Compound ID |
Compound Name |
Compound Formula |
CP0579965
|
US10155731, Example 270
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|
C22H32N6O4
|
1
|
1 |
IC50 = 0.4 nM
|
|
|
CP0580055
|
methyl N-[3-[3-[(1R)-1-[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]ethyl]pyrrolo[2,3-b]pyridin-1-yl]propyl]carbamate
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|
C22H31N5O4
|
1
|
1 |
IC50 = 0.4 nM
|
|
|
CP0570268
|
methyl N-[3-[3-[[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]methyl]-6-methylpyrrolo[2,3-b]pyridin-1-yl]propyl]carbamate
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|
C22H31N5O4
|
1
|
1 |
IC50 = 0.8 nM
|
|
|
CP0579590
|
methyl N-[3-[3-[[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]methyl]indol-1-yl]propyl]carbamate
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|
C22H30N4O4
|
1
|
1 |
IC50 = 0.9 nM
|
|
|
CP0571665
|
methyl N-[3-[7-[(1R)-1-[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]ethyl]pyrrolo[2,3-b]pyrazin-5-yl]propyl]carbamate
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|
C21H30N6O4
|
1
|
1 |
IC50 = 1.7 nM
|
|
|
CP0576867
|
methyl N-[3-[3-[[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]methyl]pyrrolo[2,3-b]pyridin-1-yl]propyl]carbamate
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|
C21H29N5O4
|
1
|
1 |
IC50 = 3.1 nM
|
|
|
CP0580056
|
US10155731, Example 268
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|
C21H30N6O4
|
1
|
1 |
IC50 = 3.6 nM
|
|
|
CP0577007
|
US10155731, Example 271
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|
C22H32N6O4
|
1
|
1 |
IC50 = 3.7 nM
|
|
|
CP0577006
|
methyl N-[3-[3-[[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]methyl]-4-methylpyrrolo[2,3-b]pyridin-1-yl]propyl]carbamate
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|
C22H31N5O4
|
1
|
1 |
IC50 = 7.8 nM
|
|
|
CP0569514
|
US8975252, 39
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|
C21H29N3O3
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0570269
|
methyl N-[3-[3-[(1S)-1-[cyclopropyl-[(2R)-morpholine-2-carbonyl]amino]ethyl]pyrrolo[2,3-b]pyridin-1-yl]propyl]carbamate
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|
C22H31N5O4
|
1
|
1 |
IC50 = 84 nM
|
|
|
CP0578794
|
(2R)-N-cyclopropyl-N-[[1-(3-methoxypropyl)pyrrolo[2,3-b]pyridin-3-yl]methyl]morpholine-2-carboxamide
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|
C20H28N4O3
|
1
|
1 |
IC50 = 159 nM
|
|
|
CP0569913
|
(2R)-N-cyclopropyl-N-[[1-(3-methoxypropyl)pyrrolo[3,2-b]pyridin-3-yl]methyl]morpholine-2-carboxamide
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|
C20H28N4O3
|
1
|
1 |
IC50 = 453 nM
|
|
|
CP0576866
|
(2R)-N-cyclopropyl-N-[[1-(3-methoxypropyl)indazol-3-yl]methyl]morpholine-2-carboxamide
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|
C20H28N4O3
|
1
|
1 |
IC50 = 1076 nM
|
|
|
CP0570267
|
(2R)-N-cyclopropyl-N-[[1-(3-methoxypropyl)pyrrolo[2,3-c]pyridin-3-yl]methyl]morpholine-2-carboxamide
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|
C20H28N4O3
|
1
|
1 |
IC50 > 5000 nM
|
|
|
CP0578289
|
(2R)-N-cyclopropyl-N-[[1-(3-methoxypropyl)pyrrolo[3,2-c]pyridin-3-yl]methyl]morpholine-2-carboxamide
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|
C20H28N4O3
|
1
|
1 |
IC50 > 5000 nM
|
|
|