Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT05334 , ATP-binding cassette sub-family C member 4
Gene Name ABCC4
Organism Homo sapiens, Human
Protein Classification Transporter
Uniprot ID O15439
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT05334
 
Compound ID Compound Name Compound Formula
CP0069487
2-({6-[bis(2-hydroxyethyl)amino]-4,8-bis(piperidin-1-yl)pyrimido[5,4-d][1,3]diazin-2-yl}(2-hydroxyethyl)amino)ethan-1-ol
   Show/Hide
C24H40N8O4
 1
1
IC50 = 2000 nM
   TI
   LI
   LO
   TS
CP0078757
(E)-3-((3-(2-(7-chloroquinolin-2-yl)vinyl)phenyl)(3-(dimethylamino)-3-oxopropylthio)methylthio)propanoic acid
   Show/Hide
C26H27ClN2O3S2
 1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0275436
9,10-Dimethoxy-3-methyl-2-(2,4,6-trimethyl-phenylimino)-2,3,6,7-tetrahydro-pyrimido[6,1-a]isoquinolin-4-one
   Show/Hide
C24H27N3O3
 1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0010658
5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-one
   Show/Hide
C22H30N6O4S
 1
1
IC50 = 20000 nM
   TI
   LI
   LO
   TS
CP0046621
3-[4-[3-(3,4,5-trimethoxybenzoyl)oxypropyl]-1,4-diazepan-1-yl]propyl 3,4,5-trimethoxybenzoate
   Show/Hide
C31H44N2O10
 1
1
IC50 = 20000 nM
   TI
   LI
   LO
   TS
CP0076031
(2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-{[(4-nitrophenyl)methyl]sulfanyl}-9H-purin-9-yl)oxolane-3,4-diol
   Show/Hide
C17H17N5O6S
 1
1
IC50 = 75000 nM
   TI
   LI
   LO
   TS
CP0003146
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
   Show/Hide
C22H21Cl3N4O
 1
1
Ki = 4000 nM
   TI
   LI
   LO
   TS
CP0395393
3,4-diarylpyrazoline derivative
   Show/Hide
C20H24ClN5O2S
 1
1
Ki = 7000 nM
   TI
   LI
   LO
   TS