Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT01071 , Tyrosine-protein kinase ABL1
Gene Name ABL1
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID P00519
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT01071
 
Compound ID Compound Name Compound Formula
CP0367938
US10196378, Compound C03
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C28H27F3N6O2
 1
1
IC50 = 15.7 nM
   TI
   LI
   LO
   TS
CP0273432
US10196378, Compound C05
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C29H28F3N5O2
 1
1
IC50 = 38.3 nM
   TI
   LI
   LO
   TS
CP0574991
US10196378, Compound C08
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C31H27N7O2
 1
1
IC50 = 64.7 nM
   TI
   LI
   LO
   TS
CP0260268
1-(5-tert-butyl-2-quinolin-6-ylpyrazol-3-yl)-3-(4-quinolin-6-yloxyphenyl)urea
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C32H28N6O2
 1
1
IC50 = 345 nM
   TI
   LI
   LO
   TS
CP0495185
US10196378, Compound C06
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C29H28F3N5O2
 1
1
IC50 = 637 nM
   TI
   LI
   LO
   TS
CP0527925
US10196378, Compound C09
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C32H28N6O2
 1
1
IC50 = 719 nM
   TI
   LI
   LO
   TS
CP0113988
CEP-32496
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C24H22F3N5O5
 1
1
Kd = 3 nM
   TI
   LI
   LO
   TS