| Compound ID |
Compound Name |
Compound Formula |
|
CP0068632
|
5-cyclohexylpentyl N-[(2S,3R)-2-methyl-4-oxooxetan-3-yl]carbamate
Show/Hide
|
C16H27NO4
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0152909
|
[(2S)-nonan-2-yl] N-[(2S,3R)-2-methyl-4-oxooxetan-3-yl]carbamate
Show/Hide
|
C14H25NO4
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0410125
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(4-methylsulfonylphenoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C22H32N2O6S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0575428
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(2-methylsulfonylphenoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C22H32N2O6S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0068505
|
(4-phenylphenyl)methyl N-[(2S,3R)-2-methyl-4-oxooxetan-3-yl]carbamate
Show/Hide
|
C18H17NO4
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0092310
|
5-phenylpentyl N-[(2S,3R)-2-methyl-4-oxooxetan-3-yl]carbamate
Show/Hide
|
C16H21NO4
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0351079
|
(4-butylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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|
C15H20N2O3
|
2
|
| 1 |
IC50 = 7 nM
|
|
|
| 2 |
IC50 = 23 nM
|
|
|
|
CP0567192
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(3-methylsulfonylphenoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C22H32N2O6S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0078765
|
(4-cyclohexylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C17H22N2O3
|
2
|
| 1 |
IC50 = 12 nM
|
|
|
| 2 |
IC50 = 41 nM
|
|
|
|
CP0417224
|
4-cyclohexylbutyl N-[(3S)-1-methoxy-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H26N2O4
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0968803
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-(ethoxymethyl)phenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C21H29N3O4S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0410124
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(4-nitrophenoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C21H29N3O6
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0516034
|
methyl 4-[(2S,3S)-3-(4-cyclohexylbutoxycarbonylamino)-2-methyl-4-oxoazetidin-1-yl]oxybenzoate
Show/Hide
|
C23H32N2O6
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0966515
|
(1R,3r,5S)-3-((5-Butylpyrazin-2-yl)oxy)-8-((3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C20H29N5O3S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0969760
|
(1R,3r,5s)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-hexylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C24H35N3O3S
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0092309
|
3-phenylmethoxypropyl N-[(2S,3R)-2-methyl-4-oxooxetan-3-yl]carbamate
Show/Hide
|
C15H19NO5
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0516031
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(4-methylphenoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C22H32N2O4
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0758513
|
(2,2-Difluoro-1,3-benzodioxol-5-yl)-methyl-N-[(S)-2-oxoazetidin-3-yl]-carbamate
Show/Hide
|
C12H10F2N2O5
|
2
|
| 1 |
IC50 = 22 nM
|
|
|
| 2 |
IC50 = 85 nM
|
|
|
|
CP0457682
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-phenoxyazetidin-3-yl]carbamate
Show/Hide
|
C21H30N2O4
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0962020
|
(1R,3r,5S)-3-(4-Butylphenoxy)-8-((3,5-dimethyl-1H-pyrazol-4-yl)-suffonyl)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C22H31N3O3S
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0101729
|
4-cyclohexylbutyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C14H24N2O3
|
2
|
| 1 |
IC50 = 27 nM
|
|
|
| 2 |
IC50 = 73 nM
|
|
|
|
CP0516033
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-[4-(trifluoromethyl)phenoxy]azetidin-3-yl]carbamate
Show/Hide
|
C22H29F3N2O4
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0561077
|
4-cyclopentylbutyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C13H22N2O3
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0911958
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sufonyl)-3-(p-tolyloxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H25N3O3S
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0354758
|
octyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C12H22N2O3
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0457681
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-(4-phenylphenoxy)azetidin-3-yl]carbamate
Show/Hide
|
C27H34N2O4
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0915335
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-((5-(ethoxymethyl)pyrazin-2-yl)oxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H27N5O4S
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0474611
|
3-cyclohexylpropyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C13H22N2O3
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0264214
|
(4-propoxyphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C14H18N2O4
|
2
|
| 1 |
IC50 = 48 nM
|
|
|
| 2 |
IC50 = 250 nM
|
|
|
|
CP0569046
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-(4-phenoxyphenoxy)azetidin-3-yl]carbamate
Show/Hide
|
C27H34N2O5
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0531391
|
5-cyclohexylpentyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H26N2O3
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0447286
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(3-methylsulfonylpropoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C19H34N2O6S
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0955689
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-ethylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C20H27N3O3S
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0404336
|
(4-propylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C14H18N2O3
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0547379
|
4-cyclohexylbutyl N-[(3R)-1-methoxy-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H26N2O4
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0479726
|
4-cyclohexylbutyl N-[(2S,3S)-1-methoxy-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C16H28N2O4
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0946594
|
(4-Cyclopentylphenyl)-methyl-N-[(S)-2-oxoazetidin-3-yl]-carbamate
Show/Hide
|
C16H20N2O3
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0564155
|
4-[4-(trifluoromethyl)phenyl]butyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H17F3N2O3
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0549002
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-(4-oxopentoxy)azetidin-3-yl]carbamate
Show/Hide
|
C20H34N2O5
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0101728
|
4-(4,4-difluorocyclohexyl)butyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C14H22F2N2O3
|
2
|
| 1 |
IC50 = 76 nM
|
|
|
| 2 |
IC50 = 330 nM
|
|
|
|
CP0570195
|
4-cyclohexylbutyl N-[(2S,3S)-1-(3-methoxypropoxy)-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C19H34N2O5
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0955688
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-phenoxy-8-azabicyclo[3.2.1]octane
Show/Hide
|
C18H23N3O3S
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0954093
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-isopentylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C23H33N3O3S
|
1
|
| 1 |
IC50 = 114 nM
|
|
|
|
CP0490428
|
heptyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C11H20N2O3
|
1
|
| 1 |
IC50 = 122 nM
|
|
|
|
CP0538422
|
2,3-dihydro-1H-inden-5-ylmethyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C14H16N2O3
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0399845
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-propoxyazetidin-3-yl]carbamate
Show/Hide
|
C18H32N2O4
|
1
|
| 1 |
IC50 = 133 nM
|
|
|
|
CP0510867
|
5,6,7,8-tetrahydronaphthalen-2-ylmethyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H18N2O3
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0968799
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-fluorophenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C18H22FN3O3S
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0531390
|
(4-ethylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C13H16N2O3
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0970032
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(pyridin-2-yloxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C17H22N4O3S
|
1
|
| 1 |
IC50 = 162 nM
|
|
|
|
CP0397834
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-(3-methylsulfanylpropoxy)-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C19H34N2O4S
|
1
|
| 1 |
IC50 = 167 nM
|
|
|
|
CP0966514
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrozol-4-yl)sulfonyl)-3-(4-methoxyphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H25N3O4S
|
1
|
| 1 |
IC50 = 175 nM
|
|
|
|
CP0454507
|
4-cyclohexylbutyl N-[(2S,3S)-1-(2-ethoxyethoxy)-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C19H34N2O5
|
1
|
| 1 |
IC50 = 187 nM
|
|
|
|
CP0965877
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-(trifluoromethyl)phenoxy)-8-azabicyclo[3.2.1]octone
Show/Hide
|
C19H22F3N3O3S
|
1
|
| 1 |
IC50 = 212 nM
|
|
|
|
CP0510870
|
4-(4-ethylphenyl)butyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C16H22N2O3
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0970031
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(pyrazin-2-yloxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C16H21N5O3S
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0564153
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H26N2O3
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0940942
|
(1R,3r,55)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sufonyl)-3-(o-tolyloxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H25N3O3S
|
1
|
| 1 |
IC50 = 291 nM
|
|
|
|
CP0490429
|
5-phenylpentyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H20N2O3
|
1
|
| 1 |
IC50 = 298 nM
|
|
|
|
CP0468347
|
(4-tert-butylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C15H20N2O3
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0468349
|
(4-butylcyclohexyl) N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C14H24N2O3
|
1
|
| 1 |
IC50 = 323 nM
|
|
|
|
CP0542277
|
2-[1-[(5-methyl-3-propyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
Show/Hide
|
C16H23N5O3S
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0337327
|
N-[(3S)-2-oxoazetidin-3-yl]nonanamide
Show/Hide
|
C12H22N2O2
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0940913
|
(1R,3r,5S)-9-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(pyrazin-2-yloxy)-9-azabicyclo[3.3.1]nonane
Show/Hide
|
C17H23N5O3S
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0560461
|
4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-pentoxyazetidin-3-yl]carbamate
Show/Hide
|
C20H36N2O4
|
1
|
| 1 |
IC50 = 387 nM
|
|
|
|
CP0968801
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-propoxyphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C21H29N3O4S
|
1
|
| 1 |
IC50 = 450 nM
|
|
|
|
CP0510869
|
(4-phenylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
|
C17H16N2O3
|
1
|
| 1 |
IC50 = 513 nM
|
|
|
|
CP0900672
|
4-(4-Methoxyphenyl)-butyl-N-[(S)-2-oxoazetidin-3-yl]-carbamate
Show/Hide
|
C15H20N2O4
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0962019
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sufonyl)-3-(m-tolyloxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H25N3O3S
|
1
|
| 1 |
IC50 = 614 nM
|
|
|
|
CP0575530
|
2-[1-[(3-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
Show/Hide
|
C15H21N5O3S
|
1
|
| 1 |
IC50 = 620 nM
|
|
|
|
CP0572980
|
2-[1-[(5-methyl-3-propan-2-yl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
Show/Hide
|
C16H23N5O3S
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0964592
|
(1R,3s,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)suIfonyl)-3-phenoxy-8-azabicyclo[3.2.1]octane
Show/Hide
|
C18H23N3O3S
|
1
|
| 1 |
IC50 = 655 nM
|
|
|
|
CP0956201
|
(1R,5S,9s)-3-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-9-(pyrazin-2-yloxy)-3-azabicyclo[3.3.1]nonane
Show/Hide
|
C17H23N5O3S
|
1
|
| 1 |
IC50 = 690 nM
|
|
|
|
CP0967231
|
(1R,3r,5S)-8-(3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-isopropylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C21H29N3O3S
|
1
|
| 1 |
IC50 = 744 nM
|
|
|
|
CP0970033
|
(1R,3r,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(4-ethynylphenoxy)-8-azabicyclo[3.2.1]octane
Show/Hide
|
C19H22N4O3S
|
1
|
| 1 |
IC50 = 757 nM
|
|
|
|
CP0527627
|
2-[1-[(3-tert-butyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
Show/Hide
|
C17H25N5O3S
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0548330
|
2-[1-[(3-butyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
Show/Hide
|
C17H25N5O3S
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0490427
|
(4-methylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C12H14N2O3
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1
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| 1 |
IC50 = 1040 nM
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CP0572981
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2-[1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
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C14H19N5O3S
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1
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| 1 |
IC50 = 1090 nM
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CP0474614
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4-phenylbutyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C14H18N2O3
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1
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| 1 |
IC50 = 1110 nM
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CP0544152
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2-[1-[(3,5-diethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl]oxypyrazine
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C16H23N5O3S
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1
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| 1 |
IC50 = 1110 nM
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CP0535866
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4-cyclohexylbutyl N-[(2S,3S)-2-methyl-4-oxo-1-(4-phenylbutoxy)azetidin-3-yl]carbamate
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C25H38N2O4
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1
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| 1 |
IC50 = 1240 nM
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CP0490430
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2-(cyclohexylmethoxy)ethyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C13H22N2O4
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1
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| 1 |
IC50 = 1280 nM
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CP0900671
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(4-Tetrahydropyran-4-yl-phenyl)-methyl-N-[(S)-2-oxoazetidin-3-yl]-carbamate
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C16H20N2O4
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1
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| 1 |
IC50 = 1370 nM
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CP0456860
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[(Z)-4-phenylbut-3-enyl] N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C14H16N2O3
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1
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| 1 |
IC50 = 1510 nM
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CP0468348
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(3-cyclohexylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C17H22N2O3
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1
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| 1 |
IC50 = 1720 nM
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CP0564154
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[4-(1,3-oxazol-4-yl)phenyl]methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C14H13N3O4
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1
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| 1 |
IC50 = 1880 nM
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CP0465789
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4-cyclohexylbutyl N-[(3S)-1-methyl-2-oxoazetidin-3-yl]carbamate
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C15H26N2O3
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1
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| 1 |
IC50 = 1983 nM
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CP0490426
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(4-cyclohexyloxyphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C17H22N2O4
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1
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| 1 |
IC50 = 2070 nM
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CP0538421
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1,3-benzodioxol-5-ylmethyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C12H12N2O5
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1
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| 1 |
IC50 = 2190 nM
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CP0548739
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4-cyclohexylbutyl N-[(2S,3S)-1-heptoxy-2-methyl-4-oxoazetidin-3-yl]carbamate
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C22H40N2O4
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1
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| 1 |
IC50 = 2230 nM
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CP0958416
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(1R,5S,7s)-9-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-7-(pyrazin-2-yloxy)-3-oxa-9-azabicyclo[3.3.1]nonane
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C16H21N5O4S
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1
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| 1 |
IC50 = 2330 nM
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CP0538423
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3-cyclohexyloxypropyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C13H22N2O4
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1
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| 1 |
IC50 = 2670 nM
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CP0424845
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[(E)-4-phenylbut-3-enyl] N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C14H16N2O3
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1
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| 1 |
IC50 = 2890 nM
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CP0479728
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4-cyclohexylbutyl N-[(2S,3S)-1-cyclohexyloxy-2-methyl-4-oxoazetidin-3-yl]carbamate
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C21H36N2O4
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1
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| 1 |
IC50 = 3010 nM
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CP0510866
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4-cyclohexylbutyl N-[(3R)-2-oxoazetidin-3-yl]carbamate
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C14H24N2O3
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1
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| 1 |
IC50 = 3110 nM
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CP0578832
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2-[1-[[5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]sulfonyl]piperidin-4-yl]oxypyrazine
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C14H16F3N5O3S
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1
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| 1 |
IC50 = 3290 nM
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CP0535864
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4-cyclohexylbutyl N-[(2S,3S)-1-(4-cyclohexylbutoxy)-2-methyl-4-oxoazetidin-3-yl]carbamate
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C25H44N2O4
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1
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| 1 |
IC50 = 3470 nM
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CP0578831
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N,3,5-trimethyl-N-(3-pyrazin-2-yloxypropyl)-1H-pyrazole-4-sulfonamide
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C13H19N5O3S
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1
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| 1 |
IC50 = 4290 nM
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CP0474610
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1-(4-cyclohexylphenyl)ethyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C18H24N2O3
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1
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| 1 |
IC50 = 4470 nM
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CP0534451
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2-[1-(2,6-dimethylphenyl)sulfonylpiperidin-4-yl]oxypyrazine
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C17H21N3O3S
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1
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| 1 |
IC50 = 4480 nM
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CP0569272
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4-cyclohexylbutyl N-[(2S,3R)-1-methoxy-2-methyl-4-oxoazetidin-3-yl]carbamate
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C16H28N2O4
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1
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| 1 |
IC50 = 5070 nM
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CP0547378
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methyl (3S)-3-(4-cyclohexylbutoxycarbonylamino)-2-oxoazetidine-1-carboxylate
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C16H26N2O5
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1
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| 1 |
IC50 = 7180 nM
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CP0237970
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6-(1-methylpiperidin-4-yl)-N-(2-methylpropyl)-2-oxo-1,3-benzoxazole-3-carboxamide
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C18H25N3O3
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1
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| 1 |
IC50 = 8000 nM
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CP0568136
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(4-pyridin-3-ylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C16H15N3O3
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1
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| 1 |
IC50 = 8110 nM
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CP0958417
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(1R,3s,5S)-8-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-(p-tolyloxy)-8-azabicyclo[3.2.1]octane
Show/Hide
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C19H25N3O3S
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1
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| 1 |
IC50 = 8710 nM
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CP0490431
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4-(oxan-4-yl)butyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
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C13H22N2O4
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1
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| 1 |
IC50 = 9510 nM
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CP0958418
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(1R,3s,5S)-3-(4-Butylphenoxy)-8-((3,5-dimethyl-1H-pyrazol-4-yl)-sulfonyl)-8-azabicyclo[3.2.1]octane
Show/Hide
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C22H31N3O3S
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1
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| 1 |
IC50 = 10260 nM
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CP0510868
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(2-cyclohexylphenyl)methyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
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C17H22N2O3
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1
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| 1 |
IC50 = 12830 nM
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CP0490424
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4-cyclohexylbutyl N-[(2S,3R)-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C15H26N2O3
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1
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| 1 |
IC50 = 12910 nM
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CP0902758
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(1R,5S,8r)-3-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)-8-(pyrazin-2-yloxy)-3-azabicyclo[3.2.1]octane
Show/Hide
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C16H21N5O3S
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1
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| 1 |
IC50 = 15400 nM
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CP0548738
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4-cyclohexylbutyl N-[(2R,3R)-1-methoxy-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C16H28N2O4
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1
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| 1 |
IC50 = 15700 nM
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CP0531389
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4-cyclohexylbutyl N-[(3R)-2,2-dimethyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C16H28N2O3
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1
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| 1 |
IC50 = 17300 nM
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CP0424840
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4-cyclohexylbutyl N-[(3S)-2,2-dimethyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C16H28N2O3
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1
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| 1 |
IC50 = 25420 nM
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CP0536200
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4-cyclohexylbutyl N-[(2R,3R)-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C15H26N2O3
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1
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| 1 |
IC50 = 29360 nM
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CP0404337
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4-pyridin-2-ylbutyl N-[(3S)-2-oxoazetidin-3-yl]carbamate
Show/Hide
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C13H17N3O3
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1
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| 1 |
IC50 = 30650 nM
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CP0417113
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4-cyclohexylbutyl N-[(2S,3S)-1-hydroxy-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C15H26N2O4
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1
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| 1 |
IC50 = 47690 nM
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CP0404334
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4-cyclohexylbutyl N-[(2R,3S)-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C15H26N2O3
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1
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| 1 |
IC50 > 50000 nM
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CP0411205
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4-cyclohexylbutyl N-[(2R,3S)-1-methoxy-2-methyl-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C16H28N2O4
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1
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| 1 |
IC50 > 50000 nM
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CP0479727
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4-cyclohexylbutyl N-[(2S,3S)-2-methyl-1-[(2-methylpropan-2-yl)oxy]-4-oxoazetidin-3-yl]carbamate
Show/Hide
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C19H34N2O4
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1
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| 1 |
IC50 > 50000 nM
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CP0548737
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4-cyclohexylbutyl N-[(3S)-1-acetyl-2-oxoazetidin-3-yl]carbamate
Show/Hide
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C16H26N2O4
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1
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| 1 |
IC50 > 50000 nM
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