Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
 Cell Line Info 
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT03373 , Gamma-aminobutyric acid receptor subunit alpha-3
 Protein Info 
Gene Name GABRA3
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID P34903
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006
 Cell Line Info 
 Protein ID: PT03373
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0000200
 Compound Info 
ethyl 8-ethynyl-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate
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C17H15N3O3
  1
1
Ki = 25.8 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0008001
 Compound Info 
ethyl 12-ethynyl-9-phenyl-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(10),3,5,8,11,13-hexaene-5-carboxylate
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C22H17N3O2
  1
1
Ki = 96 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002342
 Compound Info 
3-({12-ethynyl-9-phenyl-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,8,10,12-hexaen-5-yl}carbonyloxy)propyl 12-ethynyl-9-phenyl-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(10),3,5,8,11,13-hexaene-5-carboxylate
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C43H30N6O4
  1
1
Ki = 272 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0002647
 Compound Info 
3-({12-ethynyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,10,12-pentaen-5-yl}carbonyloxy)propyl 12-ethynyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(10),3,5,11,13-pentaene-5-carboxylate
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C33H26N6O6
  1
1
Ki = 858 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0008002
 Compound Info 
XLi374, 5
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C32H24N6O7
  1
1
Ki = 1864 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0008003
 Compound Info 
5-({12-ethynyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,10,12-pentaen-5-yl}carbonyloxy)pentyl 12-ethynyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(10),3,5,11,13-pentaene-5-carboxylate
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C35H30N6O6
  1
1
Ki = 2666 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0008395
 Compound Info 
3-({12-ethyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,10,12-pentaen-5-yl}carbonyloxy)propyl 12-ethyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(10),3,5,11,13-pentaene-5-carboxylate
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C33H34N6O6
  1
1
Ki = 8545 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS