Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT01407 , Glutamate receptor 3
Gene Name GRIA3
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID P42263
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT01407
 
Compound ID Compound Name Compound Formula
CP0470950
N-[2-[4-(4-cyanophenyl)cyclohexyl]propyl]propane-2-sulfonamide
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C19H28N2O2S
 1
1
EC50 = 1660 nM
   TI
   LI
   LO
   TS
CP0374874
(+/-) Propane-2-sulfonic acid [2-(4'-cyano-biphenyl-4-yl)-propyl]-amide
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C19H22N2O2S
 1
1
EC50 = 1660 nM
   TI
   LI
   LO
   TS
CP0000104
3-Bicyclo[2.2.1]hept-5-en-2-yl-6-chloro-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[1,2,4]thiadiazine-7-sulfonic acid amide
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C14H16ClN3O4S2
 1
1
EC50 = 13700 nM
   TI
   LI
   LO
   TS
CP0008315
2,3-Dihydroxy-6-nitro-benzo[f]quinoxaline-7-sulfonic acid amide
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C12H8N4O6S
 1
1
IC50 = 1900 nM
   TI
   LI
   LO
   TS
CP0162369
2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid
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C14H10BrClN2O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0374730
4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid
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C18H13ClN2O3
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0204536
(2S,4R)-2-amino-4-[(E)-3-(4-chlorophenyl)prop-2-enyl]pentanedioic acid
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C14H16ClNO4
 1
1
Ki > 10000 nM
   TI
   LI
   LO
   TS