Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT06968 , Trace amine-associated receptor 7b
Gene Name TAAR7B
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID Q923X8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT06968
 
Compound ID Compound Name Compound Formula
CP0442136
US8802673, 211
   Show/Hide
C16H16ClF3N4O2
 1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0491107
US8802673, 194
   Show/Hide
C17H19ClN4O
 1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0539099
US8802673, 171
   Show/Hide
C17H19ClN4O
 1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0536190
US8802673, 170
   Show/Hide
C17H19ClN4O
 1
1
Ki = 1.2 nM
   TI
   LI
   LO
   TS
CP0384786
US8802673, 149
   Show/Hide
C17H19ClN4O
 1
1
Ki = 1.4 nM
   TI
   LI
   LO
   TS
CP0520648
US8802673, 203
   Show/Hide
C16H16ClF3N4O2
 1
1
Ki = 1.7 nM
   TI
   LI
   LO
   TS
CP0491106
US8802673, 184
   Show/Hide
C16H16ClF3N4O2
 1
1
Ki = 2 nM
   TI
   LI
   LO
   TS
CP0491109
US8802673, 204
   Show/Hide
C15H14ClF3N4O
 1
1
Ki = 2.1 nM
   TI
   LI
   LO
   TS
CP0442942
US8802673, 209
   Show/Hide
C16H15F5N4O2
 1
1
Ki = 2.5 nM
   TI
   LI
   LO
   TS
CP0484454
US8802673, 137
   Show/Hide
C16H17F3N4O2
 1
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
CP0521300
US8802673, 192
   Show/Hide
C17H19FN4O
 1
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
CP0528997
US8802673, 118
   Show/Hide
C17H19FN4O
 1
1
Ki = 3 nM
   TI
   LI
   LO
   TS
CP0516796
US8802673, 188
   Show/Hide
C16H16F4N4O2
 1
1
Ki = 3.3 nM
   TI
   LI
   LO
   TS
CP0520283
US8802673, 98
   Show/Hide
C17H19FN4O
 1
1
Ki = 3.3 nM
   TI
   LI
   LO
   TS
CP0539102
US8802673, 208
   Show/Hide
C16H16F4N4O2
 1
1
Ki = 3.5 nM
   TI
   LI
   LO
   TS
CP0503591
US8802673, 128
   Show/Hide
C17H21FN4O
 1
1
Ki = 3.9 nM
   TI
   LI
   LO
   TS
CP0539101
US8802673, 196
   Show/Hide
C15H14F4N4O
 1
1
Ki = 4 nM
   TI
   LI
   LO
   TS
CP0535952
US8802673, 101
   Show/Hide
C17H21FN4O
 1
1
Ki = 4.1 nM
   TI
   LI
   LO
   TS
CP0491093
US8802673, 53
   Show/Hide
C19H18BrN3O
 1
1
Ki = 4.5 nM
   TI
   LI
   LO
   TS
CP0503700
US8802673, 144
   Show/Hide
C16H16F4N4O2
 1
1
Ki = 4.9 nM
   TI
   LI
   LO
   TS
CP0500141
US8802673, 119
   Show/Hide
C17H19FN4O
 1
1
Ki = 5.1 nM
   TI
   LI
   LO
   TS
CP0499823
US8802673, 97
   Show/Hide
C16H19FN4O
 1
1
Ki = 5.6 nM
   TI
   LI
   LO
   TS
CP0531765
US8802673, 202
   Show/Hide
C14H14Cl2N4O
 1
1
Ki = 6.5 nM
   TI
   LI
   LO
   TS
CP0491105
US8802673, 175
   Show/Hide
C19H17ClF2N6O3
 1
1
Ki = 6.6 nM
   TI
   LI
   LO
   TS
CP0503586
US8802673, 47
   Show/Hide
C19H18ClN3O
 1
1
Ki = 6.7 nM
   TI
   LI
   LO
   TS
CP0529249
US8802673, 145
   Show/Hide
C16H16F4N4O2
 1
1
Ki = 6.7 nM
   TI
   LI
   LO
   TS
CP0471189
US8802673, 129
   Show/Hide
C17H21FN4O
 1
1
Ki = 6.8 nM
   TI
   LI
   LO
   TS
CP0535954
US8802673, 116
   Show/Hide
C16H19FN4O
 1
1
Ki = 7 nM
   TI
   LI
   LO
   TS
CP0520660
US8802673, 134
   Show/Hide
C15H14F4N4O
 1
1
Ki = 7.9 nM
   TI
   LI
   LO
   TS
CP0509209
US8802673, 148
   Show/Hide
C18H18N4O2
 1
1
Ki = 8.3 nM
   TI
   LI
   LO
   TS
CP0519047
US8802673, 26
   Show/Hide
C17H16ClN3OS
 1
1
Ki = 8.3 nM
   TI
   LI
   LO
   TS
CP0555392
US8802673, 52
   Show/Hide
C19H18ClN3O
 1
1
Ki = 8.4 nM
   TI
   LI
   LO
   TS
CP0491098
US8802673, 86
   Show/Hide
C17H20N4O
 1
1
Ki = 9 nM
   TI
   LI
   LO
   TS
CP0491094
US8802673, 62
   Show/Hide
C16H18BrN3O
 1
1
Ki = 9.4 nM
   TI
   LI
   LO
   TS
CP0450195
US8802673, 121
   Show/Hide
C15H14F4N4O
 1
1
Ki = 9.6 nM
   TI
   LI
   LO
   TS
CP0450198
US8802673, 126
   Show/Hide
C14H14BrFN4O
 1
1
Ki = 9.6 nM
   TI
   LI
   LO
   TS
CP0520647
US8802673, 187
   Show/Hide
C16H17F3N4O2
 1
1
Ki = 10 nM
   TI
   LI
   LO
   TS
CP0491096
US8802673, 82
   Show/Hide
C16H15ClF3N3O
 1
1
Ki = 10.1 nM
   TI
   LI
   LO
   TS
CP0484467
US8802673, 207
   Show/Hide
C16H16F4N4O2
 1
1
Ki = 10.2 nM
   TI
   LI
   LO
   TS
CP0471188
US8802673, 117
   Show/Hide
C16H19FN4O
 1
1
Ki = 10.4 nM
   TI
   LI
   LO
   TS
CP0500335
US8802673, 44
   Show/Hide
C20H20N2O
 1
1
Ki = 11.8 nM
   TI
   LI
   LO
   TS
CP0512149
US8802673, 102
   Show/Hide
C14H14BrFN4O
 1
1
Ki = 12.6 nM
   TI
   LI
   LO
   TS
CP0384785
US8802673, 141
   Show/Hide
C22H24N4O3
 1
1
Ki = 12.9 nM
   TI
   LI
   LO
   TS
CP0553826
US8802673, 17
   Show/Hide
C17H20N4O
 1
1
Ki = 13.1 nM
   TI
   LI
   LO
   TS
CP0519048
US8802673, 54
   Show/Hide
C19H18ClN3O
 1
1
Ki = 13.8 nM
   TI
   LI
   LO
   TS
CP0509208
US8802673, 142
   Show/Hide
C22H24N4O3
 1
1
Ki = 14.6 nM
   TI
   LI
   LO
   TS
CP0551298
US8802673, 172
   Show/Hide
C16H17F3N4O2
 1
1
Ki = 16.2 nM
   TI
   LI
   LO
   TS
CP0520659
US8802673, 100
   Show/Hide
C16H19FN4O2
 1
1
Ki = 16.4 nM
   TI
   LI
   LO
   TS
CP0503699
US8802673, 127
   Show/Hide
C14H14BrFN4O
 1
1
Ki = 16.5 nM
   TI
   LI
   LO
   TS
CP0442874
US8802673, 34
   Show/Hide
C18H21ClN2O
 1
1
Ki = 18.1 nM
   TI
   LI
   LO
   TS
CP0512152
US8802673, 132
   Show/Hide
C16H19FN4O2
 1
1
Ki = 18.2 nM
   TI
   LI
   LO
   TS
CP0490531
US8802673, 99
   Show/Hide
C15H15ClFN3O
 1
1
Ki = 18.5 nM
   TI
   LI
   LO
   TS
CP0491097
US8802673, 85
   Show/Hide
C17H20BrN3O
 1
1
Ki = 19.4 nM
   TI
   LI
   LO
   TS
CP0524425
US8802673, 193
   Show/Hide
C17H19ClN4O
 1
1
Ki = 19.6 nM
   TI
   LI
   LO
   TS
CP0524421
US8802673, 147
   Show/Hide
C18H18N4O2
 1
1
Ki = 19.7 nM
   TI
   LI
   LO
   TS
CP0503593
US8802673, 135
   Show/Hide
C15H14F4N4O
 1
1
Ki = 19.8 nM
   TI
   LI
   LO
   TS
CP0471190
US8802673, 130
   Show/Hide
C14H14ClFN4O
 1
1
Ki = 19.9 nM
   TI
   LI
   LO
   TS
CP0529271
US8802673, 96
   Show/Hide
C14H14ClFN4O
 1
1
Ki = 21.6 nM
   TI
   LI
   LO
   TS
CP0520281
US8802673, 83
   Show/Hide
C16H18ClN3O
 1
1
Ki = 22.2 nM
   TI
   LI
   LO
   TS
CP0520282
US8802673, 93
   Show/Hide
C17H22N4O
 1
1
Ki = 22.2 nM
   TI
   LI
   LO
   TS
CP0536243
US8802673, 95
   Show/Hide
C15H15F3N4O
 1
1
Ki = 22.3 nM
   TI
   LI
   LO
   TS
CP0443849
US8802673, 11
   Show/Hide
C16H16F3N3O
 1
1
Ki = 23.3 nM
   TI
   LI
   LO
   TS
CP0530404
US8802673, 19
   Show/Hide
C15H15F3N4O
 1
1
Ki = 23.6 nM
   TI
   LI
   LO
   TS
CP0541879
US8802673, 21
   Show/Hide
C17H22N4O
 1
1
Ki = 24.5 nM
   TI
   LI
   LO
   TS
CP0491088
US8802673, 164
   Show/Hide
C19H20N4O
 1
1
Ki = 25 nM
   TI
   LI
   LO
   TS
CP0450191
US8802673, 3
   Show/Hide
C20H22ClF3N2
 1
1
Ki = 25.1 nM
   TI
   LI
   LO
   TS
CP0500138
US8802673, 195
   Show/Hide
C17H19FN4O
 1
1
Ki = 25.2 nM
   TI
   LI
   LO
   TS
CP0553831
US8802673, 210
   Show/Hide
C14H14ClFN4O
 1
1
Ki = 26.6 nM
   TI
   LI
   LO
   TS
CP0450197
US8802673, 125
   Show/Hide
C18H22N4O2
 1
1
Ki = 27.8 nM
   TI
   LI
   LO
   TS
CP0520649
US8802673, 5
   Show/Hide
C15H16ClN3O
 1
1
Ki = 29 nM
   TI
   LI
   LO
   TS
CP0520658
US8802673, 74
   Show/Hide
C18H22N4O
 1
1
Ki = 29.5 nM
   TI
   LI
   LO
   TS
CP0503715
US8802673, 178
   Show/Hide
C16H17F3N4O
 1
1
Ki = 29.8 nM
   TI
   LI
   LO
   TS
CP0442958
US8802673, 177
   Show/Hide
C18H18N4O
 1
1
Ki = 29.9 nM
   TI
   LI
   LO
   TS
CP0539097
US8802673, 110
   Show/Hide
C18H22N4O
 1
1
Ki = 30.6 nM
   TI
   LI
   LO
   TS
CP0491108
US8802673, 197
   Show/Hide
C15H14F4N4O
 1
1
Ki = 31.5 nM
   TI
   LI
   LO
   TS
CP0535953
US8802673, 111
   Show/Hide
C18H22N4O
 1
1
Ki = 32.2 nM
   TI
   LI
   LO
   TS
CP0519044
US8802673, 8
   Show/Hide
C16H17ClN2O
 1
1
Ki = 32.5 nM
   TI
   LI
   LO
   TS
CP0520661
US8802673, 180
   Show/Hide
C15H17ClN4O2
 1
1
Ki = 33 nM
   TI
   LI
   LO
   TS
CP0524404
US8802673, 163
   Show/Hide
C19H20N4O
 1
1
Ki = 33.2 nM
   TI
   LI
   LO
   TS
CP0519045
US8802673, 10
   Show/Hide
C15H16BrN3O
 1
1
Ki = 33.7 nM
   TI
   LI
   LO
   TS
CP0450196
US8802673, 124
   Show/Hide
C18H22N4O2
 1
1
Ki = 34.8 nM
   TI
   LI
   LO
   TS
CP0443856
US8802673, 73
   Show/Hide
C18H24N4O
 1
1
Ki = 35 nM
   TI
   LI
   LO
   TS
CP0442897
US8802673, 120
   Show/Hide
C15H17BrN4O
 1
1
Ki = 36.4 nM
   TI
   LI
   LO
   TS
CP0536242
US8802673, 87
   Show/Hide
C18H22N4O
 1
1
Ki = 37 nM
   TI
   LI
   LO
   TS
CP0531662
US8802673, 131
   Show/Hide
C14H14ClFN4O
 1
1
Ki = 37.9 nM
   TI
   LI
   LO
   TS
CP0535955
US8802673, 133
   Show/Hide
C16H19FN4O2
 1
1
Ki = 38.7 nM
   TI
   LI
   LO
   TS
CP0442130
US8802673, 30
   Show/Hide
C17H18Cl2N2O
 1
1
Ki = 41.7 nM
   TI
   LI
   LO
   TS
CP0442134
US8802673, 190
   Show/Hide
C17H19FN4O
 1
1
Ki = 42.2 nM
   TI
   LI
   LO
   TS
CP0555390
US8802673, 7
   Show/Hide
C14H15BrN4O
 1
1
Ki = 42.5 nM
   TI
   LI
   LO
   TS
CP0449984
US8802673, 69
   Show/Hide
C15H16ClN3O
 1
1
Ki = 43.8 nM
   TI
   LI
   LO
   TS
CP0550088
US8802673, 76
   Show/Hide
C16H18BrN3O
 1
1
Ki = 45 nM
   TI
   LI
   LO
   TS
CP0450192
US8802673, 15
   Show/Hide
C16H20N4O
 1
1
Ki = 46.6 nM
   TI
   LI
   LO
   TS
CP0484453
US8802673, 94
   Show/Hide
C14H15BrN4O
 1
1
Ki = 48.9 nM
   TI
   LI
   LO
   TS
CP0528999
US8802673, 136
   Show/Hide
C16H17F3N4O2
 1
1
Ki = 49.4 nM
   TI
   LI
   LO
   TS
CP0442896
US8802673, 103
   Show/Hide
C14H15ClN4O
 1
1
Ki = 50 nM
   TI
   LI
   LO
   TS
CP0539100
US8802673, 179
   Show/Hide
C15H16F2N4O2
 1
1
Ki = 51.7 nM
   TI
   LI
   LO
   TS
CP0442891
US8802673, 42
   Show/Hide
C16H16F3N3O
 1
1
Ki = 51.8 nM
   TI
   LI
   LO
   TS
CP0442876
US8802673, 38
   Show/Hide
C15H16ClN3O
 1
1
Ki = 54.4 nM
   TI
   LI
   LO
   TS
CP0550485
US8802673, 199
   Show/Hide
C14H15ClN4O
 1
1
Ki = 56 nM
   TI
   LI
   LO
   TS
CP0519050
US8802673, 84
   Show/Hide
C17H20ClN3O
 1
1
Ki = 57 nM
   TI
   LI
   LO
   TS
CP0520662
US8802673, 200
   Show/Hide
C15H15F3N4O
 1
1
Ki = 58.8 nM
   TI
   LI
   LO
   TS
CP0500144
US8802673, 189
   Show/Hide
C17H20N4O
 1
1
Ki = 60.5 nM
   TI
   LI
   LO
   TS
CP0503587
US8802673, 50
   Show/Hide
C18H17ClN4O
 1
1
Ki = 60.8 nM
   TI
   LI
   LO
   TS
CP0516775
US8802673, 173
   Show/Hide
C15H15F3N4O
 1
1
Ki = 62.5 nM
   TI
   LI
   LO
   TS
CP0442895
US8802673, 80
   Show/Hide
C16H18ClN3O
 1
1
Ki = 62.6 nM
   TI
   LI
   LO
   TS
CP0442941
US8802673, 201
   Show/Hide
C15H15F3N4O
 1
1
Ki = 62.6 nM
   TI
   LI
   LO
   TS
CP0500143
US8802673, 174
   Show/Hide
C19H18F2N6O3
 1
1
Ki = 62.8 nM
   TI
   LI
   LO
   TS
CP0524416
US8802673, 46
   Show/Hide
C19H19N3O
 1
1
Ki = 64.3 nM
   TI
   LI
   LO
   TS
CP0486058
US8802673, 25
   Show/Hide
C18H19F3N2O2
 1
1
Ki = 70.5 nM
   TI
   LI
   LO
   TS
CP0520280
US8802673, 79
   Show/Hide
C17H19ClN2O
 1
1
Ki = 71.6 nM
   TI
   LI
   LO
   TS
CP0443853
US8802673, 68
   Show/Hide
C16H20N4O
 1
1
Ki = 75.1 nM
   TI
   LI
   LO
   TS
CP0516778
US8802673, 4
   Show/Hide
C21H24ClF3N2
 1
1
Ki = 78.5 nM
   TI
   LI
   LO
   TS
CP0503698
US8802673, 123
   Show/Hide
C17H22N4O2
 1
1
Ki = 79.6 nM
   TI
   LI
   LO
   TS
CP0536244
US8802673, 106
   Show/Hide
C17H22N4O
 1
1
Ki = 81.4 nM
   TI
   LI
   LO
   TS
CP0536245
US8802673, 122
   Show/Hide
C17H22N4O2
 1
1
Ki = 84.7 nM
   TI
   LI
   LO
   TS
CP0503589
US8802673, 57
   Show/Hide
C15H15BrFN3O
 1
1
Ki = 86.6 nM
   TI
   LI
   LO
   TS
CP0530622
US8802673, 88
   Show/Hide
C17H22N4O
 1
1
Ki = 87.4 nM
   TI
   LI
   LO
   TS
CP0490532
US8802673, 113
   Show/Hide
C19H20N4O
 1
1
Ki = 87.7 nM
   TI
   LI
   LO
   TS
CP0499824
US8802673, 107
   Show/Hide
C17H22N4O
 1
1
Ki = 87.7 nM
   TI
   LI
   LO
   TS
CP0426462
US8802673, 185
   Show/Hide
C16H15ClF3N3O
 1
1
Ki = 88.8 nM
   TI
   LI
   LO
   TS
CP0516779
US8802673, 9
   Show/Hide
C17H19ClN2O
 1
1
Ki = 89.3 nM
   TI
   LI
   LO
   TS
CP0553829
US8802673, 151
   Show/Hide
C17H21FN4O3
 1
1
Ki = 95.4 nM
   TI
   LI
   LO
   TS
CP0524443
US8802673, 206
   Show/Hide
C14H15ClN4O
 1
1
Ki = 96.3 nM
   TI
   LI
   LO
   TS
CP0521217
US8802673, 64
   Show/Hide
C16H18BrN3O
 1
1
Ki = 101 nM
   TI
   LI
   LO
   TS
CP0550263
US8802673, 49
   Show/Hide
C21H17F6N3O
 1
1
Ki = 103.8 nM
   TI
   LI
   LO
   TS
CP0512150
US8802673, 104
   Show/Hide
C14H15ClN4O
 1
1
Ki = 104.8 nM
   TI
   LI
   LO
   TS
CP0530402
US8802673, 13
   Show/Hide
C18H22N2O
 1
1
Ki = 108.5 nM
   TI
   LI
   LO
   TS
CP0499822
US8802673, 91
   Show/Hide
C14H15BrN4O
 1
1
Ki = 123.3 nM
   TI
   LI
   LO
   TS
CP0500336
US8802673, 45
   Show/Hide
C17H19BrN2O
 1
1
Ki = 126.1 nM
   TI
   LI
   LO
   TS
CP0449985
US8802673, 105
   Show/Hide
C16H20N4O2
 1
1
Ki = 126.5 nM
   TI
   LI
   LO
   TS
CP0384789
US8802673, 162
   Show/Hide
C20H22N4O
 1
1
Ki = 127.3 nM
   TI
   LI
   LO
   TS
CP0550264
US8802673, 77
   Show/Hide
C15H15ClFN3O
 1
1
Ki = 130.4 nM
   TI
   LI
   LO
   TS
CP0539098
US8802673, 146
   Show/Hide
C17H22N4O
 1
1
Ki = 140.4 nM
   TI
   LI
   LO
   TS
CP0536246
US8802673, 150
   Show/Hide
C15H18F2N4O
 1
1
Ki = 148.6 nM
   TI
   LI
   LO
   TS
CP0519046
US8802673, 24
   Show/Hide
C18H19F3N2O
 1
1
Ki = 149 nM
   TI
   LI
   LO
   TS
CP0530405
US8802673, 29
   Show/Hide
C16H20N4O2
 1
1
Ki = 155.5 nM
   TI
   LI
   LO
   TS
CP0491104
US8802673, 166
   Show/Hide
C16H17F3N4O
 1
1
Ki = 158.9 nM
   TI
   LI
   LO
   TS
CP0442135
US8802673, 205
   Show/Hide
C14H15ClN4O
 1
1
Ki = 162.1 nM
   TI
   LI
   LO
   TS
CP0553830
US8802673, 198
   Show/Hide
C15H15F3N4O
 1
1
Ki = 162.8 nM
   TI
   LI
   LO
   TS
CP0539094
US8802673, 36
   Show/Hide
C19H24N2O
 1
1
Ki = 163.3 nM
   TI
   LI
   LO
   TS
CP0443855
US8802673, 71
   Show/Hide
C17H20ClN3O2
 1
1
Ki = 168 nM
   TI
   LI
   LO
   TS
CP0491091
US8802673, 183
   Show/Hide
C16H20N4O3
 1
1
Ki = 173.7 nM
   TI
   LI
   LO
   TS
CP0512148
US8802673, 89
   Show/Hide
C15H17BrN4O
 1
1
Ki = 176.7 nM
   TI
   LI
   LO
   TS
CP0442132
US8802673, 40
   Show/Hide
C15H15ClFN3O
 1
1
Ki = 188.2 nM
   TI
   LI
   LO
   TS
CP0550087
US8802673, 35
   Show/Hide
C17H18ClFN2O
 1
1
Ki = 188.3 nM
   TI
   LI
   LO
   TS
CP0503590
US8802673, 112
   Show/Hide
C17H22N4
 1
1
Ki = 196.6 nM
   TI
   LI
   LO
   TS
CP0550089
US8802673, 81
   Show/Hide
C15H17ClN4O
 1
1
Ki = 202.7 nM
   TI
   LI
   LO
   TS
CP0500140
US8802673, 59
   Show/Hide
C16H16ClFN2O
 1
1
Ki = 207.3 nM
   TI
   LI
   LO
   TS
CP0519049
US8802673, 56
   Show/Hide
C16H18BrN3O
 1
1
Ki = 211 nM
   TI
   LI
   LO
   TS
CP0470194
US8802673, 108
   Show/Hide
C14H15BrN4O
 1
1
Ki = 215.7 nM
   TI
   LI
   LO
   TS
CP0530406
US8802673, 72
   Show/Hide
C17H22N4O
 1
1
Ki = 220 nM
   TI
   LI
   LO
   TS
CP0553827
US8802673, 31
   Show/Hide
C17H19FN2O
 1
1
Ki = 222.2 nM
   TI
   LI
   LO
   TS
CP0400449
US8802673, 161
   Show/Hide
C20H22N4O
 1
1
Ki = 222.9 nM
   TI
   LI
   LO
   TS
CP0530407
US8802673, 75
   Show/Hide
C14H15N5O3
 1
1
Ki = 228 nM
   TI
   LI
   LO
   TS
CP0442943
US8802673, 6
   Show/Hide
C14H15ClN4O
 1
1
Ki = 232.2 nM
   TI
   LI
   LO
   TS
CP0491099
US8802673, 90
   Show/Hide
C14H15ClN4O
 1
1
Ki = 232.4 nM
   TI
   LI
   LO
   TS
CP0553828
US8802673, 48
   Show/Hide
C20H21N3O
 1
1
Ki = 233.6 nM
   TI
   LI
   LO
   TS
CP0530408
US8802673, 115
   Show/Hide
C18H18N4O2
 1
1
Ki = 234.9 nM
   TI
   LI
   LO
   TS
CP0566202
US8802673, 39
   Show/Hide
C16H19N3O2
 1
1
Ki = 251.4 nM
   TI
   LI
   LO
   TS
CP0521218
US8802673, 66
   Show/Hide
C19H18BrN3O
 1
1
Ki = 256.9 nM
   TI
   LI
   LO
   TS
CP0443850
US8802673, 12
   Show/Hide
C15H18N4O2
 1
1
Ki = 258.8 nM
   TI
   LI
   LO
   TS
CP0424108
US8802673, 152
   Show/Hide
C17H21FN4O3
 1
1
Ki = 267.7 nM
   TI
   LI
   LO
   TS
CP0490530
US8802673, 92
   Show/Hide
C16H19N5O
 1
1
Ki = 274.8 nM
   TI
   LI
   LO
   TS
CP0491092
US8802673, 51
   Show/Hide
C20H20ClN3O
 1
1
Ki = 280.3 nM
   TI
   LI
   LO
   TS
CP0491103
US8802673, 143
   Show/Hide
C14H17BrN4O
 1
1
Ki = 283.6 nM
   TI
   LI
   LO
   TS
CP0490529
US8802673, 67
   Show/Hide
C15H16ClN3O
 1
1
Ki = 291.7 nM
   TI
   LI
   LO
   TS
CP0521211
US8802673, 18
   Show/Hide
C15H18N4O
 1
1
Ki = 313.3 nM
   TI
   LI
   LO
   TS
CP0509210
US8802673, 165
   Show/Hide
C18H21N3O2
 1
1
Ki = 339.5 nM
   TI
   LI
   LO
   TS
CP0512151
US8802673, 109
   Show/Hide
C14H15BrN4O
 1
1
Ki = 362.4 nM
   TI
   LI
   LO
   TS
CP0491090
US8802673, 181
   Show/Hide
C15H15N5O
 1
1
Ki = 398.1 nM
   TI
   LI
   LO
   TS
CP0529250
US8802673, 182
   Show/Hide
C16H20N4O
 1
1
Ki = 446.5 nM
   TI
   LI
   LO
   TS
CP0521210
US8802673, 16
   Show/Hide
C15H15N5O
 1
1
Ki = 448.3 nM
   TI
   LI
   LO
   TS
CP0539093
US8802673, 22
   Show/Hide
C18H22N2O
 1
1
Ki = 468 nM
   TI
   LI
   LO
   TS
CP0450193
US8802673, 61
   Show/Hide
C15H15Br2N3O
 1
1
Ki = 502.4 nM
   TI
   LI
   LO
   TS
CP0530403
US8802673, 14
   Show/Hide
C14H15FN4O
 1
1
Ki = 504 nM
   TI
   LI
   LO
   TS
CP0471184
US8802673, 33
   Show/Hide
C17H18F3N3O
 1
1
Ki = 544.4 nM
   TI
   LI
   LO
   TS
CP0560268
US8802673, 28
   Show/Hide
C17H21N3O2
 1
1
Ki = 561 nM
   TI
   LI
   LO
   TS
CP0520279
US8802673, 58
   Show/Hide
C15H15Cl2N3O
 1
1
Ki = 584.4 nM
   TI
   LI
   LO
   TS
CP0553390
US8802673, 65
   Show/Hide
C17H18N2O3
 1
1
Ki = 629.1 nM
   TI
   LI
   LO
   TS
CP0539095
US8802673, 43
   Show/Hide
C15H16FN3O
 1
1
Ki = 648.4 nM
   TI
   LI
   LO
   TS
CP0539096
US8802673, 60
   Show/Hide
C17H19ClN2O
 1
1
Ki = 758.2 nM
   TI
   LI
   LO
   TS
CP0541878
US8802673, 20
   Show/Hide
C18H22N2O2
 1
1
Ki = 764.1 nM
   TI
   LI
   LO
   TS
CP0449983
US8802673, 27
   Show/Hide
C16H18BrN3O
 1
1
Ki = 808.3 nM
   TI
   LI
   LO
   TS
CP0424110
US8802673, 156
   Show/Hide
C15H18N4O
 1
1
Ki = 832.7 nM
   TI
   LI
   LO
   TS
CP0529272
US8802673, 153
   Show/Hide
C15H15F3N4O
 1
1
Ki = 839.7 nM
   TI
   LI
   LO
   TS
CP0491086
US8802673, 154
   Show/Hide
C15H15F3N4O
 1
1
Ki = 862.7 nM
   TI
   LI
   LO
   TS
CP0450194
US8802673, 114
   Show/Hide
C17H22N4O
 1
1
Ki = 995.9 nM
   TI
   LI
   LO
   TS
CP0442934
US8802673, 139
   Show/Hide
C17H22N4O3
 1
1
Ki = 1060.7 nM
   TI
   LI
   LO
   TS
CP0521212
US8802673, 41
   Show/Hide
C16H16F3N3O
 1
1
Ki = 1080.9 nM
   TI
   LI
   LO
   TS
CP0442959
US8802673, 186
   Show/Hide
C14H14Cl2N4O
 1
1
Ki = 1101.8 nM
   TI
   LI
   LO
   TS
CP0500139
US8802673, 37
   Show/Hide
C16H18FN3O
 1
1
Ki = 1173.8 nM
   TI
   LI
   LO
   TS
CP0471183
US8802673, 32
   Show/Hide
C16H18ClN3O
 1
1
Ki = 1237.5 nM
   TI
   LI
   LO
   TS
CP0509212
US8802673, 167
   Show/Hide
C16H17F3N4O
 1
1
Ki = 1353.9 nM
   TI
   LI
   LO
   TS
CP0442914
US8802673, 138
   Show/Hide
C17H22N4O3
 1
1
Ki = 1356.6 nM
   TI
   LI
   LO
   TS
CP0491095
US8802673, 63
   Show/Hide
C15H15Cl2N3O
 1
1
Ki = 1489.7 nM
   TI
   LI
   LO
   TS
CP0557095
US8802673, 1
   Show/Hide
C16H20N4
 1
1
Ki = 1510.8 nM
   TI
   LI
   LO
   TS
CP0500334
US8802673, 23
   Show/Hide
C18H19N3O
 1
1
Ki = 1644 nM
   TI
   LI
   LO
   TS
CP0384788
US8802673, 159
   Show/Hide
C16H19N5O2
 1
1
Ki = 1756.2 nM
   TI
   LI
   LO
   TS
CP0556273
US8802673, 158
   Show/Hide
C16H19N5O2
 1
1
Ki = 1854.2 nM
   TI
   LI
   LO
   TS
CP0503588
US8802673, 55
   Show/Hide
C15H16FN3O
 1
1
Ki = 1984.3 nM
   TI
   LI
   LO
   TS
CP0516774
US8802673, 160
   Show/Hide
C15H18N4O
 1
1
Ki = 2749 nM
   TI
   LI
   LO
   TS
CP0536241
US8802673, 78
   Show/Hide
C15H18N4O3S
 1
1
Ki = 3192.1 nM
   TI
   LI
   LO
   TS
CP0550084
US8802673, 2
   Show/Hide
C17H17BrF3N3
 1
1
Ki = 3514.5 nM
   TI
   LI
   LO
   TS
CP0500154
US8802673, 70
   Show/Hide
C18H21ClN2O
 1
1
Ki = 4066.5 nM
   TI
   LI
   LO
   TS
CP0509207
US8802673, 140
   Show/Hide
C14H18N4O
 1
1
Ki = 5251 nM
   TI
   LI
   LO
   TS
CP0384787
US8802673, 157
   Show/Hide
C15H18N4O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS
CP0443846
US8802673, 176
   Show/Hide
C14H16N4O
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS