Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
 Cell Line Info 
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT04124 , Proteinase-activated receptor 2
 Protein Info 
Gene Name F2RL1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P55085
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006
 Cell Line Info 
 Protein ID: PT04124
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0415492
 Compound Info 
N-[(2S)-1-[[(2S,3S)-1-[[2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1-[[(2S)-1,5-diamino-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]furan-2-carboxamide
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C36H63N11O8
  1
1
EC50 = 430 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0391712
 Compound Info 
N-[(2S)-1-[[(1S)-2-amino-1-cyclohexyl-2-oxoethyl]amino]-3-cyclohexyl-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide
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C21H32N4O4
  1
1
EC50 = 2000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0416378
 Compound Info 
N-[(2S)-1-[[2-(2-amino-2-oxoethyl)phenyl]methylamino]-3-cyclohexyl-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide
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C22H28N4O4
  1
1
EC50 = 6000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0437443
 Compound Info 
N-[(2S)-1-[[2-(2-amino-2-oxoethyl)cyclohexyl]methylamino]-3-cyclohexyl-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide
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C22H34N4O4
  1
1
EC50 = 7400 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0411027
 Compound Info 
N-[(2S)-1-[[2-(2-amino-2-oxoethyl)phenyl]methylamino]-3-cyclohexyl-1-oxopropan-2-yl]-3-methyl-1,2-oxazole-5-carboxamide
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C23H30N4O4
  1
1
EC50 = 8900 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0535094
 Compound Info 
N-[(2S)-1-[[2-(2-amino-2-oxoethyl)phenyl]methylamino]-3-cyclohexyl-1-oxopropan-2-yl]-3-ethyl-1,2-oxazole-5-carboxamide
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C24H32N4O4
  1
1
EC50 = 18000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0386689
 Compound Info 
2-Furoyl-Cha-Ile-NH2
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C20H31N3O4
  1
1
EC50 > 50000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0504401
 Compound Info 
4-(2-Methyloxazoyl)-Cha-Ile-NH2
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C20H32N4O4
  1
1
EC50 > 100000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0527231
 Compound Info 
2-Pyrazoyl-Cha-Ile-NH2
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C20H31N5O3
  1
1
EC50 > 100000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0526352
 Compound Info 
5-Isoxazoyl-Cha-Ile-NH2
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C19H30N4O4
  1
1
EC50 > 4000 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS