| Compound ID |
Compound Name |
Compound Formula |
|
CP0533812
|
3-{5-[(5- chloropyridin-2- yl)methyl]-1,3,4- oxadiazol-2-yl}-5- (2,6- dimethoxyphenyl)- 6-(ethoxymethyl) pyridine-2,4-diol
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|
C24H23ClN4O6
|
1
|
| 1 |
EC50 = 0.024 nM
|
|
|
|
CP0235875
|
(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-1-[2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-oxopyrrolidine-2-carbonyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]hexanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoic acid
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|
C69H108N22O16S
|
2
|
| 1 |
EC50 = 0.06 nM
|
|
|
| 2 |
EC50 = 0.062 nM
|
|
|
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CP0466444
|
2-[2-chloro-6-(6-methoxy-1H-benzimidazol-2-yl)phenyl]-5-[[(1R)-1-phenylbutyl]carbamoyl]benzoic acid
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|
C32H28ClN3O4
|
1
|
| 1 |
EC50 = 0.12 nM
|
|
|
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CP0514614
|
3-{5-[(4- chlorophenyl) methyl]-1,3,4- oxadiazol- 2-yl}-5-(2,6- dimethoxyphenyl)- 6-(ethoxymethyl) pyridine-2,4-diol
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|
C25H24ClN3O6
|
1
|
| 1 |
EC50 = 0.23 nM
|
|
|
|
CP0551841
|
3-{5-[(4- chlorophenyl) methyl]- 1,3,4-oxadiazol- 2-yl}-6- cyclopentyl-5-(2,6- dimethoxyphenyl) pyridine-2,4-diol
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|
C27H26ClN3O5
|
1
|
| 1 |
EC50 = 0.51 nM
|
|
|
|
CP0549142
|
3-{5-[(6- chloropyridin-3- yl)methyl]-1,3,4- oxadiazol-2-yl}-5- (2,6- dimethoxyphenyl)- 6-(ethoxymethyl) pyridine-2,4-diol
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|
C24H23ClN4O6
|
1
|
| 1 |
EC50 = 0.58 nM
|
|
|
|
CP0551840
|
6-butyl-3-{5-[(4- chlorophenyl) methyl]-1,3,4- oxadiazol- 2-yl}-5-(2,6- dimethoxyphenyl) pyridine-2,4-diol
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|
C26H26ClN3O5
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
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CP0546376
|
3-[5-[(4-chlorophenyl)methyl]-1,3,4-oxadiazol-2-yl]-5-(2,6-dimethoxyphenyl)-4-hydroxy-6-(2-methoxyethyl)-1H-pyridin-2-one
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|
C25H24ClN3O6
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0551839
|
6-butyl-3-{5-[(3- chlorophenyl) methyl]-1,3,4- oxadiazol- 2-yl}-5-(2,6- dimethoxyphenyl) pyridine-2,4-diol
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|
C26H26ClN3O5
|
1
|
| 1 |
EC50 = 7.3 nM
|
|
|
|
CP0514613
|
3-{5-[(4- chlorophenyl) methyl]-1,3,4- oxadiazol-2-yl}-6- cyclopropyl-5-(2,6- dimethoxyphenyl) pyridine-2,4-diol
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|
C25H22ClN3O5
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0507392
|
6-butyl-3-{5-[(2- chlorophenyl) methyl]-1,3,4- oxadiazol- 2-yl}-5-(2,6- dimethoxyphenyl) pyridine-2,4-diol
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|
C26H26ClN3O5
|
1
|
| 1 |
EC50 = 18 nM
|
|
|
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CP0570145
|
3-(5-benzyl-1,3,4-oxadiazol-2-yl)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-1H-pyridin-2-one
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|
C26H27N3O5
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0570000
|
3-(3-benzyl-1,2,4-oxadiazol-5-yl)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-1H-pyridin-2-one
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|
C26H27N3O5
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0422736
|
3-(5-benzyl-1H-1,2,4-triazol-3-yl)-6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-1H-pyridin-2-one
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|
C26H28N4O4
|
1
|
| 1 |
EC50 = 430 nM
|
|
|
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CP0546375
|
6-butyl-3-[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]-5-(2,6-dimethoxyphenyl)-4-hydroxy-1H-pyridin-2-one
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|
C25H24ClN3O5
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
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CP0537336
|
ethyl 6-butyl-5-(2,6-dimethoxyphenyl)-4-hydroxy-2-oxo-1H-pyridine-3-carboxylate
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|
C20H25NO6
|
1
|
| 1 |
EC50 = 980 nM
|
|
|
