
|
C15H14F4N4O
|
1
|
1 |
Ki = 9.6 nM
|
|
|
CP0450198
|
US8802673, 126
Show/Hide
|
C14H14BrFN4O
|
1
|
1 |
Ki = 9.6 nM
|
|
|
CP0520647
|
US8802673, 187
Show/Hide
|
C16H17F3N4O2
|
1
|
1 |
Ki = 10 nM
|
|
|
CP0491096
|
US8802673, 82
Show/Hide
|
C16H15ClF3N3O
|
1
|
1 |
Ki = 10.1 nM
|
|
|
CP0484467
|
US8802673, 207
Show/Hide
|
C16H16F4N4O2
|
1
|
1 |
Ki = 10.2 nM
|
|
|
CP0471188
|
US8802673, 117
Show/Hide
|
C16H19FN4O
|
1
|
1 |
Ki = 10.4 nM
|
|
|
CP0500335
|
US8802673, 44
Show/Hide
|
C20H20N2O
|
1
|
1 |
Ki = 11.8 nM
|
|
|
CP0512149
|
US8802673, 102
Show/Hide
|
C14H14BrFN4O
|
1
|
1 |
Ki = 12.6 nM
|
|
|
CP0384785
|
US8802673, 141
Show/Hide
|
C22H24N4O3
|
1
|
1 |
Ki = 12.9 nM
|
|
|
CP0553826
|
US8802673, 17
Show/Hide
|
C17H20N4O
|
1
|
1 |
Ki = 13.1 nM
|
|
|
CP0519048
|
US8802673, 54
Show/Hide
|
C19H18ClN3O
|
1
|
1 |
Ki = 13.8 nM
|
|
|
CP0509208
|
US8802673, 142
Show/Hide
|
C22H24N4O3
|
1
|
1 |
Ki = 14.6 nM
|
|
|
CP0551298
|
US8802673, 172
Show/Hide
|
C16H17F3N4O2
|
1
|
1 |
Ki = 16.2 nM
|
|
|
CP0520659
|
US8802673, 100
Show/Hide
|
C16H19FN4O2
|
1
|
1 |
Ki = 16.4 nM
|
|
|
CP0503699
|
US8802673, 127
Show/Hide
|
C14H14BrFN4O
|
1
|
1 |
Ki = 16.5 nM
|
|
|
CP0442874
|
US8802673, 34
Show/Hide
|
C18H21ClN2O
|
1
|
1 |
Ki = 18.1 nM
|
|
|
CP0512152
|
US8802673, 132
Show/Hide
|
C16H19FN4O2
|
1
|
1 |
Ki = 18.2 nM
|
|
|
CP0490531
|
US8802673, 99
Show/Hide
|
C15H15ClFN3O
|
1
|
1 |
Ki = 18.5 nM
|
|
|
CP0491097
|
US8802673, 85
Show/Hide
|
C17H20BrN3O
|
1
|
1 |
Ki = 19.4 nM
|
|
|
CP0524425
|
US8802673, 193
Show/Hide
|
C17H19ClN4O
|
1
|
1 |
Ki = 19.6 nM
|
|
|
CP0524421
|
US8802673, 147
Show/Hide
|
C18H18N4O2
|
1
|
1 |
Ki = 19.7 nM
|
|
|
CP0503593
|
US8802673, 135
Show/Hide
|
C15H14F4N4O
|
1
|
1 |
Ki = 19.8 nM
|
|
|
CP0471190
|
US8802673, 130
Show/Hide
|
C14H14ClFN4O
|
1
|
1 |
Ki = 19.9 nM
|
|
|
CP0529271
|
US8802673, 96
Show/Hide
|
C14H14ClFN4O
|
1
|
1 |
Ki = 21.6 nM
|
|
|
CP0520281
|
US8802673, 83
Show/Hide
|
C16H18ClN3O
|
1
|
1 |
Ki = 22.2 nM
|
|
|
CP0520282
|
US8802673, 93
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 22.2 nM
|
|
|
CP0536243
|
US8802673, 95
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 22.3 nM
|
|
|
CP0443849
|
US8802673, 11
Show/Hide
|
C16H16F3N3O
|
1
|
1 |
Ki = 23.3 nM
|
|
|
CP0530404
|
US8802673, 19
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 23.6 nM
|
|
|
CP0541879
|
US8802673, 21
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 24.5 nM
|
|
|
CP0491088
|
US8802673, 164
Show/Hide
|
C19H20N4O
|
1
|
1 |
Ki = 25 nM
|
|
|
CP0450191
|
US8802673, 3
Show/Hide
|
C20H22ClF3N2
|
1
|
1 |
Ki = 25.1 nM
|
|
|
CP0500138
|
US8802673, 195
Show/Hide
|
C17H19FN4O
|
1
|
1 |
Ki = 25.2 nM
|
|
|
CP0553831
|
US8802673, 210
Show/Hide
|
C14H14ClFN4O
|
1
|
1 |
Ki = 26.6 nM
|
|
|
CP0450197
|
US8802673, 125
Show/Hide
|
C18H22N4O2
|
1
|
1 |
Ki = 27.8 nM
|
|
|
CP0520649
|
US8802673, 5
Show/Hide
|
C15H16ClN3O
|
1
|
1 |
Ki = 29 nM
|
|
|
CP0520658
|
US8802673, 74
Show/Hide
|
C18H22N4O
|
1
|
1 |
Ki = 29.5 nM
|
|
|
CP0503715
|
US8802673, 178
Show/Hide
|
C16H17F3N4O
|
1
|
1 |
Ki = 29.8 nM
|
|
|
CP0442958
|
US8802673, 177
Show/Hide
|
C18H18N4O
|
1
|
1 |
Ki = 29.9 nM
|
|
|
CP0539097
|
US8802673, 110
Show/Hide
|
C18H22N4O
|
1
|
1 |
Ki = 30.6 nM
|
|
|
CP0491108
|
US8802673, 197
Show/Hide
|
C15H14F4N4O
|
1
|
1 |
Ki = 31.5 nM
|
|
|
CP0535953
|
US8802673, 111
Show/Hide
|
C18H22N4O
|
1
|
1 |
Ki = 32.2 nM
|
|
|
CP0519044
|
US8802673, 8
Show/Hide
|
C16H17ClN2O
|
1
|
1 |
Ki = 32.5 nM
|
|
|
CP0520661
|
US8802673, 180
Show/Hide
|
C15H17ClN4O2
|
1
|
1 |
Ki = 33 nM
|
|
|
CP0524404
|
US8802673, 163
Show/Hide
|
C19H20N4O
|
1
|
1 |
Ki = 33.2 nM
|
|
|
CP0519045
|
US8802673, 10
Show/Hide
|
C15H16BrN3O
|
1
|
1 |
Ki = 33.7 nM
|
|
|
CP0450196
|
US8802673, 124
Show/Hide
|
C18H22N4O2
|
1
|
1 |
Ki = 34.8 nM
|
|
|
CP0443856
|
US8802673, 73
Show/Hide
|
C18H24N4O
|
1
|
1 |
Ki = 35 nM
|
|
|
CP0442897
|
US8802673, 120
Show/Hide
|
C15H17BrN4O
|
1
|
1 |
Ki = 36.4 nM
|
|
|
CP0536242
|
US8802673, 87
Show/Hide
|
C18H22N4O
|
1
|
1 |
Ki = 37 nM
|
|
|
CP0531662
|
US8802673, 131
Show/Hide
|
C14H14ClFN4O
|
1
|
1 |
Ki = 37.9 nM
|
|
|
CP0535955
|
US8802673, 133
Show/Hide
|
C16H19FN4O2
|
1
|
1 |
Ki = 38.7 nM
|
|
|
CP0442130
|
US8802673, 30
Show/Hide
|
C17H18Cl2N2O
|
1
|
1 |
Ki = 41.7 nM
|
|
|
CP0442134
|
US8802673, 190
Show/Hide
|
C17H19FN4O
|
1
|
1 |
Ki = 42.2 nM
|
|
|
CP0555390
|
US8802673, 7
Show/Hide
|
C14H15BrN4O
|
1
|
1 |
Ki = 42.5 nM
|
|
|
CP0449984
|
US8802673, 69
Show/Hide
|
C15H16ClN3O
|
1
|
1 |
Ki = 43.8 nM
|
|
|
CP0550088
|
US8802673, 76
Show/Hide
|
C16H18BrN3O
|
1
|
1 |
Ki = 45 nM
|
|
|
CP0450192
|
US8802673, 15
Show/Hide
|
C16H20N4O
|
1
|
1 |
Ki = 46.6 nM
|
|
|
CP0484453
|
US8802673, 94
Show/Hide
|
C14H15BrN4O
|
1
|
1 |
Ki = 48.9 nM
|
|
|
CP0528999
|
US8802673, 136
Show/Hide
|
C16H17F3N4O2
|
1
|
1 |
Ki = 49.4 nM
|
|
|
CP0442896
|
US8802673, 103
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 50 nM
|
|
|
CP0539100
|
US8802673, 179
Show/Hide
|
C15H16F2N4O2
|
1
|
1 |
Ki = 51.7 nM
|
|
|
CP0442891
|
US8802673, 42
Show/Hide
|
C16H16F3N3O
|
1
|
1 |
Ki = 51.8 nM
|
|
|
CP0442876
|
US8802673, 38
Show/Hide
|
C15H16ClN3O
|
1
|
1 |
Ki = 54.4 nM
|
|
|
CP0550485
|
US8802673, 199
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 56 nM
|
|
|
CP0519050
|
US8802673, 84
Show/Hide
|
C17H20ClN3O
|
1
|
1 |
Ki = 57 nM
|
|
|
CP0520662
|
US8802673, 200
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 58.8 nM
|
|
|
CP0500144
|
US8802673, 189
Show/Hide
|
C17H20N4O
|
1
|
1 |
Ki = 60.5 nM
|
|
|
CP0503587
|
US8802673, 50
Show/Hide
|
C18H17ClN4O
|
1
|
1 |
Ki = 60.8 nM
|
|
|
CP0516775
|
US8802673, 173
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 62.5 nM
|
|
|
CP0442895
|
US8802673, 80
Show/Hide
|
C16H18ClN3O
|
1
|
1 |
Ki = 62.6 nM
|
|
|
CP0442941
|
US8802673, 201
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 62.6 nM
|
|
|
CP0500143
|
US8802673, 174
Show/Hide
|
C19H18F2N6O3
|
1
|
1 |
Ki = 62.8 nM
|
|
|
CP0524416
|
US8802673, 46
Show/Hide
|
C19H19N3O
|
1
|
1 |
Ki = 64.3 nM
|
|
|
CP0486058
|
US8802673, 25
Show/Hide
|
C18H19F3N2O2
|
1
|
1 |
Ki = 70.5 nM
|
|
|
CP0520280
|
US8802673, 79
Show/Hide
|
C17H19ClN2O
|
1
|
1 |
Ki = 71.6 nM
|
|
|
CP0443853
|
US8802673, 68
Show/Hide
|
C16H20N4O
|
1
|
1 |
Ki = 75.1 nM
|
|
|
CP0516778
|
US8802673, 4
Show/Hide
|
C21H24ClF3N2
|
1
|
1 |
Ki = 78.5 nM
|
|
|
CP0503698
|
US8802673, 123
Show/Hide
|
C17H22N4O2
|
1
|
1 |
Ki = 79.6 nM
|
|
|
CP0536244
|
US8802673, 106
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 81.4 nM
|
|
|
CP0536245
|
US8802673, 122
Show/Hide
|
C17H22N4O2
|
1
|
1 |
Ki = 84.7 nM
|
|
|
CP0503589
|
US8802673, 57
Show/Hide
|
C15H15BrFN3O
|
1
|
1 |
Ki = 86.6 nM
|
|
|
CP0530622
|
US8802673, 88
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 87.4 nM
|
|
|
CP0490532
|
US8802673, 113
Show/Hide
|
C19H20N4O
|
1
|
1 |
Ki = 87.7 nM
|
|
|
CP0499824
|
US8802673, 107
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 87.7 nM
|
|
|
CP0426462
|
US8802673, 185
Show/Hide
|
C16H15ClF3N3O
|
1
|
1 |
Ki = 88.8 nM
|
|
|
CP0516779
|
US8802673, 9
Show/Hide
|
C17H19ClN2O
|
1
|
1 |
Ki = 89.3 nM
|
|
|
CP0553829
|
US8802673, 151
Show/Hide
|
C17H21FN4O3
|
1
|
1 |
Ki = 95.4 nM
|
|
|
CP0524443
|
US8802673, 206
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 96.3 nM
|
|
|
CP0521217
|
US8802673, 64
Show/Hide
|
C16H18BrN3O
|
1
|
1 |
Ki = 101 nM
|
|
|
CP0550263
|
US8802673, 49
Show/Hide
|
C21H17F6N3O
|
1
|
1 |
Ki = 103.8 nM
|
|
|
CP0512150
|
US8802673, 104
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 104.8 nM
|
|
|
CP0530402
|
US8802673, 13
Show/Hide
|
C18H22N2O
|
1
|
1 |
Ki = 108.5 nM
|
|
|
CP0499822
|
US8802673, 91
Show/Hide
|
C14H15BrN4O
|
1
|
1 |
Ki = 123.3 nM
|
|
|
CP0500336
|
US8802673, 45
Show/Hide
|
C17H19BrN2O
|
1
|
1 |
Ki = 126.1 nM
|
|
|
CP0449985
|
US8802673, 105
Show/Hide
|
C16H20N4O2
|
1
|
1 |
Ki = 126.5 nM
|
|
|
CP0384789
|
US8802673, 162
Show/Hide
|
C20H22N4O
|
1
|
1 |
Ki = 127.3 nM
|
|
|
CP0550264
|
US8802673, 77
Show/Hide
|
C15H15ClFN3O
|
1
|
1 |
Ki = 130.4 nM
|
|
|
CP0539098
|
US8802673, 146
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 140.4 nM
|
|
|
CP0536246
|
US8802673, 150
Show/Hide
|
C15H18F2N4O
|
1
|
1 |
Ki = 148.6 nM
|
|
|
CP0519046
|
US8802673, 24
Show/Hide
|
C18H19F3N2O
|
1
|
1 |
Ki = 149 nM
|
|
|
CP0530405
|
US8802673, 29
Show/Hide
|
C16H20N4O2
|
1
|
1 |
Ki = 155.5 nM
|
|
|
CP0491104
|
US8802673, 166
Show/Hide
|
C16H17F3N4O
|
1
|
1 |
Ki = 158.9 nM
|
|
|
CP0442135
|
US8802673, 205
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 162.1 nM
|
|
|
CP0553830
|
US8802673, 198
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 162.8 nM
|
|
|
CP0539094
|
US8802673, 36
Show/Hide
|
C19H24N2O
|
1
|
1 |
Ki = 163.3 nM
|
|
|
CP0443855
|
US8802673, 71
Show/Hide
|
C17H20ClN3O2
|
1
|
1 |
Ki = 168 nM
|
|
|
CP0491091
|
US8802673, 183
Show/Hide
|
C16H20N4O3
|
1
|
1 |
Ki = 173.7 nM
|
|
|
CP0512148
|
US8802673, 89
Show/Hide
|
C15H17BrN4O
|
1
|
1 |
Ki = 176.7 nM
|
|
|
CP0442132
|
US8802673, 40
Show/Hide
|
C15H15ClFN3O
|
1
|
1 |
Ki = 188.2 nM
|
|
|
CP0550087
|
US8802673, 35
Show/Hide
|
C17H18ClFN2O
|
1
|
1 |
Ki = 188.3 nM
|
|
|
CP0503590
|
US8802673, 112
Show/Hide
|
C17H22N4
|
1
|
1 |
Ki = 196.6 nM
|
|
|
CP0550089
|
US8802673, 81
Show/Hide
|
C15H17ClN4O
|
1
|
1 |
Ki = 202.7 nM
|
|
|
CP0500140
|
US8802673, 59
Show/Hide
|
C16H16ClFN2O
|
1
|
1 |
Ki = 207.3 nM
|
|
|
CP0519049
|
US8802673, 56
Show/Hide
|
C16H18BrN3O
|
1
|
1 |
Ki = 211 nM
|
|
|
CP0470194
|
US8802673, 108
Show/Hide
|
C14H15BrN4O
|
1
|
1 |
Ki = 215.7 nM
|
|
|
CP0530406
|
US8802673, 72
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 220 nM
|
|
|
CP0553827
|
US8802673, 31
Show/Hide
|
C17H19FN2O
|
1
|
1 |
Ki = 222.2 nM
|
|
|
CP0400449
|
US8802673, 161
Show/Hide
|
C20H22N4O
|
1
|
1 |
Ki = 222.9 nM
|
|
|
CP0530407
|
US8802673, 75
Show/Hide
|
C14H15N5O3
|
1
|
1 |
Ki = 228 nM
|
|
|
CP0442943
|
US8802673, 6
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 232.2 nM
|
|
|
CP0491099
|
US8802673, 90
Show/Hide
|
C14H15ClN4O
|
1
|
1 |
Ki = 232.4 nM
|
|
|
CP0553828
|
US8802673, 48
Show/Hide
|
C20H21N3O
|
1
|
1 |
Ki = 233.6 nM
|
|
|
CP0530408
|
US8802673, 115
Show/Hide
|
C18H18N4O2
|
1
|
1 |
Ki = 234.9 nM
|
|
|
CP0566202
|
US8802673, 39
Show/Hide
|
C16H19N3O2
|
1
|
1 |
Ki = 251.4 nM
|
|
|
CP0521218
|
US8802673, 66
Show/Hide
|
C19H18BrN3O
|
1
|
1 |
Ki = 256.9 nM
|
|
|
CP0443850
|
US8802673, 12
Show/Hide
|
C15H18N4O2
|
1
|
1 |
Ki = 258.8 nM
|
|
|
CP0424108
|
US8802673, 152
Show/Hide
|
C17H21FN4O3
|
1
|
1 |
Ki = 267.7 nM
|
|
|
CP0490530
|
US8802673, 92
Show/Hide
|
C16H19N5O
|
1
|
1 |
Ki = 274.8 nM
|
|
|
CP0491092
|
US8802673, 51
Show/Hide
|
C20H20ClN3O
|
1
|
1 |
Ki = 280.3 nM
|
|
|
CP0491103
|
US8802673, 143
Show/Hide
|
C14H17BrN4O
|
1
|
1 |
Ki = 283.6 nM
|
|
|
CP0490529
|
US8802673, 67
Show/Hide
|
C15H16ClN3O
|
1
|
1 |
Ki = 291.7 nM
|
|
|
CP0521211
|
US8802673, 18
Show/Hide
|
C15H18N4O
|
1
|
1 |
Ki = 313.3 nM
|
|
|
CP0509210
|
US8802673, 165
Show/Hide
|
C18H21N3O2
|
1
|
1 |
Ki = 339.5 nM
|
|
|
CP0512151
|
US8802673, 109
Show/Hide
|
C14H15BrN4O
|
1
|
1 |
Ki = 362.4 nM
|
|
|
CP0491090
|
US8802673, 181
Show/Hide
|
C15H15N5O
|
1
|
1 |
Ki = 398.1 nM
|
|
|
CP0529250
|
US8802673, 182
Show/Hide
|
C16H20N4O
|
1
|
1 |
Ki = 446.5 nM
|
|
|
CP0521210
|
US8802673, 16
Show/Hide
|
C15H15N5O
|
1
|
1 |
Ki = 448.3 nM
|
|
|
CP0539093
|
US8802673, 22
Show/Hide
|
C18H22N2O
|
1
|
1 |
Ki = 468 nM
|
|
|
CP0450193
|
US8802673, 61
Show/Hide
|
C15H15Br2N3O
|
1
|
1 |
Ki = 502.4 nM
|
|
|
CP0530403
|
US8802673, 14
Show/Hide
|
C14H15FN4O
|
1
|
1 |
Ki = 504 nM
|
|
|
CP0471184
|
US8802673, 33
Show/Hide
|
C17H18F3N3O
|
1
|
1 |
Ki = 544.4 nM
|
|
|
CP0560268
|
US8802673, 28
Show/Hide
|
C17H21N3O2
|
1
|
1 |
Ki = 561 nM
|
|
|
CP0520279
|
US8802673, 58
Show/Hide
|
C15H15Cl2N3O
|
1
|
1 |
Ki = 584.4 nM
|
|
|
CP0553390
|
US8802673, 65
Show/Hide
|
C17H18N2O3
|
1
|
1 |
Ki = 629.1 nM
|
|
|
CP0539095
|
US8802673, 43
Show/Hide
|
C15H16FN3O
|
1
|
1 |
Ki = 648.4 nM
|
|
|
CP0539096
|
US8802673, 60
Show/Hide
|
C17H19ClN2O
|
1
|
1 |
Ki = 758.2 nM
|
|
|
CP0541878
|
US8802673, 20
Show/Hide
|
C18H22N2O2
|
1
|
1 |
Ki = 764.1 nM
|
|
|
CP0449983
|
US8802673, 27
Show/Hide
|
C16H18BrN3O
|
1
|
1 |
Ki = 808.3 nM
|
|
|
CP0424110
|
US8802673, 156
Show/Hide
|
C15H18N4O
|
1
|
1 |
Ki = 832.7 nM
|
|
|
CP0529272
|
US8802673, 153
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 839.7 nM
|
|
|
CP0491086
|
US8802673, 154
Show/Hide
|
C15H15F3N4O
|
1
|
1 |
Ki = 862.7 nM
|
|
|
CP0450194
|
US8802673, 114
Show/Hide
|
C17H22N4O
|
1
|
1 |
Ki = 995.9 nM
|
|
|
CP0442934
|
US8802673, 139
Show/Hide
|
C17H22N4O3
|
1
|
1 |
Ki = 1060.7 nM
|
|
|
CP0521212
|
US8802673, 41
Show/Hide
|
C16H16F3N3O
|
1
|
1 |
Ki = 1080.9 nM
|
|
|
CP0442959
|
US8802673, 186
Show/Hide
|
C14H14Cl2N4O
|
1
|
1 |
Ki = 1101.8 nM
|
|
|
CP0500139
|
US8802673, 37
Show/Hide
|
C16H18FN3O
|
1
|
1 |
Ki = 1173.8 nM
|
|
|
CP0471183
|
US8802673, 32
Show/Hide
|
C16H18ClN3O
|
1
|
1 |
Ki = 1237.5 nM
|
|
|
CP0509212
|
US8802673, 167
Show/Hide
|
C16H17F3N4O
|
1
|
1 |
Ki = 1353.9 nM
|
|
|
CP0442914
|
US8802673, 138
Show/Hide
|
C17H22N4O3
|
1
|
1 |
Ki = 1356.6 nM
|
|
|
CP0491095
|
US8802673, 63
Show/Hide
|
C15H15Cl2N3O
|
1
|
1 |
Ki = 1489.7 nM
|
|
|
CP0557095
|
US8802673, 1
Show/Hide
|
C16H20N4
|
1
|
1 |
Ki = 1510.8 nM
|
|
|
CP0500334
|
US8802673, 23
Show/Hide
|
C18H19N3O
|
1
|
1 |
Ki = 1644 nM
|
|
|
CP0384788
|
US8802673, 159
Show/Hide
|
C16H19N5O2
|
1
|
1 |
Ki = 1756.2 nM
|
|
|
CP0556273
|
US8802673, 158
Show/Hide
|
C16H19N5O2
|
1
|
1 |
Ki = 1854.2 nM
|
|
|
CP0503588
|
US8802673, 55
Show/Hide
|
C15H16FN3O
|
1
|
1 |
Ki = 1984.3 nM
|
|
|
CP0516774
|
US8802673, 160
Show/Hide
|
C15H18N4O
|
1
|
1 |
Ki = 2749 nM
|
|
|
CP0536241
|
US8802673, 78
Show/Hide
|
C15H18N4O3S
|
1
|
1 |
Ki = 3192.1 nM
|
|
|
CP0550084
|
US8802673, 2
Show/Hide
|
C17H17BrF3N3
|
1
|
1 |
Ki = 3514.5 nM
|
|
|
CP0500154
|
US8802673, 70
Show/Hide
|
C18H21ClN2O
|
1
|
1 |
Ki = 4066.5 nM
|
|
|
CP0509207
|
US8802673, 140
Show/Hide
|
C14H18N4O
|
1
|
1 |
Ki = 5251 nM
|
|
|
CP0384787
|
US8802673, 157
Show/Hide
|
C15H18N4O
|
1
|
1 |
Ki > 10000 nM
|
|
|
CP0443846
|
US8802673, 176
Show/Hide
|
C14H16N4O
|
1
|
1 |
Ki > 10000 nM
|
|
|