| Compound ID |
Compound Name |
Compound Formula |
|
CP0140154
|
3-(1-benzylpiperidin-4-yl)-2-[(8-hydroxyquinolin-2-yl)methyl-prop-2-ynylamino]propanenitrile
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|
C28H30N4O
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0065399
|
2-[[3-(1-benzylpiperidin-4-yl)propyl-prop-2-ynylamino]methyl]quinolin-8-ol
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|
C28H33N3O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0065400
|
2-(1-benzylpiperidin-4-yl)-2-[(8-hydroxyquinolin-2-yl)methyl-prop-2-ynylamino]acetonitrile
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|
C27H28N4O
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0065401
|
4-(1-benzylpiperidin-4-yl)-2-[(8-hydroxyquinolin-2-yl)methyl-prop-2-ynylamino]butanenitrile
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|
C29H32N4O
|
7
|
| 1 |
IC50 = 39 nM
|
|
|
| 2 |
Ki = 52 nM
|
|
|
| 3 |
Ki = 52.5 nM
|
|
|
| 4 |
Km = 249000 nM
|
|
|
| 5 |
Km = 289000 nM
|
|
|
| 6 |
Km = 456000 nM
|
|
|
| 7 |
Km = 1242000 nM
|
|
|
|
CP0072055
|
2-[[(1-benzylpiperidin-4-yl)methyl-prop-2-ynylamino]methyl]quinolin-8-ol
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|
C26H29N3O
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0072054
|
2-[[2-(1-benzylpiperidin-4-yl)ethyl-prop-2-ynylamino]methyl]quinolin-8-ol
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|
C27H31N3O
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0179369
|
4-(1-benzylpiperidin-4-yl)-2-[(8-hydroxyquinolin-5-yl)methyl-prop-2-ynylamino]butanenitrile
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|
C29H32N4O
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0673695
|
N-{[5-(3-(1-Benzylpiperidin-4-yl)propoxy)-1-methyl-1Hindol-2-yl]methyl}-N-methylprop-2-yn-1-amine
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|
C29H37N3O
|
1
|
| 1 |
IC50 = 3300 nM
|
|
|
|
CP0381947
|
N-methyl-N-[[1-methyl-5-[3-[1-[(2-methylphenyl)methyl]piperidin-4-yl]propoxy]indol-2-yl]methyl]prop-2-yn-1-amine
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|
C30H39N3O
|
1
|
| 1 |
IC50 = 4900 nM
|
|
|
|
CP0441704
|
[5-[[4-[3-[1-methyl-2-[[methyl(prop-2-ynyl)amino]methyl]indol-5-yl]oxypropyl]piperidin-1-yl]methyl]quinolin-8-yl] N,N-dimethylcarbamate
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|
C35H43N5O3
|
1
|
| 1 |
IC50 = 5900 nM
|
|
|
|
CP0400674
|
N-[[5-[3-(1-benzylpiperidin-4-yl)propoxy]-1H-indol-2-yl]methyl]-N-methylprop-2-yn-1-amine
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|
C28H35N3O
|
1
|
| 1 |
IC50 = 7100 nM
|
|
|
|
CP0381952
|
N-[[5-[3-(1-benzylpiperidin-4-yl)propoxy]-1H-indol-2-yl]methyl]prop-2-yn-1-amine
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|
C27H33N3O
|
1
|
| 1 |
IC50 = 7300 nM
|
|
|
|
CP0013001
|
(+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-indan-1-one
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|
C24H29NO3
|
2
|
| 1 |
IC50 = 7500 nM
|
|
|
| 2 |
IC50 = 8200 nM
|
|
|
|
CP0089596
|
Prochelators, 2
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|
C17H19N3O2
|
1
|
| 1 |
IC50 = 7900 nM
|
|
|
|
CP0441703
|
ethyl 5-[3-(1-benzylpiperidin-4-yl)propoxy]-1H-indole-2-carboxylate
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|
C26H32N2O3
|
1
|
| 1 |
IC50 = 9700 nM
|
|
|
|
CP0400673
|
[5-[3-(1-benzylpiperidin-4-yl)propoxy]-1H-indol-2-yl]methanol
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|
C24H30N2O2
|
1
|
| 1 |
IC50 = 31200 nM
|
|
|
|
CP0441705
|
N-[[5-[3-(1-benzylpiperidin-4-yl)propoxy]-1H-indol-2-yl]methyl]prop-2-en-1-amine
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|
C27H35N3O
|
1
|
| 1 |
IC50 = 40600 nM
|
|
|
