| Compound ID |
Compound Name |
Compound Formula |
|
CP0384519
|
US10131692, Compound 10
Show/Hide
|
C42H60ClN11O8S2
|
1
|
| 1 |
EC50 = 0.02 nM
|
|
|
|
CP0379479
|
(S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-10-(3-amino-3-oxopropyl)-13-benzyl-16-(4-hydroxybenzyl)-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carbonyl)-N-((R)-1-(2-amino-2-oxoethylamino)-5-guanidino-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
|
C46H64N14O12S2
|
1
|
| 1 |
EC50 = 0.03 nM
|
|
|
|
CP0909930
|
(S)-1-((3R,6S,9S,12S,15S)-6-(2-amino-2-oxoethyl)-15-(4-chlorobenzyl)-9-isopropyl-5,8,11,14,17-pentaoxo-12-(thiophen-2-ylmethyl)-1-thia-4,7,10,13,16-pentaazacycloicosane-3-carbonyl)-N-((R)-1-(diethylamino)-5-guanidino-1-oxopentan-2-yl)pyrrolidine-2-carboxamide
Show/Hide
|
C47H69ClN12O9S2
|
1
|
| 1 |
EC50 = 0.05 nM
|
|
|
|
CP0191782
|
1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]-3-methylbenzoyl)-2,3,4,5-tetrahydro-1H-1-benzazepine
Show/Hide
|
C26H25F2N3O2
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0507981
|
(4R)-4-Ethoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzyl-carbamoyl)-L-proline-N,N-dimethylamide
Show/Hide
|
C29H38N4O4
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0418952
|
(4R)-4-Hydroxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzylcarbamoyl)-L-proline-N,N-dimethylamide
Show/Hide
|
C27H34N4O4
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0510041
|
1-(4-[N-(2-dimethylamino-2-oxoethylcarbamoyl)aminomethyl]-3-methylbenzoyl)-2,3,4,5-tetrahydro-1H-1-benzazepine
Show/Hide
|
C24H30N4O3
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0401893
|
(4R)-4-Methoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzylcarbamoyl)-L-proline-N,N-dimethylamide
Show/Hide
|
C28H36N4O4
|
1
|
| 1 |
EC50 = 65 nM
|
|
|
|
CP0363124
|
1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzylcarbamoyl)-L-proline-N,N-dimethylamide
Show/Hide
|
C27H34N4O3
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0454321
|
(4R)-1-({4-[(2-chloro-5-fluorobenzene)amido]-3-methoxyphenyl}carbonyl)-1,2,3,5-tetrahydrospiro[1-benzazepine-4,1'-cyclopentan]-2'-ene-3'-carboxylic acid
Show/Hide
|
C30H26ClFN2O5
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
