| Compound ID |
Compound Name |
Compound Formula |
|
CP0562139
|
2,4-difluoro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]benzamide
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|
C19H18F3N3O
|
1
|
| 1 |
IC50 = 4.67 nM
|
|
|
|
CP0423482
|
4-fluoro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]benzamide
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|
C19H19F2N3O
|
1
|
| 1 |
IC50 = 6.36 nM
|
|
|
|
CP0138764
|
2,4,6-trifluoro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]benzamide
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|
C19H17F4N3O
|
1
|
| 1 |
IC50 = 19.55 nM
|
|
|
|
CP0423571
|
4-chloro-2-fluoro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]benzamide
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|
C19H18ClF2N3O
|
1
|
| 1 |
IC50 = 23.41 nM
|
|
|
|
CP0557648
|
5-fluoro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]pyridine-2-carboxamide
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|
C18H18F2N4O
|
1
|
| 1 |
IC50 = 24.32 nM
|
|
|
|
CP0423483
|
4-chloro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]benzamide
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|
C19H19ClFN3O
|
1
|
| 1 |
IC50 = 29.35 nM
|
|
|
|
CP0357652
|
COL-144
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|
C19H18F3N3O2
|
1
|
| 1 |
IC50 = 87.84 nM
|
|
|
|
CP0512435
|
5-chloro-N-[6-[fluoro-(1-methylpiperidin-4-ylidene)methyl]pyridin-2-yl]pyridine-2-carboxamide
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|
C18H18ClFN4O
|
1
|
| 1 |
IC50 = 160.9 nM
|
|
|
|
CP0547508
|
N-[6-[(1-ethylpiperidin-4-ylidene)-fluoromethyl]pyridin-2-yl]-2,4,6-trifluorobenzamide
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|
C20H19F4N3O
|
1
|
| 1 |
IC50 = 178.05 nM
|
|
|
|
CP0570281
|
N-[6-[(1-cyclopropylpiperidin-4-ylidene)-fluoromethyl]pyridin-2-yl]-2,4,6-trifluorobenzamide
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|
C21H19F4N3O
|
1
|
| 1 |
IC50 = 570.5 nM
|
|
|
|
CP0514917
|
N-[6-[[1-(difluoromethyl)piperidin-4-ylidene]-fluoromethyl]pyridin-2-yl]-2,4,6-trifluorobenzamide
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|
C19H15F6N3O
|
1
|
| 1 |
IC50 = 813.4 nM
|
|
|
|
CP0423480
|
2,4,6-trifluoro-N-[6-[fluoro-[1-(trifluoromethyl)piperidin-4-ylidene]methyl]pyridin-2-yl]benzamide
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|
C19H14F7N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0847634
|
(E)-N-[4'-(Phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-N-pyridin-3-ylmethyl-acrylamide TFA
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|
C39H36F3N3O3
|
1
|
| 1 |
Ki < 1000 nM
|
|
|
|
CP0853819
|
(E)-N-(2-Dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-3-phenyl-acrylamide TFA
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|
C37H40F3N3O3
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
|
CP0861232
|
3-Cyclopentyl-N-(2-dimethylamino-ethyl)-N-[4'-(phenethylamino-methyl)-biphenyl-4-ylmethyl]-propionamide with di TFA
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|
C38H47F6N3O5
|
1
|
| 1 |
Ki < 10000 nM
|
|
|
