| Compound ID |
Compound Name |
Compound Formula |
|
CP0400662
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((prop-2-ynyloxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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|
C25H29ClO6
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0198642
|
(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO6
|
2
|
| 1 |
IC50 = 0.8 nM
|
|
|
| 2 |
IC50 = 6.7 nM
|
|
|
|
CP0238397
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-(methoxymethyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C23H29ClO6
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0482964
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethoxybenzyl)-2-(2-methoxyethyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C24H31ClO7
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0478241
|
4-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-methylsulfanyloxan-2-yl]phenyl]methyl]phenoxy]-N-(1-hydroxy-2-methylpropan-2-yl)butanamide
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|
C27H36ClNO7S
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0398959
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-hydroxyethoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H31ClO7
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0389735
|
US9688710, 132 N-(1-((2-(dimethylamino)ethyl)(methyl)amino)-2-methyl-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide
Show/Hide
|
C33H49N3O6S
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0438889
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-fluoroethoxy)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H30ClFO6
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0535547
|
US9688710, 146 (3R,4R,5S,6R)-2-(3-(4-(3-((3-(dimethylamino)-2,2-dimethylpropyl)amino)propoxy)benzyl)-4-methylphenyl)-6-(methylthio)tetrahydro-2H-pyran-3,4,5-triol
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|
C30H46N2O5S
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0073918
|
LP-802034
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|
C21H25ClO5S
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0417976
|
(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H25ClO5
|
1
|
| 1 |
IC50 = 1.9 nM
|
|
|
|
CP0492114
|
US9688710, 113 N-(2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylsulfinyl)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide
Show/Hide
|
C33H47N3O6S
|
1
|
| 1 |
IC50 = 1.9 nM
|
|
|
|
CP0486573
|
US8614195, 4
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|
C23H27Na2O10P
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0389733
|
US9688710, 124 4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)-N-(2-(4-methylpiperazin-1-yl)-2-oxoethyl)butanamide
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|
C31H43N3O6S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0389734
|
US9688710, 120 N-(2-methyl-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide
Show/Hide
|
C34H48N2O6S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0398977
|
US9688710, 135 (3R,4R,5S,6R)-2-(3-(4-(3-((1-hydroxy-2-methylpropan-2-yl)amino)propoxy)benzyl)-4-methylphenyl)-6-(methylthio)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C27H39NO6S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0457942
|
US9688710, 116 4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)-N-(1-(4-methylpiperazine-1-carbonyl)cyclopropyl)butanamide
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|
C33H45N3O6S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0492115
|
US9688710, 136 N-(1-((2-(dimethylamino)ethyl)amino)-2-methyl-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide
Show/Hide
|
C32H47N3O6S
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0501978
|
(2S,3R,4R,5S,6R)-2-(4-chloro-2-((2,2-difluoroethoxy)methyl)-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H29ClF2O6
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0409451
|
US9688710, 129 2-methyl-2-((4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butyl)amino)-1-(4-methylpiperazin-1-yl)propan-1-one
Show/Hide
|
C33H49N3O5S
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0492112
|
US9688710, 127 N-(2,2-dimethyl-3-(4-methylpiperazin-1-yl)-3-oxopropyl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide
Show/Hide
|
C34H49N3O6S
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0417974
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-methoxyethoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H33ClO7
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0437096
|
US9688710, 104 2,2-dimethyl-3-((4-(4-(2-methyl-5-((3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butyl)amino)propanamide
Show/Hide
|
C29H42N2O5S
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0492113
|
US9688710, 149 1-(1-hydroxy-2-methylpropan-2-yl)-3-(2-(4-(2-methyl-5-((3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)ethyl)urea
Show/Hide
|
C27H38N2O7S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0519595
|
US9688710, 147 N-(2-methyl-1-((1-methylpiperidin-4-yl)amino)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide
Show/Hide
|
C34H49N3O6S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0541795
|
US9688710, 45 N-(2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butanamide
Show/Hide
|
C33H47N3O7S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0476161
|
US9688710, 2 4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butanoic acid
Show/Hide
|
C23H27ClO7S
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0456487
|
US9688710, 37 2-methyl-2-(2-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)acetamido)propanamide
Show/Hide
|
C26H34N2O7S
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
|
CP0564205
|
(2S,3R,4R,5S,6R)-2-[7-[(4-ethylphenyl)methyl]-2,3-dihydro-1H-inden-5-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H30O5
|
1
|
| 1 |
IC50 = 5.6 nM
|
|
|
|
CP0400661
|
1-(5-chloro-4-(4-ethylbenzyl)-2-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2Hpyran-2-yl)benzyloxy)propan-2-one
Show/Hide
|
C25H31ClO7
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0475790
|
(1S,3'R,4'S,5'S,6'R)-5-chloro-6-(4-ethoxybenzyl)-6'-(hydroxymethyl)-3',4',5',6'-tetrahydro-3H-spiro[isobenzofuran-1,2'-pyran]-3',4',5'-triol
Show/Hide
|
C22H25ClO7
|
1
|
| 1 |
IC50 = 6.5 nM
|
|
|
|
CP0421707
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-(2-(prop-2-ynyloxy)ethyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C26H31ClO6
|
1
|
| 1 |
IC50 = 6.7 nM
|
|
|
|
CP0499717
|
3-(4-fluorophenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C21H23FO9
|
1
|
| 1 |
IC50 = 9.1 nM
|
|
|
|
CP0879630
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-fluoropropoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H32ClFO6
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0410170
|
3-(4-hydroxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C21H24O10
|
1
|
| 1 |
IC50 = 11.9 nM
|
|
|
|
CP0514559
|
(2S,3R,4R,5S,6R)-2-(2-(2-(allyloxy)ethyl)-4-chloro-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C26H33ClO6
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0476158
|
US9688710, 4 4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanoicacid
Show/Hide
|
C23H30O7S
|
1
|
| 1 |
IC50 = 14.5 nM
|
|
|
|
CP0467478
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2-hydroxypropoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H33ClO7
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0458478
|
3-(4-methylphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C22H26O9
|
1
|
| 1 |
IC50 = 18.2 nM
|
|
|
|
CP0417033
|
3-phenyl-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C21H24O9
|
1
|
| 1 |
IC50 = 19.8 nM
|
|
|
|
CP0410123
|
3-(4-methoxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C22H26O10
|
1
|
| 1 |
IC50 = 21.3 nM
|
|
|
|
CP0417032
|
3-(4-ethoxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C23H28O10
|
1
|
| 1 |
IC50 = 21.7 nM
|
|
|
|
CP0447285
|
3-(4-propoxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one
Show/Hide
|
C24H30O10
|
1
|
| 1 |
IC50 = 22.7 nM
|
|
|
|
CP0523299
|
US8614195, 2c
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|
C26H32O9
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0428912
|
(2S,3R,4R,5S)-2-[4-Chloro-3-(4-hydroxy-benzyl)-phenyl]-6-methoxy-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C19H21ClO6
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0383615
|
(2S,3R,4R,5S)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(2-hydroxyethoxy)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H27ClO7
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0469895
|
(2S,3R,4R,5S)-2-(4-Chloro-3-(4-(2-hydroxyethoxy)benzyl)phenyl)-6-methoxytetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C21H25ClO7
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0485773
|
(2S,3R,4R,5S)-2-{4-Chloro-3-[4-(2-methoxy-ethoxy)-benzyl]-phenyl}-6-methoxy-tetrahydropyran-3,4,5-triol
Show/Hide
|
C22H27ClO7
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0421706
|
(2S,3R,4R,5S,6R)-2-(2-(allyloxymethyl)-4-chloro-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H31ClO6
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0430170
|
(2S,3R,4R,5S)-2-(3-(4-Ethoxybenzyl)-4-methylphenyl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C22H28O6
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0428915
|
(2S,3R,4R,5S)-2-[4-Chloro-3-(4-ethoxy-benzyl)-phenyl]-6-ethoxy-tetrahydro-pyran-3,4,5-triol
Show/Hide
|
C22H27ClO6
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0050531
|
1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)-3-(4-hydroxyphenyl)propan-1-one
Show/Hide
|
C21H24O10
|
2
|
| 1 |
IC50 = 58.6 nM
|
|
|
| 2 |
IC50 = 67.3 nM
|
|
|
|
CP0516684
|
US8614195, 2e
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|
C28H36O9
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
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CP0409820
|
US8614195, 2a
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|
C27H32O9
|
1
|
| 1 |
IC50 = 97 nM
|
|
|
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CP0397185
|
[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]phenyl]-(4-ethoxyphenyl)methanone
Show/Hide
|
C21H23ClO7
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
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CP0482965
|
(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((3-hydroxypropoxy)methyl)phenyl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H33ClO7
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0443900
|
ethyl 1-(4-nitrophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
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|
C15H18N4O7
|
1
|
| 1 |
IC50 = 125.9 nM
|
|
|
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CP0438998
|
(2S,3R,4R,5S,6R)-2-(4-chloro-2-((2,2-difluoropropoxy)methyl)-5-(4-ethylbenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H31ClF2O6
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0388962
|
ethyl 1-phenyl-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C15H19N3O5
|
1
|
| 1 |
IC50 = 134.7 nM
|
|
|
|
CP0486577
|
US8614195, 2f
Show/Hide
|
C32H40O9
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0388961
|
ethyl 1-(2-bromophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C15H18BrN3O5
|
1
|
| 1 |
IC50 = 146.9 nM
|
|
|
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CP0461324
|
ethyl 1-(2,5-dimethoxyphenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
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|
C17H23N3O7
|
1
|
| 1 |
IC50 = 149.1 nM
|
|
|
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CP0373281
|
(2S,3R,4R,5S)-2-(4-Chloro-3-(4-(thiazol-2-yloxy)benzyl)phenyl)-6-methoxytetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C22H22ClNO6S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
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CP0433332
|
ethyl 1-[4-(trifluoromethoxy)phenyl]-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C16H18F3N3O6
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
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CP0481579
|
ethyl 1-(4-fluorophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C15H18FN3O5
|
1
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| 1 |
IC50 = 151.8 nM
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CP0432907
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ethyl 1-(4-methylphenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
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C16H21N3O5
|
1
|
| 1 |
IC50 = 163.2 nM
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CP0428914
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(2R,3S,4S,5R)-2-(4-Chloro-3-(4-((S)-1-methylpyrrolidin-3-yloxy)benzyl)phenyl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H30ClNO6
|
1
|
| 1 |
IC50 = 170 nM
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CP0510336
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(2S,3R,4R,5S,6R)-2-(4-chloro-5-(4-ethylbenzyl)-2-((2,2,2-trifluoroethoxy)methyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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C24H28ClF3O6
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1
|
| 1 |
IC50 = 170 nM
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CP0380691
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ethyl 1-(3-nitrophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
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C15H18N4O7
|
1
|
| 1 |
IC50 = 175 nM
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CP0494274
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(2S,3R,4R,5S)-2-(4-Chloro-3-(4-methoxyphenylthio)phenyl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C19H21ClO6S
|
1
|
| 1 |
IC50 = 180 nM
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CP0391838
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ethyl 1-[2-(trifluoromethyl)phenyl]-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
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C16H18F3N3O5
|
1
|
| 1 |
IC50 = 185.8 nM
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CP0390386
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US8614195, 2b
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C29H36O9
|
1
|
| 1 |
IC50 = 186 nM
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CP0404018
|
ethyl 1-(2,4-dichlorophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
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C15H17Cl2N3O5
|
1
|
| 1 |
IC50 = 190.3 nM
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CP0479096
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ethyl 1-(4-phenylphenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
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C21H23N3O5
|
1
|
| 1 |
IC50 = 214.2 nM
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CP0486653
|
ethyl 1-(2-methoxydibenzofuran-3-yl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
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C22H23N3O7
|
1
|
| 1 |
IC50 = 227 nM
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|
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CP0498753
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(3S,4R,5R,6S)-6-[4-Chloro-3-(4-ethoxy-benzyl)-phenyl]-tetrahydro-pyran-2,3,4,5-tetraol
Show/Hide
|
C20H23ClO6
|
1
|
| 1 |
IC50 = 280 nM
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|
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CP0486654
|
ethyl 1-(4-bromophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C15H18BrN3O5
|
1
|
| 1 |
IC50 = 311 nM
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|
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CP0421307
|
ethyl 1-(2-nitrophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C15H18N4O7
|
1
|
| 1 |
IC50 = 367 nM
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|
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CP0380689
|
ethyl 1-dibenzofuran-3-yl-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate
Show/Hide
|
C21H21N3O6
|
1
|
| 1 |
IC50 = 458 nM
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|
|
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CP0425062
|
US8614195, 2g
Show/Hide
|
C32H36O9
|
1
|
| 1 |
IC50 = 567 nM
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|
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CP0430167
|
(2S,3R,4R,5S)-2-(4-Chloro-3-(4-ethoxybenzyl)phenyl)-6-methoxy-2-methyltetrahydro-2Hpyran-3,4,5-triol
Show/Hide
|
C22H27ClO6
|
1
|
| 1 |
IC50 = 590 nM
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|
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CP0401579
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(2S,3R,4R,5R)-2-[4-Chloro-3-(4-ethoxy-benzyl)-phenyl]-5-fluoro-6-methoxy-tetrahydro-pyran-3,4-diol
Show/Hide
|
C21H24ClFO5
|
1
|
| 1 |
IC50 = 600 nM
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|
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CP0455320
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(3S,4R,5R,6S)-2-(benzyloxy)-6-(4-chloro-3-(4-ethoxybenzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C27H29ClO6
|
1
|
| 1 |
IC50 = 620 nM
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|
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CP0428913
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O-[4-[[2-chloro-5-[(2S,3R,4R,5S)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]phenyl]methyl]phenyl] N,N-dimethylcarbamothioate
Show/Hide
|
C22H26ClNO6S
|
1
|
| 1 |
IC50 = 740 nM
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|
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CP0430168
|
(2S,3R,4R,5S)-2-(3-(4-Ethoxybenzyl)phenyl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H26O6
|
1
|
| 1 |
IC50 = 1100 nM
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CP0494301
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(2S,3R,4R,5S)-2-(4-Chloro-3-(4-ethoxyphenoxy)phenyl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H23ClO7
|
1
|
| 1 |
IC50 = 2400 nM
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|
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CP0388374
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(2S,3R,4R,5S)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(2-(dimethylamino)ethoxy)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H32ClNO6
|
1
|
| 1 |
IC50 = 3600 nM
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|
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CP0397188
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(2S,3R,4R,5S)-2-(4'-Ethoxybiphenyl-4-yl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C20H24O6
|
1
|
| 1 |
IC50 = 4600 nM
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|
|
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CP0038281
|
3-phenyl-1-(2,4,6-trihydroxyphenyl)-1-propanone
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|
C15H14O4
|
1
|
| 1 |
IC50 = 14700 nM
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|
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CP0457680
|
3-(4-fluorophenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
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|
C15H13FO4
|
1
|
| 1 |
IC50 = 15800 nM
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CP0397833
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3-(4-propoxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
Show/Hide
|
C18H20O5
|
1
|
| 1 |
IC50 = 16400 nM
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|
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CP0441153
|
3-(4-ethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
Show/Hide
|
C17H18O5
|
1
|
| 1 |
IC50 = 16700 nM
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CP0410171
|
3-(4-methylphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
Show/Hide
|
C16H16O4
|
1
|
| 1 |
IC50 = 18000 nM
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CP0417031
|
4-METHOXYL-2',4',6'-TRIHYDROXYCHALCONE
Show/Hide
|
C16H14O5
|
1
|
| 1 |
IC50 = 18200 nM
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|
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CP0046374
|
3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
Show/Hide
|
C15H14O5
|
1
|
| 1 |
IC50 = 18300 nM
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|
|
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CP0417034
|
3-(4-methoxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one
Show/Hide
|
C16H16O5
|
1
|
| 1 |
IC50 = 18700 nM
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CP0458479
|
(E)-3-(4-phenylmethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one
Show/Hide
|
C22H18O5
|
1
|
| 1 |
IC50 = 22700 nM
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|
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CP0410169
|
4-BROMO-2',4',6'-TRIHYDROXYCHALCONE
Show/Hide
|
C15H11BrO4
|
1
|
| 1 |
IC50 = 23500 nM
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|
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CP0456990
|
(E)-3-(4-ethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one
Show/Hide
|
C17H16O5
|
1
|
| 1 |
IC50 = 26000 nM
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|
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CP0454506
|
(E)-3-(4-prop-2-enoxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one
Show/Hide
|
C18H16O5
|
1
|
| 1 |
IC50 = 26200 nM
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|
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CP0397186
|
(2R,3S,4S,5R)-2-(4-Chloro-3-(4-ethoxybenzyl)phenyl)-6-methoxytetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C21H25ClO6
|
1
|
| 1 |
IC50 > 30000 nM
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|
|
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CP0489561
|
(2S,3R,4S)-2-(4-Chloro-3-(4-ethoxybenzyl)phenyl)-6-methoxytetrahydro-2H-pyran-3,4-diol
Show/Hide
|
C21H25ClO5
|
1
|
| 1 |
IC50 > 30000 nM
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|
|
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CP0036249
|
(E)-3-Phenyl-1-(2,4,6-trihydroxy-phenyl)-propenone
Show/Hide
|
C15H12O4
|
1
|
| 1 |
IC50 = 33300 nM
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|
|
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CP0458476
|
(E)-3-(4-methylphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one
Show/Hide
|
C16H14O4
|
1
|
| 1 |
IC50 = 34100 nM
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|
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CP0458480
|
4-FLUORO-2',4',6'-TRIHYDROXYCHALCONE
Show/Hide
|
C15H11FO4
|
1
|
| 1 |
IC50 = 51700 nM
|
|
|
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CP0375036
|
US8614195, 3a
Show/Hide
|
C28H37O10P
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0429724
|
US8614195, 3
Show/Hide
|
C27H37O10P
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
