| Compound ID |
Compound Name |
Compound Formula |
|
CP0644312
|
cis-2,6-Dimethyl-4-(6-(5-(1-methylcyclopropoxy)-1H-indazol-3-yl)pyrimidin-4-yl)morpholine
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|
C21H25N5O2
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0572948
|
3-[2-ethyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
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|
C23H22N4O2S
|
2
|
| 1 |
EC50 = 260 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0545474
|
3-[2-cyclopropyl-4-[5-methyl-3-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
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|
C25H24N4O2S
|
2
|
| 1 |
EC50 = 280 nM
|
|
|
| 2 |
EC50 = 5400 nM
|
|
|
|
CP0543342
|
3-[4-[5-methyl-3-(2-morpholin-4-ylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
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|
C25H25N5O3S
|
2
|
| 1 |
EC50 = 290 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0545472
|
3-[4-[5-(2-morpholin-4-ylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
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|
C24H23N5O3S
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0540375
|
3-[2-cyclopropyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
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|
C24H22N4O2S
|
2
|
| 1 |
EC50 = 390 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0548058
|
3-[2,6-difluoro-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
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|
C21H16F2N4O2S
|
1
|
| 1 |
EC50 = 390 nM
|
|
|
|
CP0578500
|
3-[2-ethyl-4-(5-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
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|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0579366
|
3-[2-methyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0577947
|
3-[2-fluoro-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
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|
C21H17FN4O2S
|
1
|
| 1 |
EC50 = 690 nM
|
|
|
|
CP0579422
|
3-[4-[3-(2-methoxypyridin-4-yl)-5-methyl-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
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|
C22H20N4O3S
|
1
|
| 1 |
EC50 = 750 nM
|
|
|
|
CP0574644
|
3-[4-[3-(2,6-dimethylpyridin-4-yl)-5-methyl-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C23H22N4O2S
|
1
|
| 1 |
EC50 = 760 nM
|
|
|
|
CP0545471
|
2,3-dimethyl-4-[4-[5-methyl-3-(2-morpholin-4-ylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
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|
C27H29N5O3S
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0575926
|
3-[4-[5-(2,6-dimethylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 920 nM
|
|
|
|
CP0576280
|
3-[4-[5-methyl-3-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 1080 nM
|
|
|
|
CP0554483
|
3-[2-methoxy-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O3S
|
1
|
| 1 |
EC50 = 1280 nM
|
|
|
|
CP0579421
|
3-[4-[5-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C21H18N4O2S
|
1
|
| 1 |
EC50 = 1380 nM
|
|
|
|
CP0575928
|
3-[2,6-dimethyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C23H22N4O2S
|
1
|
| 1 |
EC50 = 1440 nM
|
|
|
|
CP0579357
|
2,3-dimethyl-4-[4-[5-(2-morpholin-4-ylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
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|
C26H27N5O3S
|
2
|
| 1 |
EC50 = 1500 nM
|
|
|
| 2 |
EC50 = 76000 nM
|
|
|
|
CP0579473
|
3-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)-2-propan-2-ylphenyl]benzenesulfonamide
Show/Hide
|
C24H24N4O2S
|
1
|
| 1 |
EC50 = 1710 nM
|
|
|
|
CP0578781
|
3-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C21H18N4O2S
|
2
|
| 1 |
EC50 = 2100 nM
|
|
|
| 2 |
EC50 > 100000 nM
|
|
|
|
CP0579358
|
3-[4-[5-(2-methoxypyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C21H18N4O3S
|
1
|
| 1 |
EC50 = 2310 nM
|
|
|
|
CP0577021
|
3-[2,3-difluoro-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C21H16F2N4O2S
|
1
|
| 1 |
EC50 = 3120 nM
|
|
|
|
CP0570308
|
4-methyl-3-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
|
CP0572949
|
3-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)-2-(trifluoromethyl)phenyl]benzenesulfonamide
Show/Hide
|
C22H17F3N4O2S
|
1
|
| 1 |
EC50 = 4780 nM
|
|
|
|
CP0579994
|
4-[5-methyl-4-[3-methyl-4-(3-methylsulfonylphenyl)phenyl]-1H-pyrazol-3-yl]pyridine
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|
C23H21N3O2S
|
1
|
| 1 |
EC50 = 4900 nM
|
|
|
|
CP0572967
|
3-[4-(5-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C20H16N4O2S
|
1
|
| 1 |
EC50 = 5100 nM
|
|
|
|
CP0544064
|
2-methyl-3-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 6400 nM
|
|
|
|
CP0577215
|
3-[4-(5-phenyl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C21H17N3O2S
|
1
|
| 1 |
EC50 = 12200 nM
|
|
|
|
CP0580094
|
4-methyl-3-[4-(5-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C21H18N4O2S
|
1
|
| 1 |
EC50 = 12200 nM
|
|
|
|
CP0545473
|
3-[3-methyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 13400 nM
|
|
|
|
CP0548056
|
4-[2-ethyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C23H22N4O2S
|
1
|
| 1 |
EC50 = 14300 nM
|
|
|
|
CP0577255
|
4-[4-[3-(2,6-dimethylpyridin-4-yl)-5-methyl-1H-pyrazol-4-yl]phenyl]-2,3-dimethylbenzenesulfonamide
Show/Hide
|
C25H26N4O2S
|
1
|
| 1 |
EC50 = 15000 nM
|
|
|
|
CP0575925
|
3-[4-[3-pyridin-4-yl-5-(trifluoromethyl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C21H15F3N4O2S
|
1
|
| 1 |
EC50 = 16700 nM
|
|
|
|
CP0579367
|
3-[2-cyano-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H17N5O2S
|
1
|
| 1 |
EC50 = 19600 nM
|
|
|
|
CP0577020
|
3-[2-methyl-4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzamide
Show/Hide
|
C23H20N4O
|
1
|
| 1 |
EC50 = 21700 nM
|
|
|
|
CP0579356
|
2,3-dimethyl-4-[4-[5-methyl-3-(2-methylpyridin-4-yl)-1H-pyrazol-4-yl]phenyl]benzenesulfonamide
Show/Hide
|
C24H24N4O2S
|
1
|
| 1 |
EC50 = 57000 nM
|
|
|
|
CP0579420
|
2,3-dimethyl-4-[4-(5-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 80000 nM
|
|
|
|
CP0577216
|
3,4-dimethyl-5-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C23H22N4O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0579355
|
2,3-dimethyl-4-[4-(5-methyl-3-pyridin-4-yl-1H-pyrazol-4-yl)phenyl]benzenesulfonamide
Show/Hide
|
C23H22N4O2S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
