Compound ID |
Compound Name |
Compound Formula |
CP0505722
|
2-Amino-6-((R)-4-carboxy-4-(dodecylamino)butanamido)heptanedioic Acid
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|
C24H45N3O7
|
1
|
1 |
EC50 = 0.023 nM
|
|
|
CP0505721
|
2-Amino-6-((R)-4-carboxy-4-dodecanamidobutanamido)heptanedioic Acid
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|
C24H43N3O8
|
1
|
1 |
EC50 = 0.027 nM
|
|
|
CP0474419
|
2-Amino-6-((R)-4-amino-5-oxo-5-(undecyloxy)pentanamido)heptanedioic Acid
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|
C23H43N3O7
|
1
|
1 |
EC50 = 0.066 nM
|
|
|
CP0437178
|
2-Amino-6-((R)-4-dodecanamido-5-ethoxy-5-oxopentanamido)heptanedioic Acid
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|
C26H47N3O8
|
1
|
1 |
EC50 = 0.069 nM
|
|
|
CP0490822
|
2-Amino-6-((R)-4-carboxy-4-(dihexadecylamino)butanamido)heptanedioic Acid
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|
C44H85N3O7
|
1
|
1 |
EC50 = 0.12 nM
|
|
|
CP0539461
|
2-Amino-6-((R)-4-dodecanamido-5-oxo-5-(undecyloxy)pentanamido)heptanedioic Acid
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|
C35H65N3O8
|
1
|
1 |
EC50 = 0.134 nM
|
|
|
CP0395975
|
(2R)-5-((6-Amino-1,7-diethoxy-1,7-dioxoheptan-2-yl)amino)-2-dodecanamido-5-oxopentanoicAcid
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|
C28H51N3O8
|
1
|
1 |
EC50 = 0.145 nM
|
|
|
CP0505724
|
diethyl 2-amino-6-[[(4R)-4-amino-5-oxo-5-undecylsulfanylpentanoyl]amino]heptanedioate
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|
C27H51N3O6S
|
1
|
1 |
EC50 = 0.181 nM
|
|
|
CP0501409
|
2-Amino-6-((R)-4-carboxy-4-(dioctylamino)butanamido)heptanedioic Acid
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|
C28H53N3O7
|
1
|
1 |
EC50 = 0.2 nM
|
|
|
CP0437177
|
(15R)-10,6-Dibenzyl 15-Ethyl-2,2-dimethyl-4,12,17-trioxo-3-oxa-5,11,16-triazaoctacosane-6,10,15-tricarboxylate
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|
C24H45N5O7
|
1
|
1 |
EC50 = 0.238 nM
|
|
|
CP0505726
|
(R)-2-Amino-6-((R)-4-carboxy-4-dodecanamidobutanamido)hexanoic Acid
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|
C23H43N3O6
|
1
|
1 |
EC50 = 0.37 nM
|
|
|
CP0490823
|
2-Amino-6-(5-oxo-5-(undecyloxy)pentanamido)heptanedioic Acid
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|
C23H42N2O7
|
1
|
1 |
EC50 = 0.39 nM
|
|
|
CP0395976
|
2-Amino-6-(4-dodecanamidobutanamido)heptanedioic Acid
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|
C23H43N3O6
|
1
|
1 |
EC50 = 0.504 nM
|
|
|
CP0501408
|
2-((R)-4-Amino-4-carboxybutanamido)-6-dodecanamidoheptanedioic Acid
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|
C24H43N3O8
|
1
|
1 |
EC50 = 0.55 nM
|
|
|
CP0501412
|
(S)-6-Amino-2-((R)-4-carboxy-4-dodecanamidobutanamido)hexanoic Acid
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|
C23H43N3O6
|
1
|
1 |
EC50 = 0.57 nM
|
|
|
CP0522931
|
2-((R)-4-Carboxy-4-dodecanamidobutanamido)-6-dodecanamidoheptanedioic Acid
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|
C36H65N3O9
|
1
|
1 |
EC50 = 0.58 nM
|
|
|
CP0505723
|
2-((R)-4-Carboxy-4-dodecanamidobutanamido)-6-guanidinoheptanedioic Acid
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|
C25H45N5O8
|
1
|
1 |
EC50 = 0.622 nM
|
|
|
CP0539460
|
2-Amino-6-((R)-4-amino-5-oxo-5-(undecylamino)pentanamido)heptanedioic Acid
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|
C23H44N4O6
|
1
|
1 |
EC50 = 0.826 nM
|
|
|
CP0474420
|
(S)-2-Amino-6-((R)-4-carboxy-4-dodecanamidobutanamido)hexanoic Acid
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|
C23H43N3O6
|
1
|
1 |
EC50 = 0.96 nM
|
|
|
CP0933358
|
(2R)-5-((4-(2-Amino-4-oxo-4,5-dihydro-1H-imidazol-5-yl)-1-carboxybutyl)amino)-2-dodecanamido-5-oxopentanoic Acid
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|
C25H43N5O7
|
1
|
1 |
EC50 = 1.31 nM
|
|
|
CP0511809
|
(2R)-2-Dodecanamido-5-oxo-5-((2-oxoazepan-3-yl)amino)pentanoic Acid
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|
C23H41N3O5
|
1
|
1 |
EC50 = 1.73 nM
|
|
|
CP0404988
|
2-((R)-4-Carboxy-4-dodecanamidobutanamido)heptanedioic Acid
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|
C24H42N2O8
|
1
|
1 |
EC50 > 100 nM
|
|
|
CP0501410
|
(R)-5-((5-Aminopentyl)amino)-2-dodecanamido-5-oxopentanoic Acid
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|
C22H43N3O4
|
1
|
1 |
EC50 > 100 nM
|
|
|
CP0505725
|
(R)-6-Amino-2-((R)-4-carboxy-4-dodecanamidobutanamido)hexanoic Acid
Show/Hide
|
C23H43N3O6
|
1
|
1 |
EC50 > 100 nM
|
|
|
CP0142376
|
(1-tosylbenzimidazol-2-yl)amine
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|
C14H13N3O2S
|
1
|
1 |
IC50 = 771 nM
|
|
|
CP0552892
|
5-ethyl-N-[2-fluoro-5-(2-methyl-4-oxoquinazolin-3-yl)phenyl]thiophene-2-sulfonamide
Show/Hide
|
C21H18FN3O3S2
|
1
|
1 |
IC50 = 1000 nM
|
|
|
CP0537944
|
2-[2-[3-[benzenesulfonyl(methyl)amino]propyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C28H30N4O3S
|
1
|
1 |
IC50 = 1660 nM
|
|
|
CP0422149
|
2-[2-[2-[benzenesulfonyl(methyl)amino]ethyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C27H28N4O3S
|
1
|
1 |
IC50 = 2560 nM
|
|
|
CP0487640
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-[[5-(dimethylamino)naphthalen-1-yl]sulfonylamino]ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C32H33N5O3S
|
1
|
1 |
IC50 = 2680 nM
|
|
|
CP0422098
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-[[5-(dimethylamino)naphthalen-1-yl]sulfonyl-methylamino]ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C33H35N5O3S
|
1
|
1 |
IC50 = 3080 nM
|
|
|
CP0534935
|
2-[2-[3-(benzenesulfonamido)propyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C27H28N4O3S
|
1
|
1 |
IC50 = 9250 nM
|
|
|
CP0375351
|
4-benzyl-1-pentylbenzimidazol-2-amine
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|
C19H23N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0375352
|
N-(1-pentylbenzimidazol-2-yl)acetamide
Show/Hide
|
C14H19N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0375357
|
1-pentyl-4-phenylbenzimidazol-2-amine
Show/Hide
|
C18H21N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0375359
|
3-pentylbenzo[f]benzimidazol-2-amine
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|
C16H19N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0400246
|
1-pentylbenzo[e]benzimidazol-2-amine
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|
C16H19N3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0410599
|
1-pentyl-4-phenylmethoxybenzimidazol-2-amine
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|
C19H23N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0552400
|
3-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]-N-phenylpropanamide
Show/Hide
|
C27H26N4O2
|
1
|
1 |
IC50 = 12400 nM
|
|
|
CP0422101
|
tert-butyl 4-[2-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]ethylcarbamoyl]piperidine-1-carboxylate
Show/Hide
|
C31H39N5O4
|
1
|
1 |
IC50 = 13300 nM
|
|
|
CP0422152
|
N-[3-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]propyl]benzamide
Show/Hide
|
C28H28N4O2
|
1
|
1 |
IC50 = 17700 nM
|
|
|
CP0444014
|
N-[2-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]ethyl]benzamide
Show/Hide
|
C27H26N4O2
|
2
|
1 |
IC50 = 27600 nM
|
|
|
2 |
IC50 > 50000 nM
|
|
|
CP0422148
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-(pyridin-4-ylmethylamino)ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C26H27N5O
|
1
|
1 |
IC50 = 27800 nM
|
|
|
CP0471660
|
2-[2-[2-(benzenesulfonamido)ethyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C26H26N4O3S
|
1
|
1 |
IC50 = 28200 nM
|
|
|
CP0552399
|
2-[2-[2-(benzylamino)ethyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C27H28N4O
|
1
|
1 |
IC50 = 30700 nM
|
|
|
CP0422102
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-(pyridin-3-ylsulfonylamino)ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C25H25N5O3S
|
1
|
1 |
IC50 = 32000 nM
|
|
|
CP0565922
|
N-[2-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]ethyl]-2-pyridin-4-ylacetamide
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|
C27H27N5O2
|
1
|
1 |
IC50 = 42300 nM
|
|
|