| Compound ID |
Compound Name |
Compound Formula |
|
CP0495243
|
[(2R,4S)-1-[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]-4-hydroxypyrrolidin-2-yl]boronic acid
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|
C10H22BN5O4
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
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CP0139059
|
(R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic acid
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|
C7H15BN2O3
|
1
|
| 1 |
IC50 = 0.46 nM
|
|
|
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CP0413285
|
[(2R,4R)-1-[(2S)-2-aminopropanoyl]-4-fluoropyrrolidin-2-yl]boronic acid
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|
C7H14BFN2O3
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0420944
|
[(2R,4S)-1-[(2S)-2-aminopropanoyl]-4-hydroxypyrrolidin-2-yl]boronic acid
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|
C7H15BN2O4
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0802309
|
(R)-3-amino-1-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-4-(2,4,5-trifluorophenyl)butan-1-one phosphate
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|
C16H18F6N5O5P
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0409555
|
[(2R,4S)-4-hydroxy-1-[(2S)-pyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
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|
C9H17BN2O4
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0409556
|
[(2R,4R)-4-hydroxy-1-[(2S)-pyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
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|
C9H17BN2O4
|
1
|
| 1 |
IC50 = 6.5 nM
|
|
|
|
CP0438946
|
[(2R,4S)-4-hydroxy-1-[(2S,4S)-4-hydroxypyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
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|
C9H17BN2O5
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0409558
|
[(2R,4R)-4-hydroxy-1-[(2S,4S)-4-hydroxypyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
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|
C9H17BN2O5
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0380844
|
(5S)-5-amino-6-[(2R,4R)-2-borono-4-hydroxypyrrolidin-1-yl]-6-oxohexanoic acid
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|
C10H19BN2O6
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0409553
|
(4S)-4-amino-5-[(2R,4R)-2-borono-4-hydroxypyrrolidin-1-yl]-5-oxopentanoic acid
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|
C9H17BN2O6
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0409557
|
[(2R,4S)-4-hydroxy-1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
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|
C9H17BN2O5
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0409137
|
[(2R,4R)-1-[(2S)-2-aminopropanoyl]-4-hydroxypyrrolidin-2-yl]boronic acid
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|
C7H15BN2O4
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0443589
|
(4S)-4-amino-5-[(2R,4S)-2-borono-4-hydroxypyrrolidin-1-yl]-5-oxopentanoic acid
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|
C9H17BN2O6
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0489152
|
(3R)-1-[(5aS,9aR)-1-pyridin-2-yl-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride
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|
C24H26ClF3N6O
|
1
|
| 1 |
IC50 = 43.4 nM
|
|
|
|
CP0439727
|
[(2R,4R)-4-hydroxy-1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]pyrrolidin-2-yl]boronic acid
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|
C9H17BN2O5
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0523239
|
(3R)-1-[(5aS,9aR)-1-(2-methyl-1,3-thiazol-4-yl)-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride
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|
C23H26ClF3N6OS
|
1
|
| 1 |
IC50 = 50.2 nM
|
|
|
|
CP0443588
|
[(2R,4S)-1-[(2S)-2-amino-3,3-dimethylbutanoyl]-4-hydroxypyrrolidin-2-yl]boronic acid
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|
C10H21BN2O4
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0481345
|
[(2R,4R)-1-[(2S)-2-amino-3,3-dimethylbutanoyl]-4-hydroxypyrrolidin-2-yl]boronic acid
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|
C10H21BN2O4
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0469676
|
(3R)-1-[(5aS,9aR)-1-pyrazin-2-yl-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride
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|
C23H25ClF3N7O
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0468792
|
(3R)-1-[(5aR,9aS)-1-(trifluoromethyl)-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one
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|
C20H21F6N5O
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0408197
|
(3R)-1-[(5aS,9aR)-1-benzyl-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride
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|
C26H29ClF3N5O
|
1
|
| 1 |
IC50 = 123.3 nM
|
|
|
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CP0411645
|
(3R)-1-[(5aS,9aR)-1-(6-ethoxypyridin-2-yl)-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride
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|
C26H30ClF3N6O2
|
1
|
| 1 |
IC50 = 139 nM
|
|
|
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CP0562634
|
(3R)-1-[(5aR,9aR)-1-(trifluoromethyl)-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one
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|
C20H21F6N5O
|
1
|
| 1 |
IC50 = 145 nM
|
|
|
|
CP0469677
|
(3R)-1-[(5aR,9aR)-1-propan-2-yl-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one;hydrochloride
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|
C22H29ClF3N5O
|
1
|
| 1 |
IC50 = 151.7 nM
|
|
|
|
CP0413289
|
[(2R)-1-[(2S)-2-aminopropanoyl]-4-oxopyrrolidin-2-yl]boronic acid
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|
C7H13BN2O4
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0558874
|
(3R)-1-[(5aS,9aS)-1-(trifluoromethyl)-5,5a,6,8,9,9a-hexahydro-4H-[1,2,4]triazolo[4,3-a][1,6]naphthyridin-7-yl]-3-amino-4-(2,4,5-trifluorophenyl)butan-1-one
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|
C20H21F6N5O
|
1
|
| 1 |
IC50 = 537 nM
|
|
|
|
CP0413290
|
[(2R,4S)-1-[(2S)-2-aminopropanoyl]-4-chloropyrrolidin-2-yl]boronic acid
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|
C7H14BClN2O3
|
1
|
| 1 |
IC50 = 18000 nM
|
|
|
