| Compound ID |
Compound Name |
Compound Formula |
|
CP0849165
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-isoxazole-5-carboxamide
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|
C8H6N4O2S2
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
IC50 = 330 nM
|
|
|
|
CP0866297
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-thiophen-2-carboxamide
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|
C9H7N3OS3
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
IC50 = 420 nM
|
|
|
|
CP0911522
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-2-fluorobenzamide
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|
C11H8FN3OS2
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
IC50 = 350 nM
|
|
|
|
CP0865003
|
N-(2-thioxoimidazoIidine-1-carbothioyl)-2,4-difluorobenzamide
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|
C11H9F2N3OS2
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
IC50 = 170 nM
|
|
|
|
CP0930329
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-furan-2-carboxamide
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|
C9H7N3O2S2
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
IC50 = 250 nM
|
|
|
|
CP0849163
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-benzothiophen-2-carboxamide
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|
C13H9N3OS3
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
IC50 = 190 nM
|
|
|
|
CP0926510
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazoI-3-ylidene)-naphthyl-1-carboxamide
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|
C15H11N3OS2
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
IC50 = 450 nM
|
|
|
|
CP0896457
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-pyridine-3-carboxamide
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|
C10H8N4OS2
|
2
|
| 1 |
IC50 = 133 nM
|
|
|
| 2 |
IC50 = 670 nM
|
|
|
|
CP0861661
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-3-methylbenzamide
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|
C12H11N3OS2
|
2
|
| 1 |
IC50 = 140 nM
|
|
|
| 2 |
IC50 = 790 nM
|
|
|
|
CP0867713
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-naphthyl-2-carboxamide
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|
C15H11N3OS2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0874225
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-4-trifluoromethylbenzamide
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|
C12H8F3N3OS2
|
2
|
| 1 |
IC50 = 170 nM
|
|
|
| 2 |
IC50 = 570 nM
|
|
|
|
CP0896460
|
N-(5,6-dihydro-3H-imidazor[2,1-c]-1,2,4-dithiazol-3-ylidene)-benzamide
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|
C11H9N3OS2
|
2
|
| 1 |
IC50 = 170 nM
|
|
|
| 2 |
IC50 = 440 nM
|
|
|
|
CP0867425
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-2-(4-chlorophenyl)-3-(trifluoromethyl)pyrazole-4-carboxamide
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|
C15H9ClF3N5OS2
|
1
|
| 1 |
IC50 = 189.7 nM
|
|
|
|
CP0896463
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-2,4-difluorobenzamide
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|
C11H7F2N3OS2
|
2
|
| 1 |
IC50 = 190 nM
|
|
|
| 2 |
IC50 = 410 nM
|
|
|
|
CP0946865
|
N-(5,6-dhydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-4-fluorobenzamide
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|
C11H8FN3OS2
|
2
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
IC50 = 370 nM
|
|
|
|
CP0865004
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-4-methoxybenzamide
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|
C12H11N3O2S2
|
2
|
| 1 |
IC50 = 210 nM
|
|
|
| 2 |
IC50 = 830 nM
|
|
|
|
CP0874224
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-3-fluorobenzamide
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|
C11H8FN3OS2
|
2
|
| 1 |
IC50 = 220 nM
|
|
|
| 2 |
IC50 = 240 nM
|
|
|
|
CP0867712
|
N-(2-thioxoimidazolidine-1-carbothioyl)-benzothiophen-2-carboxamide
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|
C13H11N3OS3
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
IC50 = 4520 nM
|
|
|
|
CP0858025
|
N-(5,6-dmydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-yldiene)-4-chlorobenzamide
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|
C11H8ClN3OS2
|
2
|
| 1 |
IC50 = 270 nM
|
|
|
| 2 |
IC50 = 640 nM
|
|
|
|
CP0862364
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-3-methoxybenzamide
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|
C12H11N3O2S2
|
2
|
| 1 |
IC50 = 310 nM
|
|
|
| 2 |
IC50 = 400 nM
|
|
|
|
CP0849164
|
N-(5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazol-3-ylidene)-3,5-dimethylisoxazole-4-carboxamide
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|
C10H10N4O2S2
|
2
|
| 1 |
IC50 = 350 nM
|
|
|
| 2 |
IC50 = 460 nM
|
|
|
|
CP0849021
|
N-(5,6-dihydro-3H-imidazor[2,1-c]-1,2,4-dithiazol-3-ylidene)-4-tert-butylbenzamide
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|
C15H17N3OS2
|
2
|
| 1 |
IC50 = 370 nM
|
|
|
| 2 |
IC50 = 650 nM
|
|
|
|
CP0896459
|
N-(2-thioxoimidazoUdine-1-carbothioyl)-4-chlorobenzamide
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|
C11H10ClN3OS2
|
2
|
| 1 |
IC50 = 450 nM
|
|
|
| 2 |
IC50 = 1970 nM
|
|
|
|
CP0849158
|
N-(2-thioxoimidazolidine-1-carbothioyl)-4-fluorobenzamide
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|
C11H10FN3OS2
|
2
|
| 1 |
IC50 = 480 nM
|
|
|
| 2 |
IC50 = 1250 nM
|
|
|
|
CP0849162
|
N-(2-thioxoimidazoIidine-1-carbothioyl)-naphthyl-2-carboxamide
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|
C15H13N3OS2
|
2
|
| 1 |
IC50 = 710 nM
|
|
|
| 2 |
IC50 = 100000 nM
|
|
|
|
CP0869185
|
N-(2-thioxoimidazolidine-1-carbothioyl)-pyridine-3-carboxamide
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|
C10H10N4OS2
|
2
|
| 1 |
IC50 = 850 nM
|
|
|
| 2 |
IC50 = 6560 nM
|
|
|
|
CP0861660
|
N-(2-thioxoimidazolidine-1-carbothioyl)-4-trifluoromethylbenzamide
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|
C12H10F3N3OS2
|
2
|
| 1 |
IC50 = 1570 nM
|
|
|
| 2 |
IC50 = 3650 nM
|
|
|
|
CP0849160
|
N-(2-thioxoimidazolidine-1-carbothioyl)-thiophene-2-carboxamide
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|
C9H9N3OS3
|
2
|
| 1 |
IC50 = 1960 nM
|
|
|
| 2 |
IC50 = 2790 nM
|
|
|
|
CP0896462
|
N-(2-thioxoimidazolidine-1-carbothioyl)-isoxazole-5-carboxamide
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|
C8H8N4O2S2
|
2
|
| 1 |
IC50 = 2430 nM
|
|
|
| 2 |
IC50 = 5830 nM
|
|
|
|
CP0903230
|
N-(5,6-dihydro-3H-imidazo[2,1-c][1,2,4]dithiazol-3-ylidene)-5-methyl-3-phenylisoxazole-4-carboxamide
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|
C15H12N4O2S2
|
1
|
| 1 |
IC50 = 2460 nM
|
|
|
|
CP0896458
|
N-(2-thioxoimidazolidine-1-carbothioyl)-3-fluorobenzamide
Show/Hide
|
C11H10FN3OS2
|
2
|
| 1 |
IC50 = 2620 nM
|
|
|
| 2 |
IC50 = 3190 nM
|
|
|
|
CP0849161
|
N-(2-thioxoimidazolidine-1-carbothioyl)-3-methylbenzamide
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|
C12H13N3OS2
|
1
|
| 1 |
IC50 = 3800 nM
|
|
|
|
CP0858023
|
N-(2-thioxoimidazolidine-1-carbothioyl)-2-fluorobenzamide
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|
C11H10FN3OS2
|
1
|
| 1 |
IC50 = 43000 nM
|
|
|
|
CP0858024
|
N-(2-thioxoimidazolidine-1-carbothioyl)-3-methoxybenzamide
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|
C12H13N3O2S2
|
2
|
| 1 |
IC50 = 51000 nM
|
|
|
| 2 |
IC50 = 56000 nM
|
|
|
|
CP0862390
|
N-(2-thioxoimidazolidine-1-carbothioyl)-4-methoxybenzamide
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|
C12H13N3O2S2
|
1
|
| 1 |
IC50 = 55000 nM
|
|
|
|
CP0850352
|
N-(2-thioxoimidazolidine-1-carbothioyl)-furan-2-carboxamide
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|
C9H9N3O2S2
|
1
|
| 1 |
IC50 = 68290 nM
|
|
|
|
CP0869186
|
N-(2-thioxoimidazolidine-1-carbothioyl)-pyridine-2-methylthio-3-carboxamide
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|
C11H12N4OS3
|
1
|
| 1 |
IC50 = 80000 nM
|
|
|
|
CP0849022
|
N-(2-thioxoimidazolidine-1-carbothioyl)-benzamide
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|
C11H11N3OS2
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
|
CP0857794
|
N-(2-thioxoimidazolidine-1-carbothioyl)-naphthyl-1-carboxamide
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|
C15H13N3OS2
|
1
|
| 1 |
IC50 = 100000 nM
|
|
|
