Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT05857 , Neuropeptide S receptor
Gene Name NPSR1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q6W5P4
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT05857
 
Compound ID Compound Name Compound Formula
CP0487772
N-benzyl-3-oxo-1,1-diphenyl-5,6,8,8a-tetrahydro-[1,3]oxazolo[3,4-a]pyrazine-7-carboxamide
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C26H25N3O3
 1
1
IC50 = 1.995 nM
   TI
   LI
   LO
   TS
CP0288713
5-phenyl-2-(2-(piperidine-1-carbonyl)phenyl)-2,3-dihydro-1H-pyrrolo[1,2-c]imidazol-1-one
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C24H23N3O2
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0511931
6-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]pyridine-2-carboxamide
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C24H23N3O2
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0504543
5-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]furan-2-carboxamide
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C23H22N2O3
 1
1
IC50 = 31.62 nM
   TI
   LI
   LO
   TS
CP0504544
3-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]benzamide
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C25H24N2O2
 1
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
CP0505431
5-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]thiophene-2-carboxamide
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C23H22N2O2S
 1
1
IC50 = 794.33 nM
   TI
   LI
   LO
   TS
CP0479141
7-phenyl-2-[2-(piperidine-1-carbonyl)phenyl]-4,5-dihydro-3H-pyrrolo[1,2-a][1,4]diazepin-1-one
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C26H27N3O2
 1
1
IC50 > 5011.87 nM
   TI
   LI
   LO
   TS
CP0528689
5-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]-1H-pyrrole-2-carboxamide
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C23H23N3O2
 1
1
IC50 > 5011.87 nM
   TI
   LI
   LO
   TS
CP0531143
6-phenyl-2-[2-(piperidine-1-carbonyl)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-one
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C25H25N3O2
 1
1
IC50 > 5011.87 nM
   TI
   LI
   LO
   TS