| Compound ID |
Compound Name |
Compound Formula |
|
CP0049105
|
(SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2
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|
C63H98N18O13S
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0133180
|
((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl)-(2-methoxy-benzyl)-amine
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|
C28H32N2O
|
4
|
| 1 |
Kd = 5.37 nM
|
|
|
| 2 |
Kd = 16.6 nM
|
|
|
| 3 |
Ki = 0.3 nM
|
|
|
| 4 |
Ki = 0.4 nM
|
|
|
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CP0107813
|
3-[2-{1-[3,5-di(trifluoromethyl)phenyl]ethoxy}-3-(4-fluorophenyl)-1,4-oxazinan-4-ylmethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
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|
C23H21F7N4O3
|
3
|
| 1 |
Kd = 8.318 nM
|
|
|
| 2 |
Ki = 0.8 nM
|
|
|
| 3 |
Ki = 3 nM
|
|
|
|
CP0376848
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(2S)-2-(hydroxymethyl)-4-methylsulfonylpiperazin-1-yl]pyridin-3-yl]-N,2-dimethylpropanamide
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|
C31H33F7N4O4S
|
3
|
| 1 |
Kd = 16.98 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
| 3 |
Ki = 1.3 nM
|
|
|
|
CP0282991
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(2R,3S)-3-hydroxy-2-(hydroxymethyl)pyrrolidin-1-yl]pyridin-3-yl]-N,2-dimethylpropanamide
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|
C30H30F7N3O3
|
3
|
| 1 |
Kd = 28.84 nM
|
|
|
| 2 |
Ki = 0.7 nM
|
|
|
| 3 |
Ki = 1.1 nM
|
|
|
|
CP0381321
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]pyridin-3-yl]-N,2-dimethylpropanamide
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|
C30H30F7N3O2
|
3
|
| 1 |
Kd = 39.81 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
| 3 |
Ki = 2.8 nM
|
|
|
|
CP0410452
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(3S)-3-methyl-4-methylsulfonylpiperazin-1-yl]pyridin-3-yl]-N,2-dimethylpropanamide
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|
C31H33F7N4O3S
|
2
|
| 1 |
Ki = 0.3 nM
|
|
|
| 2 |
Ki = 0.5 nM
|
|
|
|
CP0376847
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-(4-methylsulfonylpiperazin-1-yl)pyridin-3-yl]-N,2-dimethylpropanamide
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|
C30H31F7N4O3S
|
2
|
| 1 |
Ki = 0.4 nM
|
|
|
| 2 |
Ki = 1.4 nM
|
|
|
|
CP0381342
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[4-(4-fluoro-2-methylphenyl)-6-[(3S)-3-hydroxypyrrolidin-1-yl]pyridin-3-yl]-N,2-dimethylpropanamide
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|
C29H28F7N3O2
|
2
|
| 1 |
Ki = 1.3 nM
|
|
|
| 2 |
Ki = 2.1 nM
|
|
|
|
CP0462726
|
2-[3,5-bis(trifluoromethyl)phenyl]-N-[6-(4,4-dioxo-1-oxa-4lambda6-thia-8-azaspiro[4.5]decan-8-yl)-4-(4-fluoro-2-methylphenyl)pyridin-3-yl]-N,2-dimethylpropanamide
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|
C32H32F7N3O4S
|
2
|
| 1 |
Ki = 1.4 nM
|
|
|
| 2 |
Ki = 1.7 nM
|
|
|
|
CP0397341
|
4-[4-(acetylmethyl-amino)-piperidin-1-yl]-N-(2-chloro-benzyl)-2-(3,4-dichlorophenyl)-2,N-dimethylbutyramide
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|
C27H34Cl3N3O2
|
1
|
| 1 |
Ki = 70.9 nM
|
|
|
|
CP0374063
|
4-[4-(acetylmethyl-amino)-piperidin-1-yl]-2-(3,4-dichlorophenyl)-N-(4-fluoro-3-trifluoromethylbenzyl)-2,N-dimethylbutyramide
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|
C28H33Cl2F4N3O2
|
1
|
| 1 |
Ki = 151.8 nM
|
|
|
|
CP0376631
|
2-(3,4-dichlorophenyl)-N-(4-fluoro-3-trifluoromethylbenzyl)-2,N-dimethyl-4-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-butyramide
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|
C29H33Cl2F4N3O2
|
1
|
| 1 |
Ki = 181.6 nM
|
|
|
|
CP0074738
|
(S)-(+)-N-((3-[1-Benzoyl-3-(3,4-dichlorophenyl)piperidin-3-yl]prop-1-yl)-4-phenylpiperidin-4-yl)-N-methylacetamine
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|
C35H41Cl2N3O2
|
1
|
| 1 |
Ki = 209.6 nM
|
|
|
|
CP0114970
|
(S)-(-)-N-(R-ethylbenzyl)-3-hydroxy-2-phenylquinoline-4-carboxamide
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|
C25H22N2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
