All Bioactivity

Brief Information of the Cell Line and Protein

Cell Line ID: CL000006 , HEK293

Cell Line Info

Synonyms	Hek293 HEK-293 HEK/293 HEK 293 HEK;293 293 293 HEK 293 Ad5 Graham 293 Graham-293 Human Embryonic Kidney 293
Category	Transformed cell line
Organism	Homo sapiens (Human)
Cellosaurus ID	CVCL_0045

Protein ID: PT04426 , Neuromedin-U receptor 2

Protein Info

Gene Name	NMUR2
Organism	Homo sapiens, Human
Protein Classification	Membrane receptor
Uniprot ID	Q9GZQ4

Table of Molecular Bioactivities Related to the Cell Line and Protein

Cell Line ID: CL000006

Cell Line Info

Protein ID: PT04426

Protein Info

Compound ID	Compound Name	Compound Formula
CP0468381 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-amino-2-methylpropanoyl)amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C49H76N16O9	1
1	EC50 = 0.2138 nM Bioactivity Info	TI LI LO TS
CP0382209 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C47H71N15O9	1
1	EC50 = 0.3388 nM Bioactivity Info	TI LI LO TS
CP0416860 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H84N16O11	2
1	EC50 = 0.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2.4 nM Bioactivity Info	TI LI LO TS
CP0427425 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O11	2
1	EC50 = 0.71 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2 nM Bioactivity Info	TI LI LO TS
CP0382217 Compound Info	(4S)-5-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-hydroxy-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-4-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylbutanoyl]amino]-3-carboxypropanoyl]amino]-4-carboxybutanoyl]amino]-5-oxopentanoic acid Show/Hide	C141H203N41O38	2
1	EC50 = 0.7943 nM Bioactivity Info	TI LI LO TS
2	EC50 = 6100 nM Bioactivity Info	TI LI LO TS
CP0384732 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H82N16O10	2
1	EC50 = 0.83 nM Bioactivity Info	TI LI LO TS
2	IC50 = 4.3 nM Bioactivity Info	TI LI LO TS
CP0416852 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-naphthalen-2-ylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C60H82N16O10	2
1	EC50 = 1.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 5.6 nM Bioactivity Info	TI LI LO TS
CP0389655 Compound Info	(2S)-2-[[(2S)-2-[[(2S,3aS,7aS)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]-2,3,3a,4,5,6,7,7a-octahydroindole-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C60H86N16O11	2
1	EC50 = 1.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 13.9 nM Bioactivity Info	TI LI LO TS
CP0382214 Compound Info	(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[2-[3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-(hexadecanoylamino)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C92H159N17O23	1
1	EC50 = 1.905 nM Bioactivity Info	TI LI LO TS
CP0475615 Compound Info	(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(3S)-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C55H78N16O10	2
1	EC50 = 3.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 21.4 nM Bioactivity Info	TI LI LO TS
CP0381405 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-3-amino-2-[[(2S)-2-[[(2S)-2-(3-cyclohexylpropanoylamino)-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C39H70N12O8	2
1	EC50 = 3.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 43.9 nM Bioactivity Info	TI LI LO TS
CP0412753 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3,4-dihydro-1H-naphthalene-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H82N16O11	2
1	EC50 = 3.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 40.4 nM Bioactivity Info	TI LI LO TS
CP0431735 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-naphthalen-2-ylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H80N16O9	2
1	EC50 = 4.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 9.9 nM Bioactivity Info	TI LI LO TS
CP0384721 Compound Info	(2S)-2-[[(2S)-2-[[(3S)-2-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C61H82N16O11	2
1	EC50 = 5.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 11.2 nM Bioactivity Info	TI LI LO TS
CP0389657 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O11	1
1	EC50 = 6.2 nM Bioactivity Info	TI LI LO TS
CP0384722 Compound Info	(2S)-2-[[(2S)-2-[[(2S,3aS,7aS)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]-2,3,3a,4,5,6,7,7a-octahydroindole-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H84N16O10	2
1	EC50 = 10.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 12.7 nM Bioactivity Info	TI LI LO TS
CP0468138 Compound Info	(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[2-(hexadecylamino)-2-oxoethyl]amino]acetyl]amino]-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C69H114N18O11	1
1	EC50 = 10.23 nM Bioactivity Info	TI LI LO TS
CP0417357 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(3S)-2-acetyl-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C57H80N16O11	2
1	EC50 = 13.4 nM Bioactivity Info	TI LI LO TS
2	IC50 = 12.3 nM Bioactivity Info	TI LI LO TS
CP0427494 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N'-benzylbutanediamide Show/Hide	C63H86N16O11	2
1	EC50 = 28.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 18.8 nM Bioactivity Info	TI LI LO TS
CP0384718 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O10	2
1	EC50 = 30.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1.7 nM Bioactivity Info	TI LI LO TS
CP0416855 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O10	1
1	EC50 = 34.3 nM Bioactivity Info	TI LI LO TS
CP0471661 Compound Info	(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[2-(hexadecylamino)-2-oxoethyl]-(pyridine-3-carbonyl)amino]acetyl]amino]-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C75H117N19O12	1
1	EC50 = 42.66 nM Bioactivity Info	TI LI LO TS
CP0416859 Compound Info	(2S)-2-[[(2S)-2-[[(3S)-2-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C59H80N16O10	2
1	EC50 = 45.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 13 nM Bioactivity Info	TI LI LO TS
CP0383781 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N'-methylbutanediamide Show/Hide	C57H82N16O11	2
1	EC50 = 51.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 29.1 nM Bioactivity Info	TI LI LO TS
CP0466621 Compound Info	(2S)-2-[[(3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-6-(diaminomethylideneamino)hexanoyl]amino]butanediamide Show/Hide	C57H82N16O11	2
1	EC50 = 55.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 116.5 nM Bioactivity Info	TI LI LO TS
CP0389563 Compound Info	(2S)-N-(1-amino-2-methyl-1-oxopropan-2-yl)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(2-amino-2-methylpropanoyl)amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C53H83N17O10	1
1	EC50 = 56.23 nM Bioactivity Info	TI LI LO TS
CP0427493 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(3S)-2-acetyl-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-3-aminopropanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H74N14O11	2
1	EC50 = 59.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 72.4 nM Bioactivity Info	TI LI LO TS
CP0382212 Compound Info	(2R)-N-(1-amino-2-methyl-1-oxopropan-2-yl)-2-[[(2R)-5-(diaminomethylideneamino)-2-[[(2R)-1-[(2R)-5-(diaminomethylideneamino)-2-[[(2R)-2-[[(2R)-2-[[(2S)-2-[[2-[3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-(hexadecanoylamino)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C96H166N18O24	1
1	EC50 = 107.15 nM Bioactivity Info	TI LI LO TS
CP0382213 Compound Info	(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-(hexadecanoylamino)-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C65H106N16O10	1
1	EC50 = 107.15 nM Bioactivity Info	TI LI LO TS
CP0389658 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(3S)-2-[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C57H80N16O12	2
1	EC50 = 192.6 nM Bioactivity Info	TI LI LO TS
2	IC50 = 330.8 nM Bioactivity Info	TI LI LO TS
CP0394602 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-naphthalen-1-ylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H80N16O10	2
1	EC50 = 225.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 370.5 nM Bioactivity Info	TI LI LO TS
CP0384729 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C53H73N13O11	1
1	EC50 = 242.2 nM Bioactivity Info	TI LI LO TS
CP0431739 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-naphthalen-1-ylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C60H82N16O11	2
1	EC50 = 246.5 nM Bioactivity Info	TI LI LO TS
2	IC50 = 39.1 nM Bioactivity Info	TI LI LO TS
CP0389660 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-(2-phenylethyl)amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C57H82N16O11	2
1	EC50 = 250 nM Bioactivity Info	TI LI LO TS
2	IC50 = 316.1 nM Bioactivity Info	TI LI LO TS
CP0382210 Compound Info	(2S)-N-[6-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-6-oxohexyl]-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[6-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]hexanoylamino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C63H101N19O12S2	1
1	EC50 = 281.84 nM Bioactivity Info	TI LI LO TS
CP0431736 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-naphthalen-2-ylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C60H82N16O11	2
1	EC50 = 304.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 195.3 nM Bioactivity Info	TI LI LO TS
CP0431733 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-[2-(4-hydroxyphenyl)ethyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C57H82N16O12	2
1	EC50 = 339.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 206.9 nM Bioactivity Info	TI LI LO TS
CP0427537 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-benzylbutanediamide Show/Hide	C63H86N16O11	2
1	EC50 = 354.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 28.8 nM Bioactivity Info	TI LI LO TS
CP0384716 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-(2-phenylethyl)amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C55H80N16O10	2
1	EC50 = 355.7 nM Bioactivity Info	TI LI LO TS
2	IC50 = 261.6 nM Bioactivity Info	TI LI LO TS
CP0394604 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-naphthalen-2-ylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H80N16O10	2
1	EC50 = 378 nM Bioactivity Info	TI LI LO TS
2	IC50 = 424.4 nM Bioactivity Info	TI LI LO TS
CP0384727 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-[2-(4-hydroxyphenyl)ethyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C55H80N16O11	2
1	EC50 = 382.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 428.9 nM Bioactivity Info	TI LI LO TS
CP0477382 Compound Info	(2S)-2-[[(2R)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O11	1
1	EC50 = 382.3 nM Bioactivity Info	TI LI LO TS
CP0427426 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C51H71N13O10	1
1	EC50 = 391 nM Bioactivity Info	TI LI LO TS
CP0427538 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-methylbutanediamide Show/Hide	C57H82N16O11	2
1	EC50 = 440.8 nM Bioactivity Info	TI LI LO TS
2	IC50 = 327.5 nM Bioactivity Info	TI LI LO TS
CP0402741 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(3S)-2-acetyl-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-naphthalen-2-ylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C61H82N16O11	2
1	EC50 = 459.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 301.9 nM Bioactivity Info	TI LI LO TS
CP0389654 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S,3aS,7aS)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-2,3,3a,4,5,6,7,7a-octahydroindole-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H82N16O10	2
1	EC50 = 472.1 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1546 nM Bioactivity Info	TI LI LO TS
CP0536862 Compound Info	(2S)-2-[[(2R)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O10	1
1	EC50 = 616.1 nM Bioactivity Info	TI LI LO TS
CP0389661 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(3S)-2-[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C55H78N16O11	2
1	EC50 = 624.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1010 nM Bioactivity Info	TI LI LO TS
CP0382211 Compound Info	(2S)-2-[[(2S)-2-[[(2S,3aS,7aS)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[6-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]hexanoylamino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]-2,3,3a,4,5,6,7,7a-octahydroindole-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-N-[6-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-6-oxohexyl]butanediamide Show/Hide	C67H107N19O12S2	1
1	EC50 = 724.44 nM Bioactivity Info	TI LI LO TS
CP0461928 Compound Info	(2R)-2-[[(2R)-5-(diaminomethylideneamino)-2-[[(2R)-1-[(2R)-5-(diaminomethylideneamino)-2-[[(2R)-2-[[(2R)-2-[[(2S)-2-[[2-[6-(dihexadecylamino)hexanoylamino]-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C87H151N17O10	1
1	EC50 = 794.33 nM Bioactivity Info	TI LI LO TS
CP0412755 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(3S)-2-acetyl-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-methylamino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H82N16O11	2
1	EC50 = 925.2 nM Bioactivity Info	TI LI LO TS
2	IC50 = 465.5 nM Bioactivity Info	TI LI LO TS
CP0384730 Compound Info	(2S)-2-[[(2S)-2-[[(2R)-1-[(2S)-3-amino-2-[[(2S)-2-[[(2S)-2-(3-cyclohexylpropanoylamino)-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C39H70N12O8	2
1	EC50 = 926.3 nM Bioactivity Info	TI LI LO TS
2	IC50 = 10700 nM Bioactivity Info	TI LI LO TS
CP0537487 Compound Info	(5R,15R,18R,21R,27R,30R,33S,36R,46R)-46-amino-15-(2-amino-2-oxoethyl)-30,36-dibenzyl-18,27-bis[3-(diaminomethylideneamino)propyl]-52-(hexadecylsulfanylmethyl)-33-(2-methylpropyl)-7,14,17,20,26,29,32,35,38,45-decaoxo-3,48-dithia-6,13,16,19,25,28,31,34,37,44-decazatricyclo[48.3.1.021,25]tetrapentaconta-1(53),50(54),51-triene-5-carboxamide Show/Hide	C88H141N19O12S3	1
1	EC50 = 1000 nM Bioactivity Info	TI LI LO TS
CP0431740 Compound Info	(2S)-2-[[(2S)-2-[[(2R)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O10	2
1	EC50 = 1079 nM Bioactivity Info	TI LI LO TS
2	IC50 = 802.9 nM Bioactivity Info	TI LI LO TS
CP0431738 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-benzylamino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O10	2
1	EC50 = 1103 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1403 nM Bioactivity Info	TI LI LO TS
CP0660469 Compound Info	Rutin Show/Hide	C27H30O16	1
1	EC50 = 1200 nM Bioactivity Info	TI LI LO TS
CP0384726 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-benzylamino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O11	2
1	EC50 = 1278 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1019 nM Bioactivity Info	TI LI LO TS
CP0431737 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H82N16O11	2
1	EC50 = 1286 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1649 nM Bioactivity Info	TI LI LO TS
CP0389659 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-[(4-hydroxyphenyl)methyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O11	2
1	EC50 = 1407 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1961 nM Bioactivity Info	TI LI LO TS
CP0417359 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S,3aS,7aS)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-2,3,3a,4,5,6,7,7a-octahydroindole-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H84N16O11	2
1	EC50 = 1830 nM Bioactivity Info	TI LI LO TS
2	IC50 = 253.4 nM Bioactivity Info	TI LI LO TS
CP0412793 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C60H88N16O12	2
1	EC50 = 1993 nM Bioactivity Info	TI LI LO TS
2	IC50 = 2869 nM Bioactivity Info	TI LI LO TS
CP0431734 Compound Info	(2S)-2-[[(2S)-2-[[(2R)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O11	2
1	EC50 = 2002 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1365 nM Bioactivity Info	TI LI LO TS
CP0412788 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(3S)-2-acetyl-7-hydroxy-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-[2-(4-hydroxyphenyl)ethyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H82N16O12	2
1	EC50 = 2205 nM Bioactivity Info	TI LI LO TS
2	IC50 = 598.9 nM Bioactivity Info	TI LI LO TS
CP0389656 Compound Info	(2S)-2-[[(2S)-2-[[(2R)-1-[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C54H78N16O10	2
1	EC50 = 2495 nM Bioactivity Info	TI LI LO TS
2	IC50 = 6132 nM Bioactivity Info	TI LI LO TS
CP0549774 Compound Info	(2S)-N-[6-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-6-oxohexyl]-2-[[(2S)-2-[[(3R)-2-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[6-[[(2R)-2-amino-3-sulfanylpropanoyl]amino]hexanoylamino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C68H103N19O12S2	1
1	EC50 = 2511.89 nM Bioactivity Info	TI LI LO TS
CP0394534 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-[(4-hydroxyphenyl)methyl]amino]acetyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O12	2
1	EC50 = 2686 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1813 nM Bioactivity Info	TI LI LO TS
CP0427427 Compound Info	(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C58H84N16O12	2
1	EC50 = 3675 nM Bioactivity Info	TI LI LO TS
2	IC50 = 1857 nM Bioactivity Info	TI LI LO TS
CP0468136 Compound Info	(5R,15R,18R,21R,32R,35R,38S,41R,51R)-51-amino-15-(2-amino-2-oxoethyl)-35,41-dibenzyl-18,32-bis[3-(diaminomethylideneamino)propyl]-57-(hexadecylsulfanylmethyl)-38-(2-methylpropyl)-7,14,17,20,31,34,37,40,43,50-decaoxo-3,53-dithia-6,13,16,19,30,33,36,39,42,49-decazatetracyclo[53.3.1.021,30.023,28]nonapentaconta-1(58),23,25,27,55(59),56-hexaene-5-carboxamide Show/Hide	C93H143N19O12S3	1
1	EC50 = 6309.57 nM Bioactivity Info	TI LI LO TS
CP0549775 Compound Info	(5S,15S,18S,21S,23S,28S,31S,34S,37R,40S,50S)-50-amino-15-(2-amino-2-oxoethyl)-34,40-dibenzyl-18,31-bis[3-(diaminomethylideneamino)propyl]-56-(hexadecylsulfanylmethyl)-37-(2-methylpropyl)-7,14,17,20,30,33,36,39,42,49-decaoxo-3,52-dithia-6,13,16,19,29,32,35,38,41,48-decazatetracyclo[52.3.1.021,29.023,28]octapentaconta-1(57),54(58),55-triene-5-carboxamide Show/Hide	C92H147N19O12S3	1
1	EC50 = 6309.57 nM Bioactivity Info	TI LI LO TS
CP0158214 Compound Info	CHEBI:29081 Show/Hide	C9H13NO2	1
1	EC50 = 6600 nM Bioactivity Info	TI LI LO TS
CP0468135 Compound Info	(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[hexadecyl-[2-(hexadecylamino)-2-oxoethyl]amino]acetyl]amino]-2-methylpropanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]amino]butanediamide Show/Hide	C85H146N18O11	1
1	EC50 = 10000 nM Bioactivity Info	TI LI LO TS
CP0052539 Compound Info	2-(5-bromo-2-fluorophenyl)-3-hydroxychromen-4-one Show/Hide	C15H8BrFO3	1
1	EC50 = 14000 nM Bioactivity Info	TI LI LO TS
CP0052386 Compound Info	2-(3-chloro-2-fluorophenyl)-3-hydroxychromen-4-one Show/Hide	C15H8ClFO3	1
1	EC50 = 31100 nM Bioactivity Info	TI LI LO TS
CP0051300 Compound Info	2-(2-fluorophenyl)-3-hydroxychromen-4-one Show/Hide	C15H9FO3	1
1	EC50 = 37300 nM Bioactivity Info	TI LI LO TS
CP0052537 Compound Info	2-(5-bromo-2-fluorophenyl)-3-(2-hydroxyethoxy)chromen-4-one Show/Hide	C17H12BrFO4	1
1	EC50 = 47000 nM Bioactivity Info	TI LI LO TS
CP0042940 Compound Info	2-(4-bromo-2-fluorophenyl)-3-hydroxychromen-4-one Show/Hide	C15H8BrFO3	1
1	EC50 = 73000 nM Bioactivity Info	TI LI LO TS
CP0513831 Compound Info	(2S)-2-[[(2S)-2-[[(2R)-1-[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]butanediamide Show/Hide	C56H80N16O11	1
1	IC50 = 1089 nM Bioactivity Info	TI LI LO TS

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About MolBiC

Correspondence

Prof. Feng ZHU

Prof. Leo, Lianyi Han