Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT06277 , Probable G-protein coupled receptor 139
Gene Name GPR139
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q6DWJ6
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT06277
 
Compound ID Compound Name Compound Formula
CP0390438
3-chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
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C17H17ClN2O2
 1
1
EC50 = 16 nM
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CP0381712
3-methyl-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
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C18H20N2O2
 1
1
EC50 = 24 nM
   TI
   LI
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   TS
CP0434359
3-chloro-5-fluoro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H16ClFN2O2
 1
1
EC50 = 24 nM
   TI
   LI
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   TS
CP0381711
3,5-dimethoxy-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
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C19H22N2O4
 1
1
EC50 = 32 nM
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CP0443889
3-methoxy-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C18H20N2O3
 1
1
EC50 = 33 nM
   TI
   LI
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   TS
CP0443885
2,5-dichloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H16Cl2N2O2
 1
1
EC50 = 40 nM
   TI
   LI
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   TS
CP0390372
1-[(3,5-dimethoxybenzoyl)amino]-3-naphthalen-1-ylurea
   Show/Hide
C20H19N3O4
 1
1
EC50 = 43 nM
   TI
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   TS
CP0390437
3,5-dichloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H16Cl2N2O2
 1
1
EC50 = 46 nM
   TI
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CP0443887
N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-3-(trifluoromethoxy)benzamide
   Show/Hide
C18H17F3N2O3
 1
1
EC50 = 46 nM
   TI
   LI
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   TS
CP0445235
2,3-dichloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H16Cl2N2O2
 1
1
EC50 = 52 nM
   TI
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   TS
CP0445236
N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]-3-(trifluoromethyl)benzamide
   Show/Hide
C18H17F3N2O2
 1
1
EC50 = 52 nM
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CP0443890
3-fluoro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H17FN2O2
 1
1
EC50 = 54 nM
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CP0475501
3-cyano-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C18H17N3O2
 1
1
EC50 = 59 nM
   TI
   LI
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   TS
CP0894145
3-methoxy-N-((S)-1-oxo-1-(((S)-1-phenylethyl)amino)propan-2-yl)benzamide
   Show/Hide
C19H22N2O3
 1
1
EC50 = 66 nM
   TI
   LI
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   TS
CP0381679
3-bromo-5-chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H16BrClN2O2
 1
1
EC50 = 78 nM
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CP0389352
4-chloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H17ClN2O2
 1
1
EC50 = 118 nM
   TI
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CP0853118
(S)-2-chloro-N-(2-oxo-2-((1-phenylethyl)amino)ethyl)benzamide
   Show/Hide
C17H17ClN2O2
 1
1
EC50 = 150 nM
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CP0849215
(S)-N-(2-oxo-2-((1-phenylethyl)amino)ethyl)benzamide
   Show/Hide
C17H18N2O2
 1
1
EC50 = 162 nM
   TI
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   TS
CP0417855
3,4-dichloro-N-[2-oxo-2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H16Cl2N2O2
 1
1
EC50 = 193 nM
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CP0882251
N-((S)-3-hydroxy-1-oxo-1-(((S)-1-phenylethyl)amino)propan-2-yl)-3-methoxybenzamide
   Show/Hide
C19H22N2O4
 1
1
EC50 = 283 nM
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   TS
CP0894149
3-methoxy-N-((R)-1-oxo-1-(((S)-1-phenylethyl)amino)propan-2-yl)benzamide
   Show/Hide
C19H22N2O3
 1
1
EC50 = 440 nM
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CP0574313
S-[2-oxo-2-(1-phenylethylamino)ethyl] benzenecarbothioate
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C17H17NO2S
 1
1
EC50 = 670 nM
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CP0417857
3-methoxy-N-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C18H20N2O3
 1
1
EC50 = 1700 nM
   TI
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CP0443888
3-chloro-N-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H17ClN2O2
 1
1
EC50 = 2100 nM
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CP0462020
2-[(3-chlorophenyl)methylamino]-N-[(1S)-1-phenylethyl]acetamide
   Show/Hide
C17H19ClN2O
 1
1
EC50 > 10000 nM
   TI
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CP0538923
3-chloro-N-[2-[[(1S)-1-phenylethyl]amino]ethyl]benzamide
   Show/Hide
C17H19ClN2O
 1
1
EC50 > 10000 nM
   TI
   LI
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   TS
CP0850882
3-methoxy-N-((S)-2-oxo-1-phenyl-2-(((S)-1-phenylethyl)amino)ethyl)benzamide
   Show/Hide
C25H26N2O3
 1
1
EC50 = 10000 nM
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