Compound ID |
Compound Name |
Compound Formula |
CP0064604
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-6-amino-2-[[(2S)-4-amino-2-[[(2S)-4-carboxy-2-[[(2S)-3-(4-hydroxyphenyl)-2-[[(2S)-4-methyl-2-[[(2S)-5-oxopyrrolidine-2-carbonyl]amino]pentanoyl]amino]propanoyl]amino]butanoyl]amino]-4-oxobutanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
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C78H121N21O20
|
2
|
1 |
EC50 = 110 nM
|
|
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2 |
Ki = 4.9 nM
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|
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CP0287588
|
(S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)-N-(4-hydroxyphenethyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
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C39H66N12O8
|
2
|
1 |
EC50 = 480 nM
|
|
|
2 |
Ki = 8.8 nM
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|
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CP0422801
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(S)-2-((2S,3S)-2-(2-((S)-1-((S)-6-amino-2-((S)-2,6-diaminohexanamido)hexanoyl)-N-(4-hydroxyphenethyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
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C39H66N8O8
|
2
|
1 |
EC50 = 590 nM
|
|
|
2 |
Ki = 4.3 nM
|
|
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CP0329956
|
(S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2,6-diaminohexanamido)-5-guanidinopentanoyl)-N-(4-hydroxyphenethyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
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|
C39H66N10O8
|
2
|
1 |
EC50 = 690 nM
|
|
|
2 |
Ki = 4.4 nM
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|
|
CP0240966
|
(S)-2-((2S,3S)-2-(2-((S)-1-((S)-6-amino-2-((S)-2-amino-5-guanidinopentanamido)hexanoyl)-N-(4-hydroxyphenethyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N10O8
|
2
|
1 |
EC50 = 840 nM
|
|
|
2 |
Ki = 6.7 nM
|
|
|
CP0877791
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxycyclohexa-1,3-dienyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
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|
C38H66N12O8
|
1
|
1 |
Kd = 1.2 nM
|
|
|
CP0425790
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-3-amino-6-guanidinohexanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N12O8
|
1
|
1 |
Ki = 0.61 nM
|
|
|
CP0456304
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-(2-(4-aminobutylamino)acetamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C38H64N8O8
|
1
|
1 |
Ki = 0.74 nM
|
|
|
CP0405472
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C38H64N12O8
|
2
|
1 |
Ki = 0.7413 nM
|
|
|
2 |
Ki = 1.2 nM
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|
|
CP0444542
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-[[amino-[2-[2-[2-[6-[(2E)-3,3-dimethyl-2-[(2E,4E)-5-(1,3,3-trimethylindol-1-ium-2-yl)penta-2,4-dienylidene]indol-1-yl]hexanoylamino]ethoxy]ethoxy]ethylcarbamoylamino]methylidene]amino]pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid;2,2,2-trifluoroacetate;2,2,2-trifluoroacetic acid
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|
C85H118F12N16O20
|
1
|
1 |
Ki = 0.955 nM
|
|
|
CP0424109
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-[[amino-[4-[6-[(2E)-3,3-dimethyl-2-[(2E,4E)-5-(1,3,3-trimethylindol-1-ium-2-yl)penta-2,4-dienylidene]indol-1-yl]hexanoylamino]butylcarbamoylamino]methylidene]amino]pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid;2,2,2-trifluoroacetate;2,2,2-trifluoroacetic acid
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|
C81H113F9N16O16
|
1
|
1 |
Ki = 1.202 nM
|
|
|
CP0444541
|
4-[2-[(1E,3E,5E)-5-[1-[6-[2-[2-[2-[[N'-[(4S)-4-amino-5-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-3-methylbutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-oxopentyl]carbamimidoyl]carbamoylamino]ethoxy]ethoxy]ethylamino]-6-oxohexyl]-3,3-dimethyl-5-sulfoindol-2-ylidene]penta-1,3-dienyl]-3,3-dimethylindol-1-ium-1-yl]butane-1-sulfonate;2,2,2-trifluoroacetic acid
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|
C84H122F6N16O22S2
|
1
|
1 |
Ki = 3.467 nM
|
|
|
CP0444540
|
4-[2-[(1E,3E,5E)-5-[1-[6-[4-[[N'-[(4S)-4-amino-5-[[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-3-methylbutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-oxopentyl]carbamimidoyl]carbamoylamino]butylamino]-6-oxohexyl]-3,3-dimethyl-5-sulfoindol-2-ylidene]penta-1,3-dienyl]-3,3-dimethylindol-1-ium-1-yl]butane-1-sulfonate;2,2,2-trifluoroacetic acid
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|
C82H118F6N16O20S2
|
1
|
1 |
Ki = 3.981 nM
|
|
|
CP0478019
|
(S)-2-((3S,4S)-3-((S)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-4-methylhexanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N12O8
|
1
|
1 |
Ki = 5.4 nM
|
|
|
CP0520992
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((R)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C38H64N12O8
|
1
|
1 |
Ki = 5.4 nM
|
|
|
CP0232097
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2,6-diaminohexanamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C38H64N8O8
|
1
|
1 |
Ki = 6.1 nM
|
|
|
CP0476569
|
4-[(2Z)-2-[(2E,4E)-5-[1-[6-[2-[2-[2-[[N'-[(4S)-4-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-[(2S)-2-[[(2S)-1-[[(2S,3S)-1-[[(1S)-1-carboxy-3-methylbutyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxopentyl]carbamimidoyl]carbamoylamino]ethoxy]ethoxy]ethylamino]-6-oxohexyl]-3,3-dimethylindol-1-ium-2-yl]penta-2,4-dienylidene]-3,3-dimethylindol-1-yl]butane-1-sulfonate;2,2,2-trifluoroacetic acid
Show/Hide
|
C86H123F9N16O21S
|
1
|
1 |
Ki = 7.244 nM
|
|
|
CP0451818
|
(2S)-2-[[(2S,3S)-2-[[(2R,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-hydroxyphenyl)oxolane-3-carbonyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C40H66N12O9
|
1
|
1 |
Ki = 12 nM
|
|
|
CP0451820
|
(2S)-2-[[(2S,3S)-2-[[3-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-bromophenyl)oxolane-3-carbonyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C40H65BrN12O8
|
1
|
1 |
Ki = 12 nM
|
|
|
CP0478016
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-3-((S)-2-amino-5-guanidinopentanamido)-6-guanidinohexanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N12O8
|
1
|
1 |
Ki = 16 nM
|
|
|
CP0456309
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-4-(4-hydroxyphenyl)butanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N12O8
|
1
|
1 |
Ki = 17 nM
|
|
|
CP0520993
|
(S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)-N-phenethylpyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N12O7
|
1
|
1 |
Ki = 20 nM
|
|
|
CP0495431
|
(S)-2-((2S,3S)-2-((S)-2-((S)-1-(2-((S)-2,6-diamino-N-(4-aminobutyl)hexanamido)acetyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C38H64N8O8
|
1
|
1 |
Ki = 21 nM
|
|
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CP0456307
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C35H57N9O8
|
1
|
1 |
Ki = 24 nM
|
|
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CP0456306
|
(S)-3-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-5-methylhexanoic acid
Show/Hide
|
C39H66N12O8
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1
|
1 |
Ki = 25 nM
|
|
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CP0466985
|
(2S)-2-[[2-[[(2S,3R)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-hydroxyphenyl)oxolane-3-carbonyl]amino]acetyl]amino]-4-methylpentanoic acid
Show/Hide
|
C36H58N12O9
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1
|
1 |
Ki = 29 nM
|
|
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CP0921562
|
(S)-2-((S)-2-((S)-3-((S)-1-((S)-5-guanidino-2-((S)-5-guanidino-2-methylpentanamido)pentanoyl)pyrrolidine-2-carboxamido)-4-(naphthalen-1-yl)but-1-en-2-ylamino)-4,4-dimethylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C45H71N11O6
|
1
|
1 |
Ki = 34 nM
|
|
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CP0425793
|
(S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)-N-(4-methoxyphenethyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C40H68N12O8
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1
|
1 |
Ki = 38 nM
|
|
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CP0425794
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(S)-2-((2S,3S)-2-((S)-3-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-4-(4-hydroxyphenyl)butanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C39H66N12O8
|
1
|
1 |
Ki = 44 nM
|
|
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CP0478017
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(S)-2-((2S,3S)-2-((S)-2-((S)-1-((R)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
|
C38H64N12O8
|
1
|
1 |
Ki = 51 nM
|
|
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CP0456305
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C35H57N9O8
|
1
|
1 |
Ki = 56 nM
|
|
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CP0441155
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
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|
C36H62N12O8
|
1
|
1 |
Ki = 63 nM
|
|
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CP0503235
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2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidino-pentanoylamino)-5-guanidino-pentanoyl]-pyrrolidine-2-carbonyl}-amino)-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-4-methyl-pentanoic acid
Show/Hide
|
C35H58N12O8
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1
|
1 |
Ki = 63 nM
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|
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CP0376947
|
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-6-amino-2-[[(2S)-2,6-diaminohexanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-bromophenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C38H63BrN8O7
|
1
|
1 |
Ki = 69 nM
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|
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CP0495432
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
|
C32H60N12O7
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1
|
1 |
Ki = 83 nM
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|
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CP0456308
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(S)-2-((2S,3S)-2-(2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)-N-(2-(pyridin-2-yl)ethyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
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C38H65N13O7
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1
|
1 |
Ki = 100 nM
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CP0530845
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(2S)-2-[[(2S,3S)-2-[[(2R,3S)-2-(4-bromophenyl)-3-[[(2S)-1-[(2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]oxolane-3-carbonyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
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C40H65BrN10O8
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1
|
1 |
Ki = 110 nM
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|
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CP0478018
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(S)-2-((2S,3S)-2-((R)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
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C38H64N12O8
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1
|
1 |
Ki = 140 nM
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|
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CP0542434
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(2S)-2-[[(2S,3S)-2-[[(2R,3S)-3-[[(2S)-1-[(2S)-6-amino-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-bromophenyl)oxolane-3-carbonyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
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C40H65BrN10O8
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1
|
1 |
Ki = 147 nM
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|
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CP0507780
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(S)-2-((2S,3S)-2-((S)-2-(2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidin-2-yl)acetamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
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C39H66N12O8
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1
|
1 |
Ki = 210 nM
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|
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CP0530846
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(2S)-2-[[(2S,3S)-2-[[(2R,3S)-3-[[(2S)-1-[(2S)-6-amino-2-[[(2S)-2,6-diaminohexanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-bromophenyl)oxolane-3-carbonyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
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C40H65BrN8O8
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1
|
1 |
Ki = 227 nM
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|
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CP0456310
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(S)-2-((2S,3S)-2-((S)-2-((R)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
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C38H64N12O8
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1
|
1 |
Ki = 590 nM
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|
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CP0451821
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(2S)-2-[[(2S,3S)-2-[[(2R,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-bromophenyl)oxolane-3-carbonyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
Show/Hide
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C40H65BrN12O8
|
1
|
1 |
Ki = 615 nM
|
|
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CP0441156
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(S)-2-((2R,3S)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
Show/Hide
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C38H64N12O8
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1
|
1 |
Ki = 690 nM
|
|
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CP0466984
|
(2S)-2-[[2-[[(2R,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-2-(4-hydroxyphenyl)oxolane-3-carbonyl]amino]acetyl]amino]-4-methylpentanoic acid
Show/Hide
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C36H58N12O9
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1
|
1 |
Ki = 700 nM
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|
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CP0466986
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(2S)-2-[[(2S,3S)-2-[[(2R)-2-[[(2S)-1-[(2S)-6-amino-2-[[(2S)-2,6-diaminohexanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-bromophenyl)propanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoic acid
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C38H63BrN8O7
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1
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1 |
Ki = 873 nM
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CP0522126
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(S)-2-((2S,3S)-2-(2-((S)-1-((S)-6-amino-2-((S)-2,6-diaminohexanamido)hexanoyl)-N-(4-hydroxybenzyl)pyrrolidine-2-carboxamido)acetamido)-3-methylpentanamido)-4-methylpentanoic acid
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C38H64N8O8
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1
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1 |
Ki = 1000 nM
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CP0456311
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(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]propanoic acid
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C35H58N12O8
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1
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1 |
Ki = 1300 nM
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CP0456312
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2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)-2,6-diaminohexanamido)hexanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-N-isobutyl-3-methylpentanamido)acetic acid
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C38H64N8O8
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1
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1 |
Ki = 1600 nM
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CP0511311
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(R)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino-5-guanidinopentanamido)-5-guanidinopentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid
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C38H64N12O8
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1
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1 |
Ki = 3700 nM
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