Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
 Cell Line Info 
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT01608 , Adenosine receptor A2a
 Protein Info 
Gene Name ADORA2A
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P30543
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006
 Cell Line Info 
 Protein ID: PT01608
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0039348
 Compound Info 
(2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,4-dihydroxyoxolane-2-carboxamide
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C12H16N6O4
  1
1
Ki = 12 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0039632
 Compound Info 
(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-N-cyclopropyl-3,4-dihydroxyoxolane-2-carboxamide
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C13H16N6O4
  2
1
Ki = 12 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
2
Ki = 13.4 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0039042
 Compound Info 
N-[9-chloro-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]-2-phenylacetamide
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C21H14ClN5O2
  1
1
Ki = 52 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0217091
 Compound Info 
(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxy-N-methyloxolane-2-carboxamide
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C11H14N6O4
  1
1
Ki = 67 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0198142
 Compound Info 
(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxy-N-(2,2,2-trifluoroethyl)oxolane-2-carboxamide
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C12H13F3N6O4
  1
1
Ki = 405 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0435131
 Compound Info 
(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-N-(2-chloroethyl)-3,4-dihydroxyoxolane-2-carboxamide
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C12H15ClN6O4
  1
1
Ki = 410 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0362924
 Compound Info 
(2R,3R,4S,5R)-2-[6-[[(1R,2S,4S)-2-bicyclo[2.2.1]heptanyl]amino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol
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C17H23N5O4
  1
1
Ki = 477 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0198141
 Compound Info 
(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxy-N-propyloxolane-2-carboxamide
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C13H18N6O4
  1
1
Ki = 550 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0379088
 Compound Info 
(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-N-cyclopentyl-3,4-dihydroxyoxolane-2-carboxamide
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C15H20N6O4
  1
1
Ki = 610 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0259712
 Compound Info 
N-[4-(3,5-dimethylphenyl)-5-pyridin-4-yl-1,3-thiazol-2-yl]pyridine-3-carboxamide
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C22H18N4OS
  1
1
Ki = 1150 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS