| Compound ID |
Compound Name |
Compound Formula |
|
CP0519430
|
CHEMBL4559031
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|
C26H35ClN4O4S
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
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CP0543819
|
5-cyclopropyl-N-[1-[[4-[(4-fluorophenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C26H35FN4O4S
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
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CP0549210
|
N-[1-[[4-(benzylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C26H36N4O4S
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
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CP0551369
|
5-cyclopropyl-N-[1-[[4-[(2-fluorophenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C26H35FN4O4S
|
1
|
| 1 |
EC50 = 22 nM
|
|
|
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CP0558515
|
N-[1-[[4-[(5-chloropyridin-2-yl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C25H34ClN5O4S
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
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CP0559798
|
5-cyclopropyl-N-[1-[[4-[(5-fluoropyridin-3-yl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C25H34FN5O4S
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0427691
|
N-[1-[[4-[(3-chlorophenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C26H35ClN4O4S
|
1
|
| 1 |
EC50 = 29 nM
|
|
|
|
CP0438642
|
N-[1-[[4-[(2-chlorophenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C26H35ClN4O4S
|
1
|
| 1 |
EC50 = 31 nM
|
|
|
|
CP0427692
|
5-cyclopropyl-N-[1-[[4-[(2-methylphenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C27H38N4O4S
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
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CP0519429
|
5-cyclopropyl-N-[1-[[4-[(3-fluorophenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C26H35FN4O4S
|
1
|
| 1 |
EC50 = 38 nM
|
|
|
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CP0224428
|
5-cyclopropyl-N-[1-[[4-(4,4,4-trifluorobutylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C23H35F3N4O4S
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
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CP0438646
|
5-cyclopropyl-N-[1-[[4-[(5-fluoropyridin-2-yl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C25H34FN5O4S
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
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CP0145225
|
5-cyclopropyl-N-[1-[4-(4,4,4-trifluorobutylamino)cyclohexyl]sulfonylpiperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C22H33F3N4O4S
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
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CP0558513
|
5-cyclopropyl-N-[1-[[4-[(5-methylpyridin-2-yl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C26H37N5O4S
|
1
|
| 1 |
EC50 = 48 nM
|
|
|
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CP0559797
|
5-cyclopropyl-N-[1-[[4-[(3-methylphenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C27H38N4O4S
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
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CP0559794
|
5-cyclopropyl-N-[1-[[4-[(4-methylphenyl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C27H38N4O4S
|
1
|
| 1 |
EC50 = 54 nM
|
|
|
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CP0550758
|
5-cyclopropyl-N-[1-[[4-(pyridin-3-ylmethylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C25H35N5O4S
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
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CP0534505
|
5-cyclopropyl-N-[1-[[4-[(4-fluoropyridin-2-yl)methylamino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C25H34FN5O4S
|
1
|
| 1 |
EC50 = 58 nM
|
|
|
|
CP0519431
|
CHEMBL4455165
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|
C25H35N5O4S
|
1
|
| 1 |
EC50 = 71 nM
|
|
|
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CP0534502
|
N-[1-(4-aminocyclohexyl)sulfonylpiperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C18H28N4O4S
|
1
|
| 1 |
EC50 = 71 nM
|
|
|
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CP0519428
|
5-cyclopropyl-N-[1-[[4-(3,3,3-trifluoropropylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C22H33F3N4O4S
|
1
|
| 1 |
EC50 = 72 nM
|
|
|
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CP0543818
|
CHEMBL4521928
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|
C19H30N4O4S
|
1
|
| 1 |
EC50 = 73 nM
|
|
|
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CP0427689
|
N-[1-[[4-(butylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C23H38N4O4S
|
1
|
| 1 |
EC50 = 95 nM
|
|
|
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CP0558514
|
5-cyclopropyl-N-[1-[[4-(3,3-dimethylbutylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C25H42N4O4S
|
1
|
| 1 |
EC50 = 128 nM
|
|
|
|
CP0558512
|
CHEMBL4563960
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|
C23H38N4O4S
|
1
|
| 1 |
EC50 = 156 nM
|
|
|
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CP0534710
|
N-[1-(4-aminocyclohexyl)sulfonylpiperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C18H28N4O4S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
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CP0519433
|
5-cyclopropyl-N-[1-[[4-(2,2-dimethylpropylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C24H40N4O4S
|
1
|
| 1 |
EC50 = 173 nM
|
|
|
|
CP0551372
|
CHEMBL4473729
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|
C22H36N4O4S
|
1
|
| 1 |
EC50 = 177 nM
|
|
|
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CP0557254
|
N-[1-[4-(azetidin-1-ylmethyl)phenyl]sulfonylpiperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
Show/Hide
|
C22H28N4O4S
|
1
|
| 1 |
EC50 = 179 nM
|
|
|
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CP0543817
|
5-cyclopropyl-N-[1-[[4-(methylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C20H32N4O4S
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
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CP0352195
|
5-cyclopropyl-N-(1-piperidin-4-ylsulfonylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
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|
C17H26N4O4S
|
1
|
| 1 |
EC50 = 183 nM
|
|
|
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CP0519427
|
5-cyclopropyl-N-[1-[[4-(dimethylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C21H34N4O4S
|
1
|
| 1 |
EC50 = 199 nM
|
|
|
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CP0519426
|
N-[1-[4-(aminomethyl)phenyl]sulfonylpiperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C19H24N4O4S
|
1
|
| 1 |
EC50 = 204 nM
|
|
|
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CP0427688
|
5-cyclopropyl-N-[1-[[4-(ethylamino)cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C21H34N4O4S
|
1
|
| 1 |
EC50 = 205 nM
|
|
|
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CP0519425
|
N-[1-[4-(aminomethyl)cyclohexyl]sulfonylpiperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C19H30N4O4S
|
1
|
| 1 |
EC50 = 237 nM
|
|
|
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CP0557253
|
5-cyclopropyl-N-[1-[[4-[methyl(4,4,4-trifluorobutyl)amino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C24H37F3N4O4S
|
1
|
| 1 |
EC50 = 261 nM
|
|
|
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CP0438644
|
5-cyclopropyl-N-[1-(1-methylpiperidin-4-yl)sulfonylpiperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C18H28N4O4S
|
1
|
| 1 |
EC50 = 300 nM
|
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CP0558511
|
5-cyclopropyl-N-[1-[4-(pyrrolidin-1-ylmethyl)phenyl]sulfonylpiperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C23H30N4O4S
|
1
|
| 1 |
EC50 = 373 nM
|
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CP0534709
|
N-[1-(4-aminobutylsulfonyl)piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide
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|
C16H26N4O4S
|
1
|
| 1 |
EC50 = 494 nM
|
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CP0423546
|
5-cyclopropyl-N-[1-[4-[(dimethylamino)methyl]phenyl]sulfonylpiperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C21H28N4O4S
|
1
|
| 1 |
EC50 = 597 nM
|
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CP0424121
|
5-cyclopropyl-N-(1-pyrrolidin-3-ylsulfonylpiperidin-4-yl)-1,2-oxazole-3-carboxamide
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|
C16H24N4O4S
|
1
|
| 1 |
EC50 = 611 nM
|
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CP0534504
|
5-cyclopropyl-N-[1-(1-ethylpiperidin-4-yl)sulfonylpiperidin-4-yl]-1,2-oxazole-3-carboxamide
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|
C19H30N4O4S
|
1
|
| 1 |
EC50 = 617 nM
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CP0534503
|
5-cyclopropyl-N-[1-[[4-[ethyl(4,4,4-trifluorobutyl)amino]cyclohexyl]methylsulfonyl]piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C25H39F3N4O4S
|
1
|
| 1 |
EC50 = 758 nM
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CP0519432
|
5-cyclopropyl-N-[1-[4-(piperidin-1-ylmethyl)phenyl]sulfonylpiperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C24H32N4O4S
|
1
|
| 1 |
EC50 = 919 nM
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CP0438643
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5-cyclopropyl-N-[1-(3-pyrrolidin-1-ylpropylsulfonyl)piperidin-4-yl]-1,2-oxazole-3-carboxamide
Show/Hide
|
C19H30N4O4S
|
1
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| 1 |
EC50 = 1517 nM
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